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1
المؤلفون: Claire E. Smith, Rossana Perciaccante, Peter R. Butchers, Alison J. Ford, Gillian Elizabeth Lunniss, Richard Conroy, Séverine Jeulin, Brian Edgar Looker, Graham Somers, Valerie S. Morrison, Amanda Emmons, Panayiotis A. Procopiou, Nicola Bevan, Victoria J. Barrett, Mark Ruston, Peter J. Mutch
المصدر: Bioorganic & Medicinal Chemistry. 19:4192-4201
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Hydantoin, Adrenergic, Uracil, Pharmacology, Biochemistry, In vitro, Bioavailability, Guinea pig, chemistry.chemical_compound, chemistry, In vivo, Drug Discovery, Microsome, Molecular Medicine, Molecular Biology
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2
المؤلفون: Peter R. Butchers, Claire E. Smith, Iain M. McLay, Rosemary Sasse, Keith Biggadike, Peter J. Mutch, Panayiotis A. Procopiou, Stephen A. Richards, Richard Conroy, Diane M. Coe, Edney Dean David, Stephen Barry Guntrip, Alison J. Ford, Rita Field, Brian Edgar Looker, Nicola Bevan, Michael John Monteith, Victoria J. Barrett, Valerie S. Morrison
المصدر: Journal of Medicinal Chemistry. 52:2280-2288
مصطلحات موضوعية: Models, Molecular, Agonist, Stereochemistry, medicine.drug_class, Guinea Pigs, Administration, Oral, Biological Availability, Bronchi, CHO Cells, In Vitro Techniques, Chemical synthesis, Guinea pig, Structure-Activity Relationship, Cricetulus, Dogs, In vivo, Oral administration, Cricetinae, Microsomes, Drug Discovery, Cyclic AMP, medicine, Animals, Humans, Structure–activity relationship, Albuterol, Adrenergic beta-2 Receptor Agonists, Salmeterol Xinafoate, chemistry.chemical_classification, 2-Hydroxyphenethylamine, Sulfonamides, Chemistry, Muscle, Smooth, Stereoisomerism, In vitro, Rats, Sulfonamide, Trachea, Molecular Medicine, Muscle Contraction
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3
المؤلفون: Peter R. Butchers, Nicola Bevan, Rick P. C. Cousins, Jill Coates, Valerie S. Morrison, David J. Wilson, M J Sheehan, Emma V. Edgar, Julian James GlaxoSmithKline Reeves
المصدر: European Journal of Pharmacology. 564:219-225
مصطلحات موضوعية: Agonist, Adenosine A2 Receptor Agonists, Receptor, Adenosine A2A, Neutrophils, medicine.drug_class, Stereochemistry, Adenosine A3 Receptor Antagonists, Tetrazoles, Adenosine A2A receptor, CHO Cells, Ligands, Receptor, Adenosine A2B, Radioligand Assay, Cricetulus, Genes, Reporter, Cricetinae, Cyclic AMP, medicine, Animals, Humans, Receptor, Pharmacology, Dose-Response Relationship, Drug, Receptor, Adenosine A1, Chemistry, Receptor, Adenosine A3, Adenosine A3 receptor, Receptor antagonist, Adenosine receptor, Adenosine A1 Receptor Agonists, Eosinophils, Purines, Competitive antagonist, Reactive Oxygen Species, Adenosine A2B receptor
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4
المؤلفون: Peter R. Butchers, Victoria J. Barrett, Peter J. Mutch, Andrew P. Craven, Sara C Hughes, Mark Ruston, Duncan S. Holmes, Alison J. Ford, Keith Biggadike, Brian Edgar Looker, Stephen Barry Guntrip, Anne Jones, Deborah Needham, Panayiotis A. Procopiou, Claire E. Smith
المصدر: Journal of medicinal chemistry. 57(1)
مصطلحات موضوعية: Agonist, Adrenergic receptor, medicine.drug_class, Guinea Pigs, CHO Cells, Pharmacology, Drug Administration Schedule, Sulfone, Hydroxylation, chemistry.chemical_compound, Cricetulus, Dogs, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Sulfones, Adrenergic beta-2 Receptor Agonists, respiratory system, Bioavailability, Rats, Trachea, chemistry, Toxicity, Hepatocytes, Molecular Medicine, Salmeterol, medicine.drug
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5
المؤلفون: Brian Edgar Looker, Peter R. Butchers, Peter J. Mutch, Iain Mcfarlane Mclay, Alison J. Ford, Duncan S. Holmes, Claire E. Smith, Philip Charles Box, Inderjit Singh Mann, Helen Tracey Horsley, Richard Conroy, Valerie S. Morrison, Fern Kerr, Nicola Bevan, Amanda Emmons, Victoria J. Barrett, Panayiotis A. Procopiou, Anne-Marie Li-Kwai-Cheung, Paula Tomlin, Diane Mary Coe, Keith Biggadike
المصدر: Journal of medicinal chemistry. 53(11)
مصطلحات موضوعية: Agonist, Models, Molecular, medicine.medical_specialty, medicine.drug_class, Protein Conformation, CHO Cells, Alkylation, Pharmacology, Chlorobenzenes, Guinea pig, Structure-Activity Relationship, Cricetulus, In vivo, Internal medicine, Cricetinae, Drug Discovery, medicine, Potency, Animals, Humans, Adrenergic beta-2 Receptor Agonists, Benzyl Alcohols, Chemistry, Chinese hamster ovary cell, Adrenergic beta-Agonists, In vitro, Bioavailability, Rats, Endocrinology, Molecular Medicine, Receptors, Adrenergic, beta-2, Benzyl Alcohol
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6
المؤلفون: Peter R. Butchers, R.A. Coleman, M. Johnson, Alison A. Humbles, C.J. Vardey, Douglas I. Ball, Anthony T. Nials
المصدر: European journal of pharmacology. 251(2-3)
مصطلحات موضوعية: Agonist, Male, medicine.medical_specialty, medicine.drug_class, Muscle Relaxation, Guinea Pigs, Bronchi, In Vitro Techniques, Dinoprost, immune system diseases, Bronchodilator, Internal medicine, Formoterol Fumarate, medicine, Animals, Humans, Albuterol, Mast Cells, Lung, Salmeterol Xinafoate, Cells, Cultured, Pharmacology, Bronchus, business.industry, Muscle, Smooth, respiratory system, Electric Stimulation, respiratory tract diseases, Bronchodilator Agents, Trachea, Endocrinology, medicine.anatomical_structure, Ethanolamines, Salbutamol, Bronchoconstriction, Salmeterol, Formoterol, medicine.symptom, business, hormones, hormone substitutes, and hormone antagonists, circulatory and respiratory physiology, medicine.drug