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1
المؤلفون: Natalia Diaz-Perez, Laura A. Volpicelli-Daley, Naomi Kamasawa, Nicolai T. Urban, Corinne Ida Lasmézas, Philip LoGrasso, Debbie Guerrero-Given, Minghai Zhou, Diego Grassi, Shannon Howard
المصدر: Proceedings of the National Academy of Sciences. 115
مصطلحات موضوعية: 0301 basic medicine, animal diseases, Neurotoxins, Cell Culture Techniques, Mitochondrion, environment and public health, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Mitophagy, Autophagy, Animals, Humans, Phosphorylation, Cells, Cultured, Brain Chemistry, Alpha-synuclein, Multidisciplinary, biology, Cytochrome c, Endoplasmic reticulum, Brain, Parkinson Disease, Mitochondria, nervous system diseases, Cell biology, Oxidative Stress, 030104 developmental biology, PNAS Plus, nervous system, chemistry, alpha-Synuclein, biology.protein, Unfolded protein response, Mitochondrial fission, Lysosomes, 030217 neurology & neurosurgery, Acetyl-CoA Carboxylase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e2214a423d9837eb003a7cddfa126049
https://doi.org/10.1073/pnas.1713849115 -
2
المؤلفون: Sarah Iqbal, Philip LoGrasso, Shannon Howard
المصدر: Molecular and Cellular Biology. 35:1992-2006
مصطلحات موضوعية: Male, MAP Kinase Kinase 4, Neurotoxins, Protein Serine-Threonine Kinases, Biology, Endoplasmic Reticulum, Immediate-Early Proteins, Glycogen Synthase Kinase 3, Mice, GSK-3, Cell Line, Tumor, Animals, Humans, ASK1, Oxidopamine, Protein kinase A, Molecular Biology, GSK3B, Glycogen Synthase Kinase 3 beta, Cell Death, urogenital system, Dopaminergic Neurons, c-jun, JNK Mitogen-Activated Protein Kinases, Neurodegenerative Diseases, Articles, Cell Biology, Endoplasmic Reticulum Stress, Protein kinase R, Molecular biology, Mitochondria, Cell biology, Mice, Inbred C57BL, Oxidative Stress, Neuroprotective Agents, 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine, SGK1, Signal transduction, Reactive Oxygen Species, Signal Transduction
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المؤلفون: Jun-Li Luo, Philip LoGrasso, Yuntao Wu, Yan Yin, Jia Guo, Nibal Eid, Chul Park, Ji-Hak Jeong, Ke Zheng, Yangbo Feng, Fei Yi, Pamela Hernandez, Mathieu Bibian, Weilin Wu, HaJeung Park, Shannon Howard
المصدر: Journal of Medicinal Chemistry. 58:1846-1861
مصطلحات موضوعية: Models, Molecular, Pharmacology, Article, Lim kinase, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, Animals, Humans, Urea, Structure–activity relationship, Potency, Protein Kinase Inhibitors, IC50, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Chemistry, Lim Kinases, In vitro, Rats, Biochemistry, Docking (molecular), Microsomes, Liver, Molecular Medicine
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4
المؤلفون: HaJeung Park, Sarah Iqbal, Pamela Hernandez, Ke Zheng, Yangbo Feng, Philip LoGrasso
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Membrane potential, Gene isoform, 0303 health sciences, 010405 organic chemistry, Chemistry, Kinase, Pharmacology, 01 natural sciences, Article, 3. Good health, 0104 chemical sciences, 03 medical and health sciences, Biochemistry, Pharmacokinetics, Drug Discovery, Molecular Medicine, Structure–activity relationship, Potency, Cytotoxicity, Drug metabolism, 030304 developmental biology
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المؤلفون: Shannon Howard, Su Gao, Philip LoGrasso
المصدر: Scientific Reports
مصطلحات موضوعية: 0301 basic medicine, Leptin, STAT3 Transcription Factor, medicine.medical_specialty, Hypothalamus, Diet, High-Fat, Article, 03 medical and health sciences, Eating, Mice, 0302 clinical medicine, Downregulation and upregulation, Mitogen-Activated Protein Kinase 10, Internal medicine, Weight Loss, medicine, Animals, Mitogen-Activated Protein Kinase 9, SOCS3, Obesity, Protein Kinase Inhibitors, Multidisciplinary, Kinase, Chemistry, c-jun, JNK Mitogen-Activated Protein Kinases, 030104 developmental biology, Endocrinology, Suppressor of Cytokine Signaling 3 Protein, Anorectic, Energy Metabolism, 030217 neurology & neurosurgery, Homeostasis, Signal Transduction
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المؤلفون: Theodore M. Kamenecka, Weimin Chen, Claudia Ruiz, Yuanjun He, Li Lin, Michael D. Cameron, Marcel Koenig, Philip LoGrasso, Yuan Yuan Ling, Derek R. Duckett
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:161-164
مصطلحات موضوعية: Stereochemistry, p38 mitogen-activated protein kinases, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Article, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Potency, Tissue Distribution, Isoxazole, Protein Kinase Inhibitors, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Kinase, Organic Chemistry, c-jun, JNK Mitogen-Activated Protein Kinases, Isoxazoles, Rats, Molecular Medicine, Selectivity
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المؤلفون: Yangbo Feng, Philip LoGrasso
المصدر: Expert Opinion on Therapeutic Patents. 24:295-307
مصطلحات موضوعية: Pharmacology, rho-Associated Kinases, Molecular Structure, General Medicine, Patent search, Biology, Legislation, Drug, Patents as Topic, Structure-Activity Relationship, Biochemistry, Drug Design, Expert opinion, Drug Discovery, Animals, Humans, Molecular Targeted Therapy, Protein Kinase Inhibitors, Rho-associated protein kinase, Signal Transduction
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المؤلفون: Marcel Koenig, Jeremy W. Chambers, HaJeung Park, Philip LoGrasso, Lisa Cherry, Sarah Iqbal, Pamela Hernandez, Yangbo Feng, Mariana Figuera-Losada
المصدر: ACS Chemical Biology. 8:1747-1754
مصطلحات موضوعية: Models, Molecular, Indazoles, MAP Kinase Kinase 4, Stereochemistry, Protein Serine-Threonine Kinases, Mitogen-activated protein kinase kinase, Biology, Leucine-Rich Repeat Serine-Threonine Protein Kinase-2, Biochemistry, Article, Cell Line, MAP2K7, Small Molecule Libraries, Inhibitory Concentration 50, Humans, Enzyme Inhibitors, Binding site, Benzofurans, MAPK14, Binding Sites, Protein-Serine-Threonine Kinases, MAP kinase kinase kinase, Kinase, General Medicine, Small molecule, nervous system diseases, Enzyme Activation, Molecular Probes, Molecular Medicine, Protein Binding
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المؤلفون: Philip LoGrasso, HaJeung Park, Pamela Hernandez, Valer Jeso, Glenn C. Micalizio, Michael D. Cameron, Sarah Iqbal
المصدر: Angewandte Chemie. 125:4900-4904
مصطلحات موضوعية: Stereochemistry, Cell Survival, Lactams, Macrocyclic, Stereoisomerism, Shikimic Acid, Crystallography, X-Ray, Catalysis, chemistry.chemical_compound, Polyketide, Macrocyclic Lactams, Benzoquinones, Humans, HSP90 Heat-Shock Proteins, Binding Sites, Membrane Glycoproteins, Chemistry, Ansamycin, General Chemistry, General Medicine, Shikimic acid, Benzoquinone, Protein Structure, Tertiary, Molecular Docking Simulation, Rifabutin, MCF-7 Cells, HeLa Cells
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المصدر: Journal of Biological Chemistry. 288:4000-4011
مصطلحات موضوعية: Programmed cell death, MAP Kinase Kinase 4, MAP Kinase Signaling System, Ischemia, Muscle Proteins, Myocardial Reperfusion Injury, Peptide, Mitochondrion, Biology, Pharmacology, Biochemistry, Mitochondria, Heart, Cell Line, Mitochondrial Proteins, Rats, Sprague-Dawley, In vivo, medicine, Animals, Creatine Kinase, MB Form, Humans, Myocytes, Cardiac, Creatine Kinase, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Reactive oxygen species, Cell Death, Cell Biology, medicine.disease, Molecular biology, Rats, Protein Transport, chemistry, Signal transduction, Reactive Oxygen Species, Reperfusion injury, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4fdf3216cef17f49c4be853483f57ff2
https://doi.org/10.1074/jbc.m112.406777