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المؤلفون: Eric Goffin, Pierre Fraikin, Dayana Abboud, Pascal de Tullio, Caroline Beaufour, Iuliana Botez, Julien Hanson, Laurence Danober, Pierre Francotte, Bernard Pirotte
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, General Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2dbce7893b489005fcc0c403b43869b6
https://doi.org/10.2139/ssrn.4329581 -
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المؤلفون: Daniel Tapken, Eric Goffin, Pierre Lestage, Bernard Pirotte, Laurence Danober, Pierre Fraikin, Jette S. Kastrup, Anja Probst Larsen, Pierre Francotte, Daniel-Henri Caignard, Karla Frydenvang
المصدر: ACS Chemical Neuroscience. 7:378-390
مصطلحات موضوعية: 0301 basic medicine, Physiology, Stereochemistry, Cognitive Neuroscience, Allosteric regulation, Substituent, AMPA receptor, Pharmacology, Benzothiadiazines, Crystallography, X-Ray, Receptors, Ionotropic Glutamate, Biochemistry, Structure-Activity Relationship, Xenopus laevis, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Animals, Structure–activity relationship, Receptors, AMPA, Glutamate receptor, Cell Biology, General Medicine, Potentiator, Rats, Electrophysiology, 030104 developmental biology, chemistry, Benzothiadiazine, Oocytes, 030217 neurology & neurosurgery, Ionotropic effect
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المؤلفون: Pascal De Tullio, Pierre Fraikin, Fabrice Iop, Ann-Beth Nørholm, Taru Deva, Karla Frydenvang, Jean-Yves Thomas, Lars Olsen, Sylvie Challal, Caroline Louis, Bernard Pirotte, Pierre Lestage, Pierre Francotte, Iuliana Botez-Pop, Laurence Danober, Jette S. Kastrup, Eric Goffin
المصدر: Journal of Medicinal Chemistry. 57:9539-9553
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, In vivo, Benzothiadiazine, Stereochemistry, Drug Discovery, Allosteric regulation, Molecular Medicine, Isothermal titration calorimetry, AMPA receptor, Potentiator, Receptor, Compound 32
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المؤلفون: P. Lestage, B. Lesur, L. Danober, P. de Tullio, Pierre Francotte, Iuliana Botez, Bernard Pirotte, Eric Goffin, Pierre Fraikin, Daniel-Henri Caignard
المصدر: Current Medicinal Chemistry. 17:3575-3582
مصطلحات موضوعية: Pharmacology, Thiadiazines, Organic Chemistry, Allosteric regulation, Glutamate receptor, Long-term potentiation, AMPA receptor, Biology, Potentiator, Biochemistry, Glutamatergic, Allosteric Regulation, nervous system, Drug Discovery, Humans, Molecular Medicine, Receptors, AMPA, Nervous System Diseases, Receptor, Neuroscience, Ionotropic effect
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2c92e8ae1e4c846c4fd6bd27d1f0ed0e
https://doi.org/10.2174/092986710792927859 -
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المؤلفون: Pascal De Tullio, Jean-Yves Thomas, Daniel-Henri Caignard, Tchao Podona, Bernard Pirotte, Laurence Danober, Pierre Francotte, Ousmane Diouf, Pierre Lestage, Pierre Fraikin
المصدر: Bioorganic & Medicinal Chemistry. 16:9948-9956
مصطلحات موضوعية: Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Intraperitoneal injection, Pharmaceutical Science, AMPA receptor, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Xenopus laevis, In vivo, Drug Discovery, medicine, Animals, Structure–activity relationship, Receptors, AMPA, Rats, Wistar, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Molecular Biology, Thiadiazines, Chemistry, Diazoxide, Organic Chemistry, Long-term potentiation, Potentiator, Rats, Solubility, Lipophilicity, Oocytes, Molecular Medicine
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المؤلفون: Pierre Fraikin, E. Graindorge, Pierre Francotte, Daniel-Henri Caignard, Pierre Lestage, Jean-Yves Thomas, Gaëlle Dintilhac, Bernard Pirotte, Laurence Danober, Pascal De Tullio, Eric Goffin
المصدر: Journal of Medicinal Chemistry. 50:3153-3157
مصطلحات موضوعية: Stereochemistry, Xenopus, Allosteric regulation, AMPA receptor, In Vitro Techniques, Pharmacology, Benzothiadiazines, Hippocampus, Chemical synthesis, Norepinephrine, Structure-Activity Relationship, chemistry.chemical_compound, Cognition, Allosteric Regulation, In vivo, Drug Discovery, Animals, Structure–activity relationship, RNA, Messenger, Receptors, AMPA, Rats, Wistar, Receptor, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Thiadiazines, Excitatory Postsynaptic Potentials, Recognition, Psychology, Potentiator, Electric Stimulation, Cyclic S-Oxides, Rats, chemistry, Benzothiadiazine, Drug Design, Oocytes, Molecular Medicine
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المؤلفون: Pierre, Francotte, Ann-Beth, Nørholm, Taru, Deva, Lars, Olsen, Karla, Frydenvang, Eric, Goffin, Pierre, Fraikin, Pascal, de Tullio, Sylvie, Challal, Jean-Yves, Thomas, Fabrice, Iop, Caroline, Louis, Iuliana, Botez-Pop, Pierre, Lestage, Laurence, Danober, Jette S, Kastrup, Bernard, Pirotte
المصدر: Journal of medicinal chemistry. 57(22)
مصطلحات موضوعية: Thiadiazines, Chemistry, Pharmaceutical, Temperature, Oxides, Calorimetry, Benzothiadiazines, Crystallography, X-Ray, Hippocampus, Cyclic S-Oxides, Rats, Electrophysiology, Kinetics, Mice, Drug Design, Animals, Humans, Thermodynamics, Receptors, AMPA, Propionates, Rats, Wistar, Dimerization, Allosteric Site, Hydrogen, Protein Binding
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المؤلفون: Olivier Nosjean, Pierre Fraikin, E. Graindorge, Pierre Francotte, Sylvie Challal, Eric Goffin, Pierre Lestage, Bernard Pirotte, Laurence Danober, Pascal De Tullio, Nathalie Rogez, Daniel-Henri Caignard
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Stereochemistry, Long-Term Potentiation, AMPA receptor, Thiophenes, Benzothiadiazines, Hippocampus, Membrane Potentials, chemistry.chemical_compound, Mice, Norepinephrine, Xenopus laevis, Cognition, Oral administration, In vivo, Drug Discovery, Excitatory Amino Acid Agonists, Animals, Receptors, AMPA, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Cells, Cultured, Molecular Structure, Thiadiazines, Chemistry, Diazoxide, Excitatory Postsynaptic Potentials, Long-term potentiation, Potentiator, Cyclic S-Oxides, Rats, Models, Chemical, Benzothiadiazine, Drug Design, Oocytes, Molecular Medicine, Female
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المؤلفون: Pierre Fraikin, Bernard Pirotte, Dominique Heymann, László G. Puskás, Thomas H. Lubben, Luca Munaron, C. Philippe, Susanna Antoniotti, Haim J. Wolfson, Zsolt Lo\\'rincz, Barbara Malawska, Antal Simay, C. Garcia-Echeverria, Péter Mátyus, Alessandra Fiorio Pla, Ruth Nussinov, Marcin Gruchala, Peter J. Scammells, Martin Eggert, Szilvia Vajda, Gurbir S. Bhatia, András Varró, Bruce G. Szczepankiewicz, Panagiotis Zoumpoulakis, Ildikó Varga, Mark S. Levi, Jerry Ryan Holder, Péter Krajcsi, Margaret A. Brimble, László Ürge, Thomas Mavromoustakos, Nastiti Wijayanti, William A. Banks, William H. Bunnelle, Zhonghua Pei, Krista R. Wilson, Paola Zaccone, David W. Dunne, O.M. Zack Howard, Tomozumi Imamichi, Gregory Y.H. Lip, Christine G. Joseph, Carrie Haskell-Luevano, Maria Zervou, R. Efremov, Ákos Kocsis, G.B. Mahady, Tingjun Hou, Marcel J. de Groot, David R. Davies, Thomas D.C. Thomas, Michael R. Schrimpf, Allen B. Reitz, Stewart B. Kirton, Boman G. Irani, Seppo Ylä-Herttuala, Xiaojie Xu, Zoltán Kovári, Uwe K. Zettl, Gang Liu, Andreas Klüter, Tivadar Rettegi, Rebecca Deprez-Poulain, Péter Kovács, László Károlyházy, Dimitra Hadjipavlou-Litina, Kuo-Chen Chou, Benoit Deprez, Ferenc Darvas, Mark Levis, Donald Small, M. Iqbal Choudhary, Thang K. Chiu, Julius Gy. Papp, Michael J. Dart, Pascal de Tullio, Atta-ur-Rahman, Andrzej Wilczynski, György Dormán, Himadri Roy, Russell C. Davis, C. Bor-Luen, Stephan Immenschuh, Michael D. Sosin, Alexandra Shulman-Peleg, Anne Cooke, Davide Lovisolo, Michael J. Sutcliffe, Dina Schneidman-Duhovny, Oranit Dror, Gunther Neeck, Aleksandar Todorovic, István Pénzes, Shalini Bhardwaj, Sally A. Hutchinson, P.R. Bernstein, Pierre Francotte, Cheryl P. Kordik, David A. Jans
المصدر: Frontiers in Medicinal Chemistry
مصطلحات موضوعية: Traditional medicine, Chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3f72de8108bc0fb8e384ae8a8f7537eb
https://doi.org/10.2174/97816080546401130601 -
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