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1
المؤلفون: Chunhui Huang, Christian Fischer, Michelle R. Machacek, Stephane Bogen, Tesfaye Biftu, Xianhai Huang, Michael H. Reutershan, Ryan Otte, Qingmei Hong, Zhicai Wu, Yang Yu, Min Park, Lei Chen, Purakkattle Biju, Ian Knemeyer, Ping Lu, Christopher J. Kochansky, Michael Brendan Hicks, Yong Liu, Roy Helmy, Xavier Fradera, Anthony Donofrio, Josh Close, Matthew L. Maddess, Catherine White, David L. Sloman, Nunzio Sciammetta, Jun Lu, Craig Gibeau, Vladimir Simov, Hongjun Zhang, Peter Fuller, David Witter
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::13ecfd534a4182e5c705a82b16c3ffcc
https://europepmc.org/articles/PMC9014435/ -
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المؤلفون: Craig C. Correll, Robert G. Aslanian, Li Xiao, Rema Bitar, Wei Zhou, John W. Butcher, Charles G. Garlisi, Joshua Close, Rachel N. Maccoss, Joon Jung, Scott Crawford, Kevin M. Maloney, Purakkattle Biju, Anandan Palani, Xianhai Huang, Xiaoxin Yang, Kevin D. McCormick, Scott Peterson, Hongjun Zhang, Diane Rindgen, Ying Huang, Alexei V. Buevich, Ning Shao, Li Dong, Phieng Siliphaivanh, Jason D. Brubaker, Michelle Martinez, Hongchen Qiu, François G. Gervais, Ravi P. Nargund, Zhidan Liu
المصدر: ACS Medicinal Chemistry Letters. 9:679-684
مصطلحات موضوعية: 0301 basic medicine, Drug, chemistry.chemical_classification, 010405 organic chemistry, Chemistry, medicine.drug_class, media_common.quotation_subject, Organic Chemistry, Pharmacology, medicine.disease, Receptor antagonist, 01 natural sciences, Biochemistry, 0104 chemical sciences, 03 medical and health sciences, 030104 developmental biology, Pharmacokinetics, Drug Discovery, medicine, Antagonism, Crth2 antagonist, Receptor, media_common, Asthma, Tricyclic
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3دورية أكاديمية
المؤلفون: Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, Ruiz, Manuel De, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
المصدر: In Bioorganic & Medicinal Chemistry Letters 15 February 2016 26(4):1348-1354
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4
المؤلفون: Purakkattle Biju, Yeon-Hee Lim, Kevin D. McCormick, Michael Berlin, Ying Wang, Rema Bitar, Robert G. Aslanian
المصدر: Tetrahedron Letters. 56:636-638
مصطلحات موضوعية: Ring-closing metathesis, Stereochemistry, medicine.drug_class, Chemistry, Organic Chemistry, Drug Discovery, medicine, Prednisolone, Biochemistry, Anti-inflammatory, medicine.drug
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5
المؤلفون: Rema Bitar, John C. Anthes, Jonathan E. Phillips, Purakkattle Biju, Robert G. Aslanian, Aileen House, Michael Berlin, Stephen Eckel, Daniel M. Solomon, George Kelly, Robbie L. McLeod, Richard Chapman, Xiomara Fernandez, Michelle Natiello, Daniel Prelusky, Kevin D. McCormick
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6343-6347
مصطلحات موضوعية: medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Cell Line, Steroid, Structure-Activity Relationship, Transactivation, chemistry.chemical_compound, Therapeutic index, Administration, Inhalation, Drug Discovery, medicine, Animals, Structure–activity relationship, Sulfhydryl Compounds, Lung, Molecular Biology, Transrepression, Chemistry, Organic Chemistry, Asthma, In vitro, Rats, Benzothiazole, Cell culture, Molecular Medicine, Steroids
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6
المؤلفون: X. Fernandez, Kevin D. McCormick, Johanna Jimenez, Hongwu Wang, Daniel Prelusky, Rema Bitar, Robert G. Aslanian, Yoon Joo Lee, Robbie L. McLeod, Gissela Lieber, Yanlin Jia, Richard Chapman, Steve Eckel, Michael Berlin, Purakkattle Biju, Yeon-Hee Lim, John C. Anthes, Jonathan E. Phillips, Aileen House
المصدر: Bioorganicmedicinal chemistry letters. 22(9)
مصطلحات موضوعية: Transcriptional Activation, Hydrocortisone, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrazole, Sulfides, Ring (chemistry), Biochemistry, Transactivation, chemistry.chemical_compound, Structure-Activity Relationship, Quinoxaline, Glucocorticoid receptor, Receptors, Glucocorticoid, Thioether, Drug Discovery, Structure–activity relationship, Humans, Molecular Biology, Transrepression, Organic Chemistry, chemistry, Molecular Medicine, Pyrazoles, Steroids
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7
المؤلفون: Jonathan E. Phillips, Yanlin Jia, Gissela Lieber, Daniel Prelusky, Rema Bitar, Stephen Eckel, George Kelly, Purakkattle Biju, Michael Berlin, Johanna Jimenez, Richard Chapman, John C. Anthes, Hongwu Wang, Robbie L. McLeod, Daniel M. Solomon, Aileen House, Yoon Joo Lee, X. Fernandez, Robert G. Aslanian, Kevin D. McCormick
المصدر: Bioorganicmedicinal chemistry letters. 22(2)
مصطلحات موضوعية: Functional assay, Benzimidazole, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, Sulfides, Biochemistry, Cell Line, chemistry.chemical_compound, Transactivation, Structure-Activity Relationship, Glucocorticoid receptor, Receptors, Glucocorticoid, Thioether, Rats, Inbred BN, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Transrepression, Tyrosine Transaminase, Dose-Response Relationship, Drug, Organic Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Stereoisomerism, Hep G2 Cells, Bioavailability, Rats, chemistry, Prednisolone, Molecular Medicine, medicine.drug
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8دورية أكاديمية
المؤلفون: Yu, Younong, Dwyer, Michael P., Chao, Jianping, Aki, Cynthia, Chao, Jianhua, Purakkattle, Biju, Rindgen, Diane, Bond, Richard, Mayer-Ezel, Rosemary, Jakway, James, Qiu, Hongchen, Hipkin, R. William, Fossetta, James, Gonsiorek, Waldemar, Bian, Hong, Fan, Xuedong, Terminelli, Carol, Fine, Jay, Lundell, Daniel, Merritt, J. Robert, He, Zhenmin, Lai, Gaifa, Wu, Minglang, Taveras, Arthur
المصدر: In Bioorganic & Medicinal Chemistry Letters 2008 18(4):1318-1322
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9دورية أكاديمية
المؤلفون: Chao, Jianhua, Taveras, Arthur G., Chao, Jianping, Aki, Cynthia, Dwyer, Michael, Yu, Younong, Purakkattle, Biju, Rindgen, Diane, Jakway, James, Hipkin, William, Fosetta, James, Fan, Xuedong, Lundell, Daniel, Fine, Jay, Minnicozzi, Michael, Phillips, Jonathan, Merritt, J. Robert
المصدر: In Bioorganic & Medicinal Chemistry Letters 2007 17(13):3778-3783
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10دورية أكاديمية
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