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1
المؤلفون: Anne-Françoise Aubry, Yunlin Fu, Mark E. Arnold, Duxi Zhang, Qianping Peng, Yuan-Qing Xia, Long Yuan
المصدر: Journal of Chromatography B. 969:60-68
مصطلحات موضوعية: Bioanalysis, Electrospray, Clinical Biochemistry, Tandem mass spectrometry, Sensitivity and Specificity, Biochemistry, High-performance liquid chromatography, Analytical Chemistry, Carboxylesterase, Drug Stability, Tandem Mass Spectrometry, Animals, Chromatography, High Pressure Liquid, Chromatography, Chemistry, Reproducibility of Results, Cell Biology, General Medicine, Rats, Phenylmethylsulfonyl Fluoride, Standard curve, Epothilones, Linear Models, Female, Sample collection, Esterase inhibitor, Carboxylic Ester Hydrolases
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2
المؤلفون: Zheng Ouyang, Qianping Peng, Long Yuan, Mark E. Arnold, Yuan-Qing Xia, Hao Jiang, Anne-Françoise Aubry, Jianing Zeng, Yuzhong Deng, Robert W. Lange
المصدر: Journal of Chromatography B. :81-86
مصطلحات موضوعية: Analyte, Electrospray, Clinical Biochemistry, Hepacivirus, Viral Nonstructural Proteins, Tandem mass spectrometry, Mass spectrometry, Antiviral Agents, Sensitivity and Specificity, Biochemistry, Analytical Chemistry, Mice, chemistry.chemical_compound, Dogs, Tandem Mass Spectrometry, Liquid chromatography–mass spectrometry, Animals, Protease Inhibitors, Sulfonamides, Chromatography, Chemistry, Extraction (chemistry), Haplorhini, Cell Biology, General Medicine, Isoquinolines, Hepatitis C, Rats, Standard curve, Asunaprevir, Rabbits, Chromatography, Liquid
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3
المؤلفون: Zheng Ouyang, Mark E. Arnold, Qianping Peng, Naiyu Zheng, Jianing Zeng, Adela Buzescu, Terry Van Vleet, Stephanie Pasas-Farmer, Mohammed Jemal
المصدر: Journal of Chromatography B. :64-74
مصطلحات موضوعية: Analyte, Bioanalysis, Indazoles, Sample (material), Clinical Biochemistry, Tandem mass spectrometry, Receptors, Corticotropin-Releasing Hormone, Sensitivity and Specificity, Biochemistry, Specimen Handling, Analytical Chemistry, Dogs, Calcitonin Gene-Related Peptide Receptor Antagonists, Tandem Mass Spectrometry, Animals, Humans, Sample preparation, Solid phase extraction, Quinazolinones, Reproducibility, Chromatography, Triazines, Chemistry, Elution, Solid Phase Extraction, Equipment Design, Haplorhini, Cell Biology, General Medicine, High-Throughput Screening Assays, Pyrazoles, Chromatography, Liquid
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4
المؤلفون: Jack L. Valentine, Robert W. Lange, Hao Jiang, Mark E. Arnold, Qianping Peng, Jianing Zeng, Hamza Kandoussi, Naiyu Zheng
المصدر: Analytical Chemistry. 83:6237-6244
مصطلحات موضوعية: Quality Control, Drug, Spectrometry, Mass, Electrospray Ionization, Analyte, Serial dilution, media_common.quotation_subject, Hepacivirus, Tandem mass spectrometry, Mass spectrometry, Antiviral Agents, Analytical Chemistry, Matrix (chemical analysis), Dogs, Tandem Mass Spectrometry, Liquid chromatography–mass spectrometry, Animals, Dog Diseases, media_common, Chromatography, Tissue Extracts, Chemistry, Reproducibility of Results, Hepatitis C, Dilution, Liver, Research Design, Calibration, Chromatography, Liquid
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5
المؤلفون: Palucki Brenda, Patrick G. Pollard, Liangqin Guo, Tung M. Fong, Matthew J. Wyvratt, Randy R. Miller, Shuwen He, Constantin Tamvakopoulos, Iyassu K. Sebhat, Qianping Peng, Ravi P. Nargund, Zhixiong Ye, Airu S. Chen, Doreen E. Cashen, David H. Weinberg, Min K. Park, Raman K. Bakshi, D. Euan MacIntyre, Howard Y. Chen, Rui Tang, Tanya MacNeil, Qingmei Hong, Alison M. Strack, Ralph A. Stearns, Jian Liu, William J. Martin
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2330-2334
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, Partial agonist, Piperazines, Rats, Sprague-Dawley, Eating, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Oral administration, In vivo, Drug Discovery, medicine, Animals, Urea, Obesity, Receptor, Molecular Biology, Organic Chemistry, Haplorhini, Rats, Disease Models, Animal, Piperazine, chemistry, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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6
المؤلفون: Yingjie Lai, Ralph A. Stearns, Qianping Peng, Ravi P. Nargund, Qingmei Hong, Jian Liu, Rui Tang, Matthew J. Wyvratt, Raman K. Bakshi, Randy R. Miller, Tianying Jian, Alison M. Strack, Tanya MacNeil, Liangqin Guo, Howard Y. Chen, James Dellureficio, Iyassu K. Sebhat, Peter H. Dobbelaar, Airu S. Chen, Constantin Tamvakopoulos, David H. Weinberg, Tung M. Fong, Christopher L. Franklin, Shuwen He, Zhixiong Ye
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4399-4405
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Pyrrolidines, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Anti-Obesity Agents, Internal medicine, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Spiro Compounds, Obesity, Molecular Biology, Mice, Knockout, Chemistry, Body Weight, Organic Chemistry, Amides, Rats, Endocrinology, Drug development, Anorectic, Receptor, Melanocortin, Type 4, Molecular Medicine
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7
المؤلفون: Howard Y. Chen, William J. Martin, D. Euan MacIntyre, Zhixiong Ye, Raman K. Bakshi, Alison M. Strack, Doreen E. Cashen, Jian Liu, Yingjie Lai, Tianying Jian, Constantin Tamvakopoulos, Nancy N. Tsou, Shuwen He, James Dellureficio, Tung M. Fong, Peter H. Dobbelaar, David H. Weinberg, Airu S. Chen, Qingmei Hong, Iyassu K. Sebhat, Tanya MacNeil, Christopher L. Franklin, Ravi P. Nargund, Ralph A. Stearns, Rui Tang, Richard G. Ball, Matthew J. Wyvratt, Randy R. Miller, Liangqin Guo, Qianping Peng
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2106-2110
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, Cricetulus, Dogs, Erectile Dysfunction, Cricetinae, Drug Discovery, medicine, Animals, Humans, Spiro Compounds, Receptor, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Haplorhini, Rats, Bioavailability, Indans, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding
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8
المؤلفون: Marc L. Reitman, Cheng Guo, Theresa M. Kelly, Constantin Tamvakopoulos, Joseph M. Metzger, Tianying Jian, Howard Y. Chen, Arthur A. Patchett, Oksana C. Palyha, Alison M. Strack, Allan J. Goodman, Ravi P. Nargund, Peter H. Dobbelaar, Yanqing Kan, Mark Hadden, Larry Yet, Peter R. Guzzo, Qianping Peng, Linus S. Lin, Shuwen He, Lauren P. Shearman, Alan J. Henderson, Carina P. Tan, Sargent Bruce J, Xiao-Ming Guan, Scott D. Feighner, Iyassu K. Sebhat, Jie Pan, Jian Liu, Donald J. Marsh, Matthew J. Wyvratt, Andrew D. Howard, Megan Ruenz
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1913-1917
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Molecular Biology, Biphenyl, Chemistry, Drug discovery, fungi, Organic Chemistry, Imidazoles, Rats, Bombesin receptor, Bioavailability, Receptors, Bombesin, Molecular Medicine, Bombesin Receptor Subtype-3
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9
المؤلفون: Heather L. Sings, Mark T. Goulet, Matthew J. Wyvratt, Iyassu K. Sebhat, Liangqin Guo, Rui Tang, Ravi P. Nargund, Qianping Peng, Euan Macintyre, Feroze Ujjainwalla, Constantin Tamvakopoulos, Zhixiong Ye, Lex H.T. Van der Ploeg, David H. Weinberg, Tanya MacNeil, John Huber
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:3242-3247
مصطلحات موضوعية: Agonist, Pyrrolidines, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, Melanocortin receptor, Drug Discovery, medicine, Humans, Structure–activity relationship, Receptor, Telomerase, Molecular Biology, G protein-coupled receptor, Molecular Structure, digestive, oral, and skin physiology, Organic Chemistry, Stereoisomerism, chemistry, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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10
المؤلفون: Doreen E. Cashen, Constantin Tamvakopoulos, Qianping Peng, William J. Martin, David H. Weinberg, Charles Rosenblum, Arthur A. Patchett, Tanya MacNeil, Patrick G. Pollard, Zhixiong Ye, Raman K. Bakshi, Ralph A. Stearns, Rubana N. Kalyani, Palucki Brenda, Joseph M. Metzger, Alison M. Strack, Lex H.T. Van der Ploeg, D. Euan MacIntyre, Iyassu K. Sebhat, Aurawan Vongs, Airu S. Chen, Ravi P. Nargund, Liangqin Guo, Matthew J. Wyvratt, Randy R. Miller, Rui Tang, Howard Y. Chen, Khaled J. Barakat
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3501-3505
مصطلحات موضوعية: Male, Agonist, Quinuclidines, Time Factors, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Rodentia, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Rats, Sprague-Dawley, Eating, Structure-Activity Relationship, Piperidines, In vivo, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Aza Compounds, Bicyclic molecule, Chemistry, Penile Erection, digestive, oral, and skin physiology, Organic Chemistry, Small molecule, Rats, Microsomes, Liver, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding