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1دورية أكاديمية
المؤلفون: Guohui Sun, Peiying Bai, Tengjiao Fan, Lijiao Zhao, Rugang Zhong, R. Stanley McElhinney, T. Brian H. McMurry, Dorothy J. Donnelly, Joan E. McCormick, Jane Kelly, Geoffrey P. Margison
المصدر: Pharmaceutics, Vol 15, Iss 8, p 2170 (2023)
مصطلحات موضوعية: MGMT, pseudosubstrates, inactivating agents, methyltransferase assay, MGMT activity determination, QSAR, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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2دورية أكاديمية
المصدر: ARKIVOC, Vol 2003, Iss 7, Pp 180-189 (2003)
مصطلحات موضوعية: Organic chemistry, QD241-441
وصف الملف: electronic resource
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المؤلفون: Sergio Lopez, Isabel Rozas, R. Stanley McElhinney, Geoffrey P. Margison, T. Brian H. McMurry, Alessandra Cordeiro
المصدر: Bioorganic & Medicinal Chemistry. 19:1658-1665
مصطلحات موضوعية: Methyltransferase, Molecular model, Stereochemistry, Chemistry, DNA repair, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, O-6-methylguanine-DNA methyltransferase, Biochemistry, DNA methyltransferase, Chemical synthesis, Enzyme Activation, Inhibitory Concentration 50, O(6)-Methylguanine-DNA Methyltransferase, chemistry.chemical_compound, Pyrimidines, Docking (molecular), Drug Discovery, Humans, Molecular Medicine, Computer Simulation, Enzyme Inhibitors, Molecular Biology, DNA
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المؤلفون: Nicola Glynn, R. Stanley McElhinney, Takayuki Shibata, Geoffrey P. Margison, T. Brian H. McMurry, David M. Williams
المصدر: Nucleic Acids Research
مصطلحات موضوعية: Guanine, Human dna, biology, O6-methylguanine, O-6-methylguanine-DNA methyltransferase, DNA methyltransferase, Molecular biology, Article, Proliferating cell nuclear antigen, O(6)-Methylguanine-DNA Methyltransferase, chemistry.chemical_compound, Organophosphorus Compounds, Oligodeoxyribonucleotides, chemistry, Biochemistry, Genetics, biology.protein, Humans, IC50, DNA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ee70bd67f3e0ed9ba0919a2417f35d88
https://doi.org/10.1093/nar/gkl117 -
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المؤلفون: Malcolm R Ranson, T. Brian H. McMurry, R. Stanley McElhinney, Martin J Dawson, Siow Ming Lee, Helen McGrath, J Bridgewater, L Gumbrell, Mark R Middleton, Geoffrey P. Margison, Dorothy Josephine Donnelly, Sue Waller, Debra Jowle, Gavin Halbert
المصدر: Clinical Cancer Research. 12:1577-1584
مصطلحات موضوعية: Adult, Male, Cancer Research, Guanine, Methyltransferase, Adolescent, Pharmacology, O(6)-Methylguanine-DNA Methyltransferase, Pharmacokinetics, Neoplasms, Antineoplastic Combined Chemotherapy Protocols, Temozolomide, medicine, Humans, Enzyme Inhibitors, Neoplasm Metastasis, Aged, Adenosine Triphosphatases, Dose-Response Relationship, Drug, biology, business.industry, Middle Aged, Dacarbazine, Regimen, Dose–response relationship, Oncology, Enzyme inhibitor, Pharmacodynamics, Toxicity, biology.protein, Female, Safety, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cde10c57e9db41a7dfa6b677c78520e0
https://doi.org/10.1158/1078-0432.ccr-05-2198 -
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المصدر: Synthesis. :983-988
مصطلحات موضوعية: NMR spectra database, chemistry.chemical_compound, Chemistry, Group (periodic table), Stereochemistry, Diamine, Organic Chemistry, Molecule, Protecting group, Medicinal chemistry, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b0ee12dffd2085b045607ccc7966d979
https://doi.org/10.1055/s-2006-926362 -
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المؤلفون: Vincent A. Barvaux, Malcolm Ranson, Robert Brown, R. Stanley McElhinney, T. Brian H. McMurry, Geoffrey P. Margison
المصدر: Molecular Cancer Therapeutics. 3:123-127
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::314e9f80823e8e3504e9f6164223aec6
https://doi.org/10.1158/1535-7163.123.3.2 -
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المصدر: Tetrahedron Letters. 50:6022-6024
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Electrophilic aromatic substitution, Biochemistry, Chloride, chemistry.chemical_compound, Group (periodic table), Drug Discovery, medicine, Nitro, Reactivity (chemistry), DNA, medicine.drug