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المصدر: Current Medicinal Chemistry. 27:1337-1349
مصطلحات موضوعية: Drug, media_common.quotation_subject, Drug Evaluation, Preclinical, Computational biology, drug testing, proteomics, transcriptomics, mass spectrometry, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, In vivo, Drug Discovery, Animals, Medicine, Drug Interactions, 030304 developmental biology, media_common, Pharmacology, 0303 health sciences, business.industry, Organic Chemistry, Computational Biology, Omics, Pre-clinical development, Drug development, 030220 oncology & carcinogenesis, Molecular Medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ced81a9d78d683b7870b0c0624cd7b99
https://doi.org/10.2174/0929867326666190711122819 -
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المؤلفون: Vlatka Bencetić Mihaljević, Andrea Fajdetić, Jasna Padovan, Domingo Gargallo-Viola, Amanda Mathis, Esperanza Herreros, Mihailo Banjanac, María Santos Martínez, Radan Spaventi, Albane Kessler, Iñigo Angulo-Barturen, Mihaela Perić, Vesna Eraković Haber, Vesna Munic Kos, Santiago Ferrer-Bazaga, Sulejman Alihodžić, María Belén Jiménez-Díaz, Dijana Pesic, Francisco-Javier Gamo, Mirjana Bukvić
المصدر: British journal of pharmacology. 178(2)
مصطلحات موضوعية: 0301 basic medicine, Plasmodium falciparum, Drug resistance, Azalide, Pharmacology, Azithromycin, antimalarial, azalide, in vivo efficacy, macrolide, malaria, mode of action, pharmacokinetics, 03 medical and health sciences, Antimalarials, Mice, 0302 clinical medicine, Dogs, In vivo, Chloroquine, medicine, Animals, Antimalarial Agent, Chloroquine / therapeutic use, Mode of action, Antimalarials* / pharmacology, biology, Chemistry, Chloroquine / pharmacology, biology.organism_classification, Malaria* / drug therapy, Malaria, Rats, 030104 developmental biology, Azithromycin / therapeutic use, Antimalarials* / therapeutic use, 030217 neurology & neurosurgery, Azithromycin / pharmacology, medicine.drug
وصف الملف: application/pdf
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المؤلفون: Vesna, Erakovic Haber, Radan, Spaventi
المصدر: Progress in molecular and subcellular biology. 55
مصطلحات موضوعية: Aquatic Organisms, Biological Products, Pharmaceutical Preparations, Chemistry, Pharmaceutical, Drug Design, Drug Evaluation, Preclinical, Combinatorial Chemistry Techniques, Technology, Pharmaceutical, High-Throughput Screening Assays
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::2100429cfc097d6a243a3abd40c70f25
https://pubmed.ncbi.nlm.nih.gov/28238036 -
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المؤلفون: Esperanza Herreros, Ana Toplak, Mihaela Perić, Dijana Pesic, Radan Spaventi, Kristina Starčević, J. Vidal, Dubravko Jelić, Sulejman Alihodžić, Maria Jesus Almela
المصدر: Journal of Medicinal Chemistry. 55:3216-3227
مصطلحات موضوعية: Stereochemistry, Plasmodium falciparum, Drug Resistance, Azalide, Gram-Positive Bacteria, Azithromycin, Antimalarials, Structure-Activity Relationship, chemistry.chemical_compound, Chloroquine, Cell Line, Tumor, Drug Discovery, medicine, Humans, malaria, antimalarial, azalide, quinoline, hybrid molecules, Aza Compounds, biology, Drug discovery, Quinoline, biology.organism_classification, Combinatorial chemistry, In vitro, Anti-Bacterial Agents, Erythromycin, chemistry, Quinolines, Molecular Medicine, Antibacterial activity, medicine.drug
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المؤلفون: Radan Spaventi, Santiago Ferrer, Sulejman Alihodžić, Goran Landek, Kristina Starčević, Esperanza Herreros, Ana Toplak, Dijana Pesic, Mihaela Perić
المصدر: European Journal of Medicinal Chemistry. 49:365-378
مصطلحات موضوعية: Plasmodium falciparum, Azithromycin, Pharmacology, Azalide, Cell Line, Antimalarials, Chloroquine, malaria, antimalarial, azalide, quinoline, hybrid molecules, synthesis, parasitic diseases, Drug Discovery, medicine, Humans, Antimalarial Agent, biology, Chemistry, Organic Chemistry, General Medicine, biology.organism_classification, medicine.disease, In vitro, Malaria, Aminoquinolines, Macrolides, Antibacterial activity, medicine.drug
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المؤلفون: Zrinka Ivezić Schoenfeld, Jasna Padovan, Sulejman Alihodžić, Samra Kapić, Adrijana Vinter, Ivana Palej Jakopović, Darko Filic, Radan Spaventi, Marina Modrić, Hana Čipčić Paljetak, Andrea Fajdetić, Vesna Eraković Haber, Roberto Antolović, Stjepan Mutak, Nada Košutić-Hulita
المصدر: European Journal of Medicinal Chemistry. 46:3388-3397
مصطلحات موضوعية: Male, Models, Molecular, medicine.drug_class, Stereochemistry, Carboxylic Acids, Administration, Oral, Biological Availability, Microbial Sensitivity Tests, Azithromycin, Crystallography, X-Ray, Chemical synthesis, Pneumococcal Infections, Drug Stability, Drug Discovery, medicine, Animals, Humans, Rats, Wistar, Antibacterial agent, Pharmacology, Chemistry, Organic Chemistry, Esters, Biological activity, General Medicine, Quinolone, Anti-Bacterial Agents, Rats, Bioavailability, Streptococcus pneumoniae, makrolide, resistance, antibacterial activity, pharmacokinetics, oral bioavailability, Injections, Intravenous, Microsomes, Liver, Macrolides, Efflux, Antibacterial activity, Isopropyl
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المؤلفون: Mihaela Perić, Wilbur K. Milhous, Nedjeljko Kujundžić, Jasna Padovan, Zrinka Ivezić Schönfeld, Andrea Fajdetić, Kirsten S. Smith, Dubravko Jelić, Colin Ohrt, Wolfgang Schönfeld, William Y. Ellis, Arba L. Ager, Radan Spaventi, Dinko Žiher, Mirjana Bukvić Krajačić, Goran Landek
المصدر: Journal of Medicinal Chemistry. 54:3595-3605
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Plasmodium falciparum, Azithromycin, Azalide, Ring (chemistry), Antimalarials, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Humans, Urea, Structure–activity relationship, Aromatic moiety, Chemistry, Thiourea, SAR, antimalarial acivity, urea, thiourea, azalides, In vitro, Models, Chemical, Drug Design, Lipophilicity, Molecular Medicine, Macrolides, medicine.drug
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المؤلفون: Krešimir Pavelić, Radan Spaventi, Mladen Jokić, Sanja Kapitanović, Tamara Čačev
المصدر: Journal of Cancer Research and Clinical Oncology. 132:200-204
مصطلحات موضوعية: Cancer Research, Loss of Heterozygosity, Single-nucleotide polymorphism, real-time PCR, SNP, E-cadherin, Biology, Polymorphism, Single Nucleotide, law.invention, Loss of heterozygosity, law, Polymorphism (computer science), Biomarkers, Tumor, Humans, Polymerase chain reaction, Genetics, Reverse Transcriptase Polymerase Chain Reaction, General Medicine, Cadherins, Molecular biology, Real-time polymerase chain reaction, Genetic Techniques, Oncology, Genetic marker, Colonic Neoplasms, Microsatellite Repeats, SNP array
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المؤلفون: Krešimir Pavelić, Sanja Kapitanović, Tamara Čačev, Radan Spaventi
المصدر: Journal of Molecular Medicine. 79:333-337
مصطلحات موضوعية: Electrophoresis, Male, Genes, APC, Adenomatous polyposis coli, APC gene, mutation detection, submerged gel electrophoresis, DNA Mutational Analysis, Gene mutation, Biology, medicine.disease_cause, Polymerase Chain Reaction, Familial adenomatous polyposis, law.invention, law, Drug Discovery, medicine, Humans, Genetic Testing, Polyacrylamide gel electrophoresis, Gene, Genetics (clinical), Polymerase chain reaction, Gel electrophoresis, Genetics, Mutation, medicine.disease, Molecular biology, Pedigree, Adenomatous Polyposis Coli, biology.protein, Molecular Medicine, Electrophoresis, Polyacrylamide Gel, Female, Polymorphism, Restriction Fragment Length
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المؤلفون: Duje Kovačević, Šime Spaventi, Sanja Kapitanović, Sanda Šturlan, Radan Spaventi, Krešimir Pavelić, Josip Lukač
المصدر: Journal of Molecular Medicine. 77:316-321
مصطلحات موضوعية: Deleted in Colorectal Cancer, Tumor suppressor gene, Colorectal cancer, Adenomatous Polyposis Coli Protein, Loss of Heterozygosity, Receptors, Cell Surface, Locus (genetics), Adenocarcinoma, Biology, Loss of heterozygosity, Tandem repeat, Colon cancer, Tumor suppressor genes, APC, DCC, Drug Discovery, medicine, Humans, Genes, Tumor Suppressor, Genetics (clinical), DNA Primers, Genetics, Tumor Suppressor Proteins, fungi, DCC Receptor, medicine.disease, Cytoskeletal Proteins, Tumor progression, Colonic Neoplasms, Cancer research, Molecular Medicine, Restriction fragment length polymorphism, Cell Adhesion Molecules, Polymorphism, Restriction Fragment Length, Microsatellite Repeats