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1دورية أكاديمية
المؤلفون: Lani S. Chun, Rakesh H. Vekariya, R. Benjamin Free, Yun Li, Da-Ting Lin, Ping Su, Fang Liu, Yoon Namkung, Stephane A. Laporte, Amy E. Moritz, Jeffrey Aubé, Kevin J. Frankowski, David R. Sibley
المصدر: Frontiers in Synaptic Neuroscience, Vol 10 (2018)
مصطلحات موضوعية: D2 dopamine receptor, functional selectivity, biased signaling, structure-activity relationship, MLS1547, quinoline, Neurosciences. Biological psychiatry. Neuropsychiatry, RC321-571
وصف الملف: electronic resource
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المؤلفون: Louis B. Nabors, James Mobley, Peter H. King, Michael R. Crowley, David K. Crossman, David Namkoong, Emily N. Hayward, Edward Ofori, Sixue Zhang, Rakesh H. Vekariya, Larry Bratton, Vibha Pathak, Jennifer Calano, Subramaniam Ananthan, Xiuhua Yang, Natalia Filippova
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::20d1d8f1d3bedc69b53f1a0309174161
https://doi.org/10.1158/0008-5472.22429090.v1 -
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المؤلفون: Louis B. Nabors, James Mobley, Peter H. King, Michael R. Crowley, David K. Crossman, David Namkoong, Emily N. Hayward, Edward Ofori, Sixue Zhang, Rakesh H. Vekariya, Larry Bratton, Vibha Pathak, Jennifer Calano, Subramaniam Ananthan, Xiuhua Yang, Natalia Filippova
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::15bb7da9799fd8f191594bce88cdcc84
https://doi.org/10.1158/0008-5472.22429084.v1 -
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المؤلفون: Jun Zhu, Pamela M. Quizon, Yingying Wang, Charles A. Adeniran, Matthew J. Strauss, Ana C. Jiménez-Torres, Palak Patel, Thomas J. Cirino, Shainnel O. Eans, Haylee R. Hammond, Laure S. Deliscar, Priscilla O'Hara, Surendra K. Saini, Edward Ofori, Rakesh H. Vekariya, Sixue Zhang, Omar Moukha-Chafiq, Theresa H. Nguyen, Subramaniam Ananthan, Corinne E. Augelli-Szafran, Chang-Guo Zhan, Jay P. McLaughlin
المصدر: Neuropharmacology. 220:109239
مصطلحات موضوعية: Pharmacology, Dopamine Plasma Membrane Transport Proteins, Dopamine, Mice, Transgenic, Cocaine-Related Disorders, Mice, Cellular and Molecular Neuroscience, Cricetulus, Cocaine, Reward, Cricetinae, Doxycycline, HIV-1, Trans-Activators, Animals, Humans, tat Gene Products, Human Immunodeficiency Virus, Transcription Factor DP1
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المؤلفون: Rakesh H. Vekariya, Subramaniam Ananthan, Wei Lei, John M. Streicher
المصدر: J Pain
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Anti-Inflammatory Agents, Receptors, Opioid, mu, Pharmacology, Article, Cell Line, δ-opioid receptor, Mice, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, 030202 anesthesiology, Naltrindole, Receptors, Opioid, delta, medicine, Animals, AIDS-Associated Nephropathy, Mice, Inbred ICR, Behavior, Animal, business.industry, Ovary, Chronic pain, medicine.disease, Analgesics, Opioid, Disease Models, Animal, Anesthesiology and Pain Medicine, Peripheral neuropathy, Neurology, Neuropathic pain, Morphine, Neuralgia, Female, Neurotoxicity Syndromes, Neurology (clinical), μ-opioid receptor, business, 030217 neurology & neurosurgery, medicine.drug
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6
المؤلفون: Rakesh H. Vekariya, Matthew C. Horton, Jeffrey Aubé, Feng Peng, Kevin Campos
المصدر: Organic Syntheses
مصطلحات موضوعية: chemistry.chemical_compound, 010405 organic chemistry, Chemistry, Intramolecular force, 010402 general chemistry, 01 natural sciences, Hexafluoro-2-propanol, Friedel–Crafts reaction, Medicinal chemistry, 0104 chemical sciences
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8f93f74b492ba2ee8158f63bf035acc1
https://doi.org/10.1002/0471264229.os095.32 -
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المؤلفون: Jennifer A. Calano, Xiuhua Yang, Peter H. King, Rakesh H. Vekariya, Sixue Zhang, David K. Crossman, Michael R. Crowley, Larry Bratton, James A. Mobley, Subramaniam Ananthan, Emily N. Hayward, Vibha Pathak, Edward Ofori, Natalia Filippova, Louis B. Nabors, David Namkoong
المصدر: Cancer Res
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Cell signaling, Carcinogenesis, Cell, Mice, Nude, Apoptosis, medicine.disease_cause, Deep sequencing, Article, ELAV-Like Protein 1, 03 medical and health sciences, Mice, Structure-Activity Relationship, 0302 clinical medicine, Downregulation and upregulation, Cell Line, Tumor, medicine, Animals, Humans, Precision Medicine, Tumor Stem Cell Assay, Cell Proliferation, Chemistry, Brain Neoplasms, RNA, Cell biology, Up-Regulation, 030104 developmental biology, medicine.anatomical_structure, Oncology, Cytoplasm, Blood-Brain Barrier, 030220 oncology & carcinogenesis, Cancer cell, Protein Multimerization, Glioblastoma, Algorithms, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a042e7e07dbe385617cd7874c523a0f7
https://pubmed.ncbi.nlm.nih.gov/33602784 -
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المؤلفون: John M. Streicher, Edward J. Bilsky, Gabriella Molnar, Subramaniam Ananthan, Kelly L. Karlage, Abhisek Ray, Rakesh H. Vekariya, Wei Lei, Karen L. Houseknecht, Deborah Barlow, Sixue Zhang, Tally M. Largent-Milnes, Surendra K. Saini
المصدر: J Med Chem
مصطلحات موضوعية: Agonist, Male, Morphinan, medicine.drug_class, Pyridines, Narcotic Antagonists, Receptors, Opioid, mu, CHO Cells, Pharmacology, 01 natural sciences, Article, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Cricetulus, Opioid receptor, In vivo, Receptors, Opioid, delta, mental disorders, Drug Discovery, medicine, Animals, Humans, 030304 developmental biology, 0303 health sciences, Molecular Structure, Chemistry, Antagonist, 0104 chemical sciences, Analgesics, Opioid, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Nociception, Opioid, Morphinans, Drug Design, Morphine, Microsomes, Liver, Molecular Medicine, medicine.drug, Protein Binding
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المؤلفون: Jeffrey Aubé, Rakesh H. Vekariya
المصدر: Organic Letters. 18:3534-3537
مصطلحات موضوعية: integumentary system, 010405 organic chemistry, Aryl, education, Organic Chemistry, Intermolecular force, 010402 general chemistry, behavioral disciplines and activities, 01 natural sciences, Biochemistry, Hexafluoro-2-propanol, 0104 chemical sciences, Acylation, chemistry.chemical_compound, chemistry, Yield (chemistry), Reagent, Organic chemistry, Physical and Theoretical Chemistry, Friedel–Crafts reaction, health care economics and organizations
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10
المؤلفون: Kelsey S. Hideshima, Diomedes E. Logothetis, Jose M. Eltit, Jason Younkin, Lia Baki, Amr Ellaithy, Supriya A Gaitonde, Javier González-Maeso, Malgorzata Dukat, José L. Moreno, Rakesh H. Vekariya, Sneha Shah, Richard A. Glennon, Peter Drossopoulos
المصدر: ACS Chemical Neuroscience. 7:1292-1299
مصطلحات موضوعية: 0301 basic medicine, Serotonin, Physiology, Stereochemistry, Cognitive Neuroscience, Voltage clamp, Tritium, 010402 general chemistry, 01 natural sciences, Biochemistry, Article, Calcium in biology, Membrane Potentials, Xenopus laevis, 03 medical and health sciences, chemistry.chemical_compound, medicine, Animals, Humans, Receptor, Serotonin, 5-HT2A, Receptor, 5-HT receptor, Risperidone, Benzisoxazole, Cell Biology, General Medicine, 0104 chemical sciences, HEK293 Cells, 030104 developmental biology, G Protein-Coupled Inwardly-Rectifying Potassium Channels, chemistry, Barium, Mutation, Oocytes, Serotonin 5-HT2 Receptor Antagonists, Calcium, Amine gas treating, Ketanserin, Serotonin Antagonists, Pharmacophore, Hydrophobic and Hydrophilic Interactions, Protein Binding, medicine.drug