-
1
المؤلفون: Randall R. Miller, Barbara A. Robinson
المصدر: Proceedings of the Water Environment Federation. 2012:1087-1099
مصطلحات موضوعية: Hydrology, Infiltration (hydrology), General Engineering, Inflow, Geology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::228aee309a45b5ab59b1e0b3fc90f528
https://doi.org/10.2175/193864712811741449 -
2
المؤلفون: George A. Doss, Lex H.T. Van der Ploeg, Qianping Peng, Ravi P. Nargund, Charles Rosenblum, Randall R. Miller, Aurawan Vongs, Palucki Brenda, Tanya MacNeil, Ralph A. Stearns, Min K. Park, David H. Weinberg, Rui Tang, Arthur A. Patchett, Constantin Tamvakopoulos
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1993-1996
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Receptor, Molecular Biology, biology, Chemistry, Organic Chemistry, biology.organism_classification, In vitro, Piperazine, Microsoma, Microsome, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
-
3
المؤلفون: William J. Martin, D. Euan MacIntyre, Ravi P. Nargund, Rubana N. Kalyani, Rui Tang, George A. Doss, Min K. Park, Alison M. Strack, Erin McGowan, Joseph M. Metzger, Charles Rosenblum, Randall R. Miller, Palucki Brenda, Qianping Peng, Arthur A. Patchett, Ralph A. Stearns, Patrick G. Pollard, Lex H.T. Van der Ploeg, Iyassu K. Sebhat, Constantin Tamvakopoulos, Cherrie Shepherd, Aurawan Vongs, Tanya MacNeil, David H. Weinberg, Zhixiong Ye
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:171-175
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Mice, Dogs, Erectile Dysfunction, Piperidines, In vivo, Drug Discovery, medicine, Animals, Obesity, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Haplorhini, In vitro, Rats, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
-
4
المؤلفون: George A. Doss, Randall R. Miller, Ralph A. Stearns
المصدر: Drug Metabolism and Disposition. 32:178-185
مصطلحات موضوعية: Male, Magnetic Resonance Spectroscopy, Swine, Hydrochloride, Stereochemistry, Metabolite, Administration, Oral, Pharmaceutical Science, In Vitro Techniques, Hydroxylamines, Mass Spectrometry, Piperazines, chemistry.chemical_compound, Glucuronides, Hydroxylamine, Species Specificity, Animals, Hypoglycemic Agents, Chromatography, High Pressure Liquid, Pharmacology, Glucuronic acid, Macaca mulatta, Piperazine, chemistry, Microsomes, Liver, Microsome, Glucuronide, Chromatography, Liquid, Conjugate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6f35d3b9ef842fd823e9107888add6bf
https://doi.org/10.1124/dmd.32.2.178 -
5
المؤلفون: Thomas A. Baillie, Wei Tang, Robert J. Mathvink, Carol Ann Keohane, Ralph A. Stearns, Randall R. Miller, Gloria Y. Kwei, George A. Doss, Ann E. Weber, Shuet Hing L Chiu, John R. Strauss, Jason S. Ngui
المصدر: Drug Metabolism and Disposition. 30:778-787
مصطلحات موضوعية: Male, Agonist, Taurine, Swine, medicine.drug_class, Metabolite, Carboxylic acid, Isethionic Acid, Pharmaceutical Science, Adrenergic beta-3 Receptor Agonists, Pharmacology, Cell Line, Rats, Sprague-Dawley, Mice, chemistry.chemical_compound, Dogs, medicine, Animals, Humans, chemistry.chemical_classification, Sulfonamides, CYP3A4, Chemistry, Isethionic acid, Metabolism, Macaca mulatta, Rats, Amino acid, Thiazoles, Biochemistry, Receptors, Adrenergic, beta-3, Microsomes, Liver, Female, Oxidation-Reduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::92f5c62aea74eaaf1cc50986422f421f
https://doi.org/10.1124/dmd.30.7.778 -
6
المؤلفون: Patricia Brown, Anthony Sanfiz, Ann E. Weber, Richard A. Berger, Liping Wang, Katherine L. Villa, Scott D. Edmondson, Christopher Moyes, Amanda L. Hurley, Andra S. Stevenson, Aileen Fitzmaurice, Dong-Ming Shen, Stephen D. Goble, Nina Jochnowitz, Karen H. Dingley, Jerry Di Salvo, Mary Struthers, Loise Gichuru, Randall R. Miller, Hiroshi Nagabukuro, Gino Salituro, Airu S. Chen, Beata Zamlynny, Alka Bansal, Bart Harper, Shruty Mistry
المصدر: Journal of medicinal chemistry. 57(4)
مصطلحات موضوعية: medicine.medical_specialty, AS-19, Magnetic Resonance Spectroscopy, Molecular Conformation, Adrenergic beta-3 Receptor Agonists, CHO Cells, chemistry.chemical_compound, Cricetulus, Internal medicine, Cricetinae, Drug Discovery, medicine, Potency, Animals, Humans, Receptor, Thiazole, Acetanilide, Urinary bladder, biology, Urinary Bladder, Overactive, medicine.disease, biology.organism_classification, medicine.anatomical_structure, Endocrinology, Overactive bladder, chemistry, Drug Design, Molecular Medicine, Acetanilides
-
7
المؤلفون: Ann E. Weber, Thomas L. Shih, Michael J. Forrest, Randall R. Miller, Michael H. Fisher, Matthew J. Wyvratt, Catherine D. Strader, Margaret A. Cascieri, Liping Deng, Ralph A. Stearns, D. Euan MacIntyre, William P. Feeney, Mari R. Candelore, Gary J Hom, Lawrence F. Colwell, Laurie Tota, Shuet-Hing Lee Chiu
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:1251-1254
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Biological Availability, Tetrazoles, Pharmaceutical Science, Pharmacology, Biochemistry, Inhibitory Concentration 50, Dogs, Pharmacokinetics, In vivo, Oral administration, Drug Discovery, medicine, Animals, Humans, Molecular Biology, ED50, Sulfonamides, Chemistry, Organic Chemistry, Biological activity, Adrenergic beta-Agonists, In vitro, Rats, Bioavailability, Kinetics, Molecular Medicine
-
8
المؤلفون: Matthew J. Wyvratt, Leroy Perkins, Randall R. Miller, Ann E. Weber, William P. Feeney, Vincent J. Colandrea, Michael J. Forrest, Emma R. Parmee, Laurie Tota, Michael H. Fisher, Mari R. Candelore, Gary J Hom, Hyun O. Ok, Elizabeth M. Naylor, Catherine D. Strader, Margaret A. Cascieri, Ralph A. Stearns, Liping Deng, D. Euan MacIntyre
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:749-754
مصطلحات موضوعية: Agonist, Beta-3 adrenergic receptor, medicine.medical_specialty, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Adrenergic, Biochemistry, Partial agonist, Structure-Activity Relationship, Dogs, Heart Rate, In vivo, Internal medicine, Receptors, Adrenergic, beta, Drug Discovery, medicine, Animals, Humans, Urea, Lipolysis, Receptor, Adrenergic beta-2 Receptor Agonists, Molecular Biology, ED50, Sulfonamides, Chemistry, Organic Chemistry, Adrenergic beta-Agonists, Macaca mulatta, Endocrinology, Adrenergic beta-1 Receptor Agonists, Receptors, Adrenergic, beta-3, Molecular Medicine
-
9
المصدر: The Journal of Antibiotics. 50:418-423
مصطلحات موضوعية: Antifungal Agents, Stereochemistry, Metabolite, Mutant, Microbial Sensitivity Tests, Streptomyces, Tacrolimus, Mice, chemistry.chemical_compound, Drug Discovery, polycyclic compounds, Animals, Chromatography, High Pressure Liquid, Pharmacology, biology, Streptomycetaceae, Biological activity, biology.organism_classification, In vitro, Mice, Inbred C57BL, Biochemistry, chemistry, Fermentation, Aspergillus niger, Actinomycetales, Genetic Engineering, Immunosuppressive Agents, Bacteria
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f3bfbb6dddd05467c266d2208b6dd8ba
https://doi.org/10.7164/antibiotics.50.418 -
10
المؤلفون: Sheng-Jian Cai, Randall R. Miller, Haideh Motamedi, Ali Shafiee, S L Streicher, Byron H. Arison
المصدر: Journal of Bacteriology. 178:5243-5248
مصطلحات موضوعية: DNA, Bacterial, Streptomyces tsukubaensis, Molecular Sequence Data, Mutant, Microbiology, Streptomyces, Tacrolimus, Mixed Function Oxygenases, Gene product, Bacterial Proteins, Cytochrome P-450 Enzyme System, polycyclic compounds, Amino Acid Sequence, Molecular Biology, Gene, Base Sequence, Sequence Homology, Amino Acid, biology, Methyltransferases, biology.organism_classification, Molecular biology, Open reading frame, Biochemistry, Genes, Bacterial, Heterologous expression, Streptomyces hygroscopicus, Immunosuppressive Agents, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0bbceb5319819ef1bd63adb6a7dc5d26
https://doi.org/10.1128/jb.178.17.5243-5248.1996