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1
المؤلفون: Katarina, Zmajkovicova, Sumit, Pawar, Sabine, Maier-Munsa, Barbara, Maierhofer, Ivana, Wiest, Renato, Skerlj, Arthur G, Taveras, Adriana, Badarau
المصدر: Genes and immunity. 23(6)
مصطلحات موضوعية: Receptors, CXCR4, Neutropenia, Primary Immunodeficiency Diseases, Immunologic Deficiency Syndromes, Butylamines, Immunoglobulin A, Agammaglobulinemia, Aminoquinolines, Humans, Benzimidazoles, Warts, Proto-Oncogene Proteins c-akt, Biomarkers, Genetic Association Studies
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2
المؤلفون: Frank C Firkin, David C. Dale, Weihua Tang, Sarah L. Cohen, Audrey Anna Bolyard, Varun Garg, Kenneth J. Gorelick, Vahagn Makaryan, Honghua Jiang, Merideth L. Kelley, Tarek M Ebrahim, Renato Skerlj
المصدر: Blood. 136(26)
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Receptors, CXCR4, Adolescent, Neutrophils, Primary Immunodeficiency Diseases, Immunology, Administration, Oral, Butylamines, Biochemistry, CXCR4, Gastroenterology, Hypogammaglobulinemia, Leukocyte Count, Internal medicine, medicine, Humans, Prospective Studies, Adverse effect, Myelokathexis, business.industry, Cell Biology, Hematology, Middle Aged, medicine.disease, Tolerability, Pharmacodynamics, Absolute neutrophil count, Aminoquinolines, Benzimidazoles, Female, Warts, business, WHIM syndrome
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ddc7fa05a51a626a3064127bd0ece88a
https://pubmed.ncbi.nlm.nih.gov/33367549 -
3
المصدر: ACS Medicinal Chemistry Letters. 8:22-26
مصطلحات موضوعية: 0301 basic medicine, Chemistry, Stereochemistry, Organic Chemistry, Biochemistry, Protein–protein interaction, 03 medical and health sciences, 030104 developmental biology, Membrane, Nucleophile, Covalent bond, Drug Discovery, Electrophile, Helix, Peptide bond, Cysteine
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4
المؤلفون: Leo A. Paquette, John L. King, Renato Skerlj, Satomi Niwayama, Dean R. Lagerwall
المصدر: Tetrahedron Letters. 60:151179
مصطلحات موضوعية: chemistry.chemical_compound, Dodecahedron, Direct entry, Computational chemistry, Chemistry, Organic Chemistry, Drug Discovery, Electrophile, Tetrahedron, Biochemistry, Derivative (chemistry)
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5
المؤلفون: Stephen G. Davies, Renato Skerlj, Mark Whittaker
مصطلحات موضوعية: Inorganic Chemistry, Reduction (complexity), Chemistry, Organic Chemistry, Chemical reduction, Organic chemistry, Stereoselectivity, Physical and Theoretical Chemistry, Enantiomeric excess, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::87f2c8d91149063d7c6285fb98bf85fb
https://ora.ox.ac.uk/objects/uuid:af0a2547-e691-480e-916a-c354e84fc536 -
6
المؤلفون: Dana Huskens, Marilyn C. Darkes, Gary Bridger, Jennifer H. Cox, Simon P. Fricker, Zefferino Santucci, Renee Mosi, Jean Labrecque, Kim L. Nelson, Renato Skerlj, Stefan R. Idzan, Virginia Anastassova, Dominique Schols, Ketan Patel, Rebecca S.Y. Wong, Gloria Lau
المصدر: Biochemical Pharmacology. 83:472-479
مصطلحات موضوعية: CCR1, Receptors, CXCR4, Anti-HIV Agents, Allosteric regulation, Administration, Oral, Biological Availability, C-C chemokine receptor type 7, Pharmacology, Biology, Butylamines, Virus Replication, CXCR3, Biochemistry, Cell Line, Heterocyclic Compounds, 1-Ring, Dogs, Calcium flux, medicine, Animals, Humans, Receptor, Molecular Structure, Ligand binding assay, Virus Internalization, Chemokine CXCL12, Entry inhibitor, Gene Expression Regulation, Aminoquinolines, HIV-1, Benzimidazoles, Protein Binding, Signal Transduction, medicine.drug
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7
المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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8
المؤلفون: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Ernest McEachern, Jonathan Langille, Curtis Harwig, Duane Veale, Wen Yang, Tongshong Li, Yongbao Zhu, Michael Bey, Ian Baird, Michael Sartori, Markus Metz, Renee Mosi, Kim Nelson, Veronique Bodart, Rebecca Wong, Simon Fricker, Ron Mac Farland, Dana Huskens, Dominique Schols
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6950-6954
مصطلحات موضوعية: Tertiary amine, Anti-HIV Agents, Pyridines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CCR5 receptor antagonist, Pharmacology, Virus Replication, Biochemistry, Peripheral blood mononuclear cell, Chemical synthesis, Inhibitory Concentration 50, Dogs, Piperidines, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, virus diseases, Amides, In vitro, Rats, Viral replication, Drug Design, CCR5 Receptor Antagonists, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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9
المؤلفون: Ling Qin, Renato Skerlj, Yongbao Zhu, Zefferino Santucci, Renee Mosi, Jennifer H. Cox, Simon P. Fricker, Virginia Anastassov, Beth R. Cameron, Markus Metz
المصدر: Journal of Inorganic Biochemistry. 105:754-762
مصطلحات موضوعية: Male, Cathepsin, Chemistry, Stereochemistry, Cathepsin K, Antineoplastic Agents, Biological activity, Mice, SCID, Cysteine Proteinase Inhibitors, Biochemistry, Cysteine protease, Cathepsin B, Inorganic Chemistry, Mice, Cathepsin O, Cysteine Proteases, Cell Line, Tumor, Animals, Humans, Gold, Cysteine
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10
المؤلفون: Tong-Shuang Li, Simon P. Fricker, Gang Chen, Renato Skerlj, David Bogucki, Markus Metz, Gary Bridger, Susan Nan, Rebecca S.Y. Wong, Dominique Schols, Jean Labrecque, Gloria Lau, Marilyn C. Darkes, Bryon Carpenter
المصدر: Virology. 413(2):231-243
مصطلحات موضوعية: Models, Molecular, Receptors, CCR5, Protein Conformation, Vicriviroc, viruses, Aplaviroc, Drug design, CCR5 receptor antagonist, Computational biology, Biology, Maraviroc, chemistry.chemical_compound, HIV Fusion Inhibitors, Virology, High-Throughput Screening Assays, medicine, Homology modeling, Binding site characterization, virus diseases, Reproducibility of Results, Stereoisomerism, Virus Internalization, Molecular biology, Small molecule, Small molecule antagonists, Antifusogenic assay, chemistry, Mutagenesis, CCR5 Receptor Antagonists, Mutation, HIV-1, Mutagenesis, Site-Directed, CCR5, medicine.drug