-
1
المؤلفون: Robert L. Hudkins, Joanne R. Mathiasen, Reddeppa reddy Dandu, Lisa D. Aimone, Rita Raddatz, Val R. Marcy, Greg A. Hostetler, John A. Gruner, Caitlyn Benfield, Robert J. Bendesky
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6362-6365
مصطلحات موضوعية: Phenethylamine, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Molecular Biology, Electromyography, Organic Chemistry, Electroencephalography, Metabolic stability, Rats, Bioavailability, chemistry, Molecular Medicine, Histamine H3 receptor, Selectivity, Histamine H3 Antagonists
-
2
المؤلفون: Kurt A. Josef, Allison L. Zulli, Lisa D. Aimone, Derek Dunn, Rita Raddatz, Jacquelyn A. Lyons, Ming Tao, Joanne R. Mathiasen, Reddeppa reddy Dandu, Thomas R. Bailey, Val R. Marcy, Babu G. Sundar, John A. Gruner, Edward R. Bacon, Robert L. Hudkins, Robert J. Bendesky, Yin-Guo Lin
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5493-5497
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Histamine h, Biochemistry, In vivo, Drug Discovery, Molecular Medicine, Inverse agonist, Potency, Selectivity, Antagonism, Receptor, Molecular Biology, Linker
-
3
المؤلفون: Robert J. Bendesky, Wai C. Wong, Theodore P. Broten, Fengqi Zhang, Dake Tian, Carlos Forray, James Fang, Sriram Tyagarajan, Dhanapalan Nagarathnam, and Kamlesh P. Vyas, Shou Wu Miao, George Chiu, Mohammad R. Marzabadi, T. G. Murali Dhar, Charles Gluchowski, Kathryn Schneck, Paul J. Kling, Raymond S.L. Chang, Bharat Lagu, Jack Zhang, Wanying Sun, Stacey O'Malley, Tsing B. Chen, Richard W. Ransom, Terry W. Schorn, Charles M. Harrell, John M. Wetzel
المصدر: Journal of Medicinal Chemistry. 42:4764-4777
مصطلحات موضوعية: Male, medicine.drug_class, Drug Evaluation, Preclinical, Nitro compound, Blood Pressure, Carboxamide, Pyrimidinones, In Vitro Techniques, Pharmacology, Binding, Competitive, Chemical synthesis, Rats, Sprague-Dawley, Radioligand Assay, Dogs, Urethra, In vivo, Receptors, Adrenergic, alpha-1, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Receptor, Adrenergic alpha-Antagonists, chemistry.chemical_classification, Prostate, Antagonist, Stereoisomerism, In vitro, Rats, chemistry, Biochemistry, Drug Design, Adrenergic alpha-1 Receptor Antagonists, Molecular Medicine
-
4
المؤلفون: Tsing-B. Chen, Kristie A. Faust, Elizabeth M. Naylor, Bradley V. Clineschmidt, Prasun K. Chakravarty, Victor J. Lotti, Robert J. Bendesky, Stacey A. O'Malley, Paul J. Kling, Raymond S.L. Chang, Arthur A. Patchett, William J. Greenlee
المصدر: Drug Development Research. 32:161-171
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Angiotensin II receptor type 1, Aldosterone, medicine.drug_class, Antagonist, Molecular biology, Angiotensin II, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, Drug Discovery, Renin–angiotensin system, medicine, Receptor, IC50
-
5
المؤلفون: L.W. Schaffer, Victor J. Lotti, Prasun K. Chakravarty, Wallace T. Ashton, Arthur A. Patchett, Tsing-Bau Chen, K. L. Flanagan, Salah D. Kivlighn, Elizabeth M. Naylor, W.J. Greenlee, Robert J. Bendesky, Linda L. Chang, Peter K. S. Siegl, R. S. L. Chang, Terry W. Schorn, Kristie A. Faust, Gloria J. Zingaro, Paul J. Kling
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:115-120
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Sulfonamide (medicine), Pharmaceutical Science, Pharmacology, Biochemistry, Angiotensin II, Chemical synthesis, chemistry.chemical_compound, Orally active, chemistry, Oral administration, In vivo, Drug Discovery, medicine, Triazole derivatives, Molecular Medicine, Tetrazole, Molecular Biology, hormones, hormone substitutes, and hormone antagonists, circulatory and respiratory physiology, medicine.drug
-
6
المؤلفون: Robert L, Hudkins, Lisa D, Aimone, Thomas R, Bailey, Robert J, Bendesky, Reddeppa Reddy, Dandu, Derek, Dunn, John A, Gruner, Kurt A, Josef, Yin-Guo, Lin, Jacquelyn, Lyons, Val R, Marcy, Joanne R, Mathiasen, Babu G, Sundar, Ming, Tao, Allison L, Zulli, Rita, Raddatz, Edward R, Bacon
المصدر: Bioorganicmedicinal chemistry letters. 21(18)
مصطلحات موضوعية: Male, Dose-Response Relationship, Drug, Molecular Structure, Drinking, Stereoisomerism, Rats, Histamine Agonists, Pyridazines, Disease Models, Animal, Structure-Activity Relationship, Animals, Humans, Receptors, Histamine H3, Wakefulness
-
7
المؤلفون: Mangeng Cheng, Lisa D. Aimone, Sheila J. Miknyoczki, Robert J. Bendesky, Thelma S. Angeles, Jie Qian, Robert L. Hudkins, Bruce D. Dorsey, Jean Husten, Bruce Ruggeri, Thomas Conners, Seetha Murthy, Hong Chang, Amy J. Landis, Jennifer Grobelny, Mark A. Ator
المصدر: Molecular Cancer Therapeutics. 12:C275-C275
مصطلحات موضوعية: Cancer Research, biology, Chemistry, Kinase, Cancer, medicine.disease, Receptor tyrosine kinase, Metastasis, c-Met inhibitor, Therapeutic index, Oncology, Tumor progression, Cancer cell, Immunology, biology.protein, medicine, Cancer research
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::247e348a81300a0bd69b9c09bd262614
https://doi.org/10.1158/1535-7163.targ-13-c275 -
8
المؤلفون: Bharat Lagu, Mohammad R. Marzabadi, Wanying Sun, John D. Gilbert, Douglas J. Pettibone, Sriram Tyagarajan, Robert J. Bendesky, T. G. Murali Dhar, Michael A. Patane, Theodore P. Broten, Dhanapalan Nagarathnam, Mark G. Bock, S. S. O'malley, and Roger M. Freidinger, Fengqi Zhang, George Chiu, Shou Wu Miao, Tsing Bao Chen, Jack Zhang, Kanyin Zhang, Kamlesh P. Vyas, Terry W. Schorn, Dake Tian, John M. Wetzel, Quanrong Shen, Kathryn Schneck, Charles M. Harrell, Charles Gluchowski, Wai C. Wong, Richard W. Ransom, Carlos Forray, Raymond S.L. Chang
المصدر: Journal of medicinal chemistry. 42(23)
مصطلحات موضوعية: Agonist, Male, Stereochemistry, medicine.drug_class, Metabolite, Drug Evaluation, Preclinical, Receptors, Opioid, mu, Biological Availability, Carboxamide, Blood Pressure, Pyrimidinones, In Vitro Techniques, Chemical synthesis, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Dogs, Piperidines, Urethra, GTP-Binding Proteins, Microsomes, Receptors, Adrenergic, alpha-1, Drug Discovery, medicine, Moiety, Animals, Humans, Adrenergic alpha-Antagonists, Prostate, Stereoisomerism, Recombinant Proteins, Rats, chemistry, Drug Design, Adrenergic alpha-1 Receptor Antagonists, Molecular Medicine, Piperidine, 4-Phenylpiperidine, Linker, Half-Life
-
9
المؤلفون: William J. Greenlee, Salah D. Kivlighn, Deborah Ondeyka, Peter K. S. Siegl, Victor J. Lotti, Raymond S.L. Chang, Stacey O'Malley, Paul J. Kling, Tsing-Bau Chen, Robert J. Bendesky, Nathan B. Mantlo
المصدر: European journal of pharmacology. 294(2-3)
مصطلحات موضوعية: Male, medicine.medical_specialty, Angiotensin receptor, Pyridines, Angiotensin II receptor antagonist, CHO Cells, In Vitro Techniques, Rats, Sprague-Dawley, Angiotensin Receptor Antagonists, Radioligand Assay, Internal medicine, Cricetinae, Renin–angiotensin system, medicine, Animals, Humans, Enalapril, Aldosterone, Pharmacology, Angiotensin II receptor type 1, Receptors, Angiotensin, biology, Chemistry, Angiotensin II, Imidazoles, Angiotensin-converting enzyme, Rats, Endocrinology, Vasoconstriction, biology.protein, Cattle, Rabbits, hormones, hormone substitutes, and hormone antagonists, medicine.drug
-
10
المؤلفون: Gregory E. Martin, Robert J. Bendesky
المصدر: Neuroscience Letters. 27:37-40
مصطلحات موضوعية: Agonist, Rotation, medicine.drug_class, Pharmacology, Bicuculline, chemistry.chemical_compound, In vivo, medicine, Animals, Humans, Microinjection, gamma-Aminobutyric Acid, Injections, Intraventricular, Pyrans, General Neuroscience, Rats, Inbred Strains, GABA receptor antagonist, Rats, Substantia Nigra, nervous system, Muscimol, chemistry, Biochemistry, Pyrones, Kojic amine, GABAergic, Female, Stereotyped Behavior, medicine.drug