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المؤلفون: Lee Andrew Harrison, Michael Dennis Dowle, Harry Finch, Robin Andrew Smith, Pritom Shah, K.Abhhilash Kumar, Gill Fleetwood, Simon Teanby Hodgson, George W. Hardy, Graham Murkitt, Simon J. F. Macdonald, Graham G. A. Inglis, Christopher R Molloy, Geoffrey D. Clarke, Augustin Amour, Rosalind E Godward, Tony Padfield, Davina Humphreys, M. R. Johnson, Mary Dixon, Tadeusz Skarzynski, Onkar M. P. Singh
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:895-898
مصطلحات موضوعية: Lactams, Human neutrophil, Metabolic Clearance Rate, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Dogs, Drug Stability, Piperidines, Pharmacokinetics, Cricetinae, Drug Discovery, Animals, Molecular Biology, Short duration, Serpins, Bacteria, Pancreatic Elastase, Chemistry, Serine Endopeptidases, Organic Chemistry, Elastase, Bacterial Infections, Rats, Bioavailability, Orally active, Pharmacodynamics, Molecular Medicine, Crystallization, Leukocyte Elastase, Intracellular
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المؤلفون: Alan J. Wonacott, Rosalind E Godward, Gill Fleetwood, Robin Andrew Smith, Pritom Shah, Simon J. F. Macdonald, Martin R. Johnson, Christopher R Molloy, George Hardy, Simon Teanby Hodgson, Lee Andrew Harrison, Augustin Amour, Michael Dennis Dowle, Onkar M. P. Singh, Graham G. A. Inglis, Mary Dixon, Davina Humphreys, Geoffrey D. Clarke
المصدر: Journal of medicinal chemistry. 45(18)
مصطلحات موضوعية: Male, Models, Molecular, Pyrrolidines, Lactams, Swine, Crystallography, X-Ray, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, Structure–activity relationship, Animals, Combinatorial Chemistry Techniques, Humans, Pyrroles, Enzyme Inhibitors, Pancreatic elastase, Sulfonamides, biology, Molecular Structure, Chemistry, Elastase, Stereoisomerism, In vitro, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Leukocyte Elastase