يعرض 1 - 5 نتائج من 5 نتيجة بحث عن '"Robin Van Den Hauwe"', وقت الاستعلام: 1.29s تنقيح النتائج
  1. 1
    Signaling Modulation via Minimal C-Terminal Modifications of Apelin-13

    المؤلفون: Léa Théroux, Robin Van Den Hauwe, Kien Trân, Justin Fournier, Michael Desgagné, Nathan Meneboo, Alexis Lavallée, Ulrike Fröhlich, Jérôme Côté, Charlie Hollanders, Jean-Michel Longpré, Alexandre Murza, Eric Marsault, Philippe Sarret, Pierre-Luc Boudreault, Steven Ballet

    المساهمون: Chemistry, Organic Chemistry

    مصطلحات موضوعية: Pharmacology, Pharmacology (medical)

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::15bd1073741ed01a6adbbcbf500ae054
    https://doi.org/10.1021/acsptsci.2c00219

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  2. 2
    Efficient Synthesis of Polysubstituted 1,5-Benzodiazepinone Dipeptide Mimetics via an Ugi-4CR-Ullmann Condensation Sequence

    المؤلفون: Charlie Hollanders, Steven Ballet, Robin Van Den Hauwe, Mathias Elsocht

    المساهمون: Chemistry, Faculty of Sciences and Bioengineering Sciences, Organic Chemistry

    المصدر: Synlett. 32:1719-1724

    مصطلحات موضوعية: Ullmann condensation, chemistry.chemical_compound, Dipeptide, chemistry, Ugi multicomponent reaction, Isocyanide, constrained dipeptides, Organic Chemistry, 1,5-benzodiazepinone, Sequence (biology), Cu-catalyzed Ullmann cyclization, Combinatorial chemistry

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2d48084bf1fcca1cae621629dc2ca4a7
    https://doi.org/10.1055/a-1545-2860

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  3. 3
    Constraining the Side Chain of C-Terminal Amino Acids in Apelin-13 Greatly Increases Affinity, Modulates Signaling, and Improves the Pharmacokinetic Profile

    المؤلفون: Eric Marsault, Robin Van Den Hauwe, Claude Spino, Sabrina Saibi, Xavier Sainsily, Jérôme Côté, Louise Simard, Alexandra Serre, Michel Bouvier, Steven Ballet, Mannix Auger-Messier, Jean-Michel Longpré, Lounès Haroune, Pierre Couvineau, Olivier Lesur, Alexandre Murza, Marco Echevarria, Kien Trân, Léa Théroux, Philippe Sarret

    المصدر: Journal of Medicinal Chemistry. 64:5345-5364

    مصطلحات موضوعية: Male, Stereochemistry, Blood Pressure, Plasma protein binding, Cleavage (embryo), GTP-Binding Protein alpha Subunits, G12-G13, 01 natural sciences, Rats, Sprague-Dawley, 03 medical and health sciences, In vivo, Drug Discovery, Animals, Humans, Amino Acid Sequence, Peptide sequence, 030304 developmental biology, Apelin receptor, chemistry.chemical_classification, Apelin Receptors, 0303 health sciences, Protein Stability, In vitro, Rats, 0104 chemical sciences, Amino acid, Apelin, 010404 medicinal & biomolecular chemistry, Amino Acid Substitution, chemistry, Intercellular Signaling Peptides and Proteins, Molecular Medicine, Half-Life, Protein Binding, Signal Transduction

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d6326583d9752754accc55d2ff5cb76
    https://doi.org/10.1021/acs.jmedchem.0c01941

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  4. 4
    1,5-Benzothiazepinone and arylazepinone dipeptide mimetics as local constraints in peptidomimetic design

    المؤلفون: P. Sarret, Louis Gendron, Dirk Tourwé, Robin Van Den Hauwe, Steven Ballet, Emilie Eiselt, Olivier Van der Poorten

    المصدر: Proceedings of the 35th European Peptide Symposium.

    مصطلحات موضوعية: chemistry.chemical_compound, Dipeptide, Chemistry, Peptidomimetic, Combinatorial chemistry

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::23b7dbb5dd6162f1881c4a73a2364e7a
    https://doi.org/10.17952/35eps.2018.178

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  5. 5
    χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds

    المؤلفون: Louis Gendron, Dirk Tourwé, Frédéric Bihel, Nga N. Chung, Peter W. Schiller, Olivier Van der Poorten, Cecilia Betti, Robin Van Den Hauwe, Karel Guillemyn, Emilie Eiselt, Steven Ballet, François Hallé, Philippe Sarret

    المساهمون: Laboratoire d'Innovation Thérapeutique (LIT), Université de Strasbourg (UNISTRA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Department of Organic Chemistry, Vrije Universiteit Brussel (VUB), Department of Physiology and Biophysics, Université de Sherbrooke (UdeS), Montreal Neurological Institute and Hospital, McGill University = Université McGill [Montréal, Canada], Centre National de la Recherche Scientifique (CNRS)-Université de Strasbourg (UNISTRA)-Institut de Chimie du CNRS (INC)

    المصدر: ACS Medicinal Chemistry Letters
    ACS Medicinal Chemistry Letters, American Chemical Society, 2017, 8 (11), pp.1177-1182. ⟨10.1021/acsmedchemlett.7b00347⟩

    مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Tetrapeptide, 010405 organic chemistry, Stereochemistry, Organic Chemistry, Peptide, Dermorphin, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, ANT, 0104 chemical sciences, Amino acid, 03 medical and health sciences, chemistry.chemical_compound, Residue (chemistry), 030104 developmental biology, chemistry, Drug Discovery, Receptor, Selectivity, ComputingMilieux_MISCELLANEOUS

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0eb26d3a07e8388d155d1e134bca1b18
    https://hal.archives-ouvertes.fr/hal-02368778

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