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المؤلفون: Michael Gershenovich, Yordanka Ivanova, Simon P. Fricker, Anna Zuk, Steven R. Ledbetter, Ron MacFarland
المصدر: American Journal of Physiology-Renal Physiology. 307:F783-F797
مصطلحات موضوعية: Chemokine, biology, Physiology, business.industry, Acute kidney injury, Renal function, Immune modulation, medicine.disease, CXCR4, Therapeutic approach, Immunology, biology.protein, Medicine, business, Antagonism, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ee61d691906bdabf372d3dee8004e636
https://doi.org/10.1152/ajprenal.00685.2013 -
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المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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المؤلفون: Gary Calandra, Ron MacFarland, Douglas A. Stewart, Clayton A. Smith
المصدر: Biology of Blood and Marrow Transplantation. 15(1):39-46
مصطلحات موضوعية: Adult, medicine.medical_specialty, Benzylamines, Receptors, CXCR4, Adolescent, Urology, Antigens, CD34, Cyclams, Transplantation, Autologous, Pharmacokinetics, Heterocyclic Compounds, Granulocyte Colony-Stimulating Factor, Autologous Transplantation, medicine, Autologous transplantation, Humans, Aged, Transplantation, CXCR4 antagonist, business.industry, Plerixafor, Lymphoma, Non-Hodgkin, Hematopoietic Stem Cell Transplantation, Hematology, Middle Aged, Hematopoietic Stem Cell Mobilization, Surgery, Regimen, Apheresis, Pharmacodynamics, Blood Component Removal, business, Multiple Myeloma, medicine.drug
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المؤلفون: Karin Badel, Ron MacFarland, Gary Calandra, John F. DiPersio, Feng Gao, Amanda F. Cashen, Sandra Lopez
المصدر: Biology of Blood and Marrow Transplantation. 14(11):1253-1261
مصطلحات موضوعية: Adult, Male, Oncology, Benzylamines, medicine.medical_specialty, Adolescent, Anti-HIV Agents, Population, CD34, Antigens, CD34, Cyclams, Transplantation, Autologous, CXCR4, AMD3100, Autologous stem-cell transplantation, Heterocyclic Compounds, Internal medicine, Granulocyte Colony-Stimulating Factor, medicine, Humans, education, Hematopoietic Stem Cell Mobilization, Aged, education.field_of_study, Transplantation, business.industry, Plerixafor, Hematopoietic stem cell mobilization, Hematology, Middle Aged, Hematopoietic Stem Cells, Hodgkin Disease, Surgery, Blood Component Removal, Female, Stem cell, business, Hodgkin lymphoma, Stem Cell Transplantation, medicine.drug
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المؤلفون: Ying Jun Cao, Jeong Gun Park, Nimalie D. Stone, Ron MacFarland, Charles Flexner, Beatrice Kallungal, Craig W. Hendrix, Ilene Wiggins, Sally Snyder, Camlin Tierney, Jeanne Conley, Stephen Becker, Christina M. Lalama, Karin L. Klingman, Gary Calandra, Shelia B. Dunaway
المصدر: Antimicrobial Agents and Chemotherapy. 51:2351-2358
مصطلحات موضوعية: Adult, Male, Receptors, CXCR4, Time Factors, Adolescent, medicine.medical_treatment, Administration, Oral, Pharmacology, Multiple dose, Butylamines, CXCR4, Antiviral Agents, Cohort Studies, Heterocyclic Compounds, 1-Ring, Pharmacokinetics, Oral administration, In vivo, Leukocytes, Humans, Medicine, Pharmacology (medical), Dosing, Leukocytosis, Receptor, Adverse effect, Chemotherapy, Dose-Response Relationship, Drug, business.industry, Headache, Fasting, Middle Aged, Antimicrobial, Dose–response relationship, Infectious Diseases, Area Under Curve, Toxicity, Aminoquinolines, Benzimidazoles, Erratum, medicine.symptom, business, Half-Life
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::13d810348b127b03f1d7723ff9003fee
https://doi.org/10.1128/aac.00013-07 -
6Leukocytosis and Mobilization of CD34+ Hematopoietic Progenitor Cells by AMD3100, a CXCR4 Antagonist
المؤلفون: Scott Cooper, Gary Calandra, Brent L. Wood, Ron MacFarland, Hal E. Broxmeyer, W. Conrad Liles, Gary Bridger, Elin Rodger, Kai Hübel, David C. Dale, Giao Hangoc, Geoffrey W. Henson
المصدر: Supportive Cancer Therapy. 1:165-172
مصطلحات موضوعية: Pharmacology, Cancer Research, Myeloid, business.industry, Monocyte, CD34, CXCR4, Subcutaneous injection, Haematopoiesis, medicine.anatomical_structure, Oncology, White blood cell, Immunology, Medicine, Leukocytosis, medicine.symptom, business
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7
المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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المؤلفون: Melanie Ruzek, Kim L. Nelson, Robert J. Scarborough, Stefan R. Idzan, Gary Bridger, Virginia Anastassov, Kathleen S. Neff, Gloria Lau, Marilyn C. Darkes, Rebecca S.Y. Wong, Jean Labrecque, Zefferino Santucci, Renee Mosi, Veronique Bodart, Ketan Patel, Simon P. Fricker, Ron MacFarland
المصدر: Biochemical pharmacology. 78(8)
مصطلحات موضوعية: Male, medicine.medical_specialty, Receptors, CXCR4, Maximum Tolerated Dose, Leukocytosis, Metabolic Clearance Rate, Pyridines, C-C chemokine receptor type 7, CHO Cells, Biology, Pharmacology, CXCR3, Kidney, Transfection, Biochemistry, CXCR4, Absorption, Cell Line, Chemokine receptor, Inhibitory Concentration 50, Mice, Cricetulus, Dogs, Heterocyclic Compounds, Internal medicine, Cricetinae, Calcium flux, medicine, Animals, Humans, Receptor, Fluorescent Dyes, Mice, Inbred BALB C, CXCR4 antagonist, Dose-Response Relationship, Drug, Molecular Structure, Chemotaxis, Antagonist, Fluoresceins, Chemokine CXCL12, Mice, Inbred C57BL, Endocrinology, Mice, Inbred DBA, Area Under Curve, Calcium, Half-Life, Protein Binding
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المؤلفون: Karin Badel, Stephen Becker, Gary B. Calandra, Colleen Gibney, Rebecca S.Y. Wong, X Antagonist Concept Trial Study Team, Marta Boffito, Edwin DeJesus, Gary Bridger, Graeme Moyle, Ron MacFarland
المصدر: Clinical infectious diseases : an official publication of the Infectious Diseases Society of America. 48(6)
مصطلحات موضوعية: Microbiology (medical), Adult, Male, medicine.medical_specialty, Anti-HIV Agents, Population, HIV Infections, Butylamines, Gastroenterology, Virus, Heterocyclic Compounds, 1-Ring, Receptors, HIV, Internal medicine, Medicine, Humans, Adverse effect, education, Tropism, education.field_of_study, biology, business.industry, Middle Aged, Viral Load, biology.organism_classification, CD4 Lymphocyte Count, Infectious Diseases, Treatment Outcome, Lentivirus, Immunology, Aminoquinolines, HIV-1, RNA, Viral, Benzimidazoles, Female, Viral disease, business, Viral load, Trofile assay
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::55ba3f66c1159ea682c91540a11c2c7e
https://pubmed.ncbi.nlm.nih.gov/19193109 -
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المؤلفون: Priscilla Chee, Gary Calandra, Craig W. Hendrix, Myaing M. Nyunt, Ron MacFarland, Stephanie Everts, Stephen Becker, Robert J. Scarborough
المصدر: Journal of acquired immune deficiency syndromes (1999). 47(5)
مصطلحات موضوعية: Pharmacokinetic Effect, Adult, CD4-Positive T-Lymphocytes, Male, Receptors, CXCR4, Adolescent, Leukocytosis, Midazolam, Administration, Oral, Pharmacology, CD8-Positive T-Lymphocytes, Butylamines, Dextromethorphan, Heterocyclic Compounds, 1-Ring, Pharmacokinetics, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), Drug Interactions, GABA Modulators, Volume of distribution, business.industry, Drug interaction, Middle Aged, Bioavailability, Infectious Diseases, Cytochrome P-450 CYP2D6, Aminoquinolines, Benzimidazoles, Female, business, Excitatory Amino Acid Antagonists, Drug metabolism, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::94850c41648aa2a3d293e178a0a8c3b2
https://pubmed.ncbi.nlm.nih.gov/18362694