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1دورية أكاديمية
المؤلفون: Terence G Hall, Yi Yu, Sudharshan Eathiraj, Yunxia Wang, Ronald E Savage, Jean-Marc Lapierre, Brian Schwartz, Giovanni Abbadessa
المصدر: PLoS ONE, Vol 11, Iss 9, p e0162594 (2016)
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Yi Yu, Ronald E Savage, Sudharshan Eathiraj, Justin Meade, Michael J Wick, Terence Hall, Giovanni Abbadessa, Brian Schwartz
المصدر: PLoS ONE, Vol 10, Iss 10, p e0140479 (2015)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1932-6203
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المؤلفون: Terence Hall, Yunxia Wang, Bassel F. El-Rayes, Patricia LoRusso, Walid L. Shaib, Jasgit C. Sachdev, Ronald E. Savage, R. D. Harvey, Giovanni Abbadessa, Julia Kazakin, Drew W. Rasco, Amita Patnaik, Brian Schwartz, Kyriakos P. Papadopoulos, Anthony W. Tolcher
المصدر: British Journal of Cancer
مصطلحات موضوعية: 0301 basic medicine, Adult, Male, Cancer Research, medicine.medical_specialty, Pathology, FGFR2 fusion, Nausea, Administration, Oral, Gastroenterology, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Internal medicine, Neoplasms, medicine, Adrenocortical carcinoma, Humans, Dosing, Adverse effect, Protein Kinase Inhibitors, solid tumours, Aged, Aniline Compounds, business.industry, Middle Aged, medicine.disease, Receptors, Fibroblast Growth Factor, FGFR inhibitor, 030104 developmental biology, Oncology, phase 1, 030220 oncology & carcinogenesis, Pharmacodynamics, Toxicity, Cohort, Clinical Study, Quinazolines, Female, medicine.symptom, business
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4
المؤلفون: Paul Jarosinski, Staci Martin, Neera R. Nathan, Mohammadhadi Bagheri, Brigitte C. Widemann, Julie C. Sapp, Pamela L. Wolters, Ronald E. Savage, Ashlyn Gruber, Marjorie J. Lindhurst, Scott M. Paul, Eva Dombi, Brian Schwartz, Leslie G. Biesecker, Thomas N. Darling, Kim M. Keppler-Noreuil, Jasmine Burton-Akright
مصطلحات موضوعية: 0301 basic medicine, Oncology, Adult, Male, medicine.medical_specialty, Adolescent, Maximum Tolerated Dose, AKT1, Aminopyridines, Pain, Pilot Projects, Article, Proteus Syndrome, 03 medical and health sciences, Young Adult, 0302 clinical medicine, Internal medicine, Cerebriform connective tissue nevus, Genetics, medicine, Clinical endpoint, Humans, Tissue Distribution, Phosphorylation, Child, Nevus, Genetics (clinical), Connective tissue nevus, business.industry, Imidazoles, Middle Aged, medicine.disease, Prognosis, Proteus syndrome, 030104 developmental biology, Pharmacodynamic Study, 030220 oncology & carcinogenesis, Overgrowth syndrome, Pharmacodynamics, Female, business, Proto-Oncogene Proteins c-akt
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d7abeed1fc81a195fe0f605c672bc5f
https://europepmc.org/articles/PMC6407523/ -
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المؤلفون: Jean-Marc Lapierre, Cathy O. Bull, Ronald E. Savage, Sudharshan Eathiraj, David Vensel, Sapna Makhija, Eugene Kelleher, Neil Westlund, Jeff Szwaya, Yanbin Liu, Steffi Koerner, Magdi Moussa, Susan Cornell-Kennon, Akihisa Matsuda, Darin Kizer, Nivedita Namdev, Hui Wu, Shin Iimura, Brian Schwartz, Erika Volckova
المصدر: Journal of Medicinal Chemistry. 59:6455-6469
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Allosteric regulation, Administration, Oral, Aminopyridines, AKT1, Antineoplastic Agents, AKT2, Mice, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Allosteric Regulation, Drug Discovery, Animals, Humans, Moiety, Protein Kinase Inhibitors, Protein kinase B, Cell Proliferation, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Imidazoles, Neoplasms, Experimental, Endometrial Neoplasms, 030104 developmental biology, Enzyme, chemistry, 030220 oncology & carcinogenesis, embryonic structures, Molecular Medicine, Phosphorylation, Female, Drug Screening Assays, Antitumor, Carcinoma, Endometrioid, Proto-Oncogene Proteins c-akt
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6
المؤلفون: Yi Yu, Eva Volckova, Brian Schwartz, Ronald E. Savage, Alden Harring
المصدر: Molecular Cancer Therapeutics. 18:C076-C076
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Fulvestrant, business.industry, medicine.medical_treatment, Cancer, Palbociclib, medicine.disease, Olaparib, Targeted therapy, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Oncology, chemistry, Paclitaxel, In vivo, 030220 oncology & carcinogenesis, medicine, Cancer research, business, PI3K/AKT/mTOR pathway, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d7eb1d04da6ce353cf3219752911da42
https://doi.org/10.1158/1535-7163.targ-19-c076 -
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المؤلفون: Maria Lamar, Terence Hall, Brian Schwartz, Julia Kazakin, Shubham Pant, Ronald E. Savage
المصدر: Molecular Cancer Therapeutics. 18:A034-A034
مصطلحات موضوعية: Cancer Research, business.industry, Insulin, medicine.medical_treatment, Cmax, AKT1, Pharmacology, Oncology, Pharmacokinetics, Pharmacodynamics, medicine, business, Protein kinase B, PI3K/AKT/mTOR pathway, Whole blood
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b10813e62a4002c06d4b28d9d65807c6
https://doi.org/10.1158/1535-7163.targ-19-a034 -
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المؤلفون: Jennifer A. Woyach, John C. Byrd, Ian W. Flinn, Ronald E. Savage, Lindsey Granlund, Sudharshan Eathiraj, Seema A. Bhat, Feng Chai, Deborah M. Stephens, Lyndsey A. Szuszkiewicz, Brian Schwartz
المصدر: Blood. 134:4298-4298
مصطلحات موضوعية: medicine.medical_specialty, business.industry, Immunology, Cell Biology, Hematology, medicine.disease, Biochemistry, Rash, Discontinuation, chemistry.chemical_compound, Cmin, Tolerability, chemistry, Internal medicine, Ibrutinib, Absolute neutrophil count, Medicine, Acalabrutinib, medicine.symptom, business, Febrile neutropenia
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f9c7bd3e9eb2bbfd19e26c6986087cef
https://doi.org/10.1182/blood-2019-127260 -
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المؤلفون: Lyndsey A. Szuszkiewicz, John C. Byrd, Ian W. Flinn, Ronald E. Savage, S. Eathiraj, Deborah M. Stephens, Jennifer A. Woyach, Seema A. Bhat, L. Granlund, Feng Chai
المصدر: HemaSphere. 3:521-522
مصطلحات موضوعية: Oncology, medicine.medical_specialty, medicine.anatomical_structure, Refractory, business.industry, Internal medicine, Dose escalation, medicine, In patient, Hematology, business, B cell
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المؤلفون: Daisuke Nakai, Tomoko Takayama, Ronald E. Savage, Yumi Nishiya, Takanori Yasukochi, Satoru Ohsuki, Yuji Iwano, Yoko Urasaki, Takashi Izumi, Shohei Bazyo, Atsushi Kurihara, Hideo Takakusa, Chikahiro Oza
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 46(11)
مصطلحات موضوعية: Health, Toxicology and Mutagenesis, Metabolite, Glucuronidation, Antineoplastic Agents, Biology, Pharmacology, Toxicology, Hydroxylation, 030226 pharmacology & pharmacy, Biochemistry, c-Met inhibitor, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Humans, Tivantinib, Alcohol dehydrogenase, CYP3A4, Alcohol Dehydrogenase, Cytochrome P450, General Medicine, Pyrrolidinones, Cytochrome P-450 CYP2C19, chemistry, 030220 oncology & carcinogenesis, biology.protein, Quinolines, Oxidation-Reduction