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1
المؤلفون: George L. Trainor, Jun Dai, Arvind Mathur, Francis Y. Lee, Sunilkumar Mandal, Yingru Zhang, Richard Rampulla, Kiran Babu Gona, Patrice Gill, Raja Thiruvenkadam, Victor R. Guarino, Wen-Ching Han, Ding Ren Shen, Aaron Balog, Mary Ellen Cvijic, Dauh-Rurng Wu, Gregory D. Vite, Krista Menard, Anne Rose, Sathiah Kandula, Ashvinikumar V. Gavai, Weifang Shan, John T. Hunt, Asoka Ranasinghe, Kelly McGlinchey, Richard A. Westhouse, Claude A. Quesnelle, Derek J. Norris, Mei-Li Wen, Ronald E. White, Kamalraj Thiyagarajan
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:1905-1909
مصطلحات موضوعية: Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Antineoplastic Agents, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Receptor, Solid tumor, Molecular Biology, Cell Proliferation, Benzodiazepinones, Dose-Response Relationship, Drug, Molecular Structure, Receptors, Notch, Chemistry, Organic Chemistry, Biological activity, Neoplasms, Experimental, medicine.disease, Leukemia, Orally active, Microsomes, Liver, Molecular Medicine, Drug Screening Assays, Antitumor
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2
المؤلفون: Claude A. Quesnelle, Patrice Gill, Richard Rampulla, Ching Su, Gerry Everlof, George L. Trainor, Ke Chen, Vinod Arora, Richard A. Westhouse, Celia D’Arienzo, Andrew J. Tebben, Weifang Shan, John T. Hunt, Derek J. Norris, Louis J. Lombardo, Zheng Yang, Arvind Mathur, Mei-Li Wen, Yingru Zhang, Dauh-Rurng Wu, Wen-Ching Han, Krista Menard, Victor R. Guarino, Asoka Ranasinghe, Richard E. Olson, Ashvinikumar V. Gavai, Bruce S. Fischer, Phil S. Baran, Anne Rose, Lan Xiao, Ronald E. White, Mary Ellen Cvijic, Gregory D. Vite, Ding Ren Shen, Jere E. Meredith, Haiqing Wang, Francis Y. Lee, Aaron Balog
المصدر: ACS Medicinal Chemistry Letters. 6:523-527
مصطلحات موضوعية: business.industry, Organic Chemistry, Pharmacology, medicine.disease, Biochemistry, T Acute Lymphoblastic Leukemia, Leukemia, In vivo, Drug Discovery, medicine, Receptor, business, Solid tumor, Clinical evaluation, Triple-negative breast cancer
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3
المؤلفون: Annette S. Uss, Ganfeng Wang, Samir K. Gupta, Rong Liu, F. George Njoroge, Tongtong Liu, Dan Prelusky, Lisa Broske, Yunsheng Hsieh, Ronald E. White, Anastasia Pavlosky, Cheng Li, K.-C. Cheng
المصدر: Letters in Drug Design & Discovery. 6:312-318
مصطلحات موضوعية: Chemistry, Hepatitis C virus, Pharmaceutical Science, medicine.disease_cause, Virology, In vitro, chemistry.chemical_compound, Boceprevir, Drug Discovery, medicine, Molecular Medicine, Protease inhibitor (pharmacology), Selection (genetic algorithm), In vivo pharmacokinetics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6e480d708b3dacfed0ba6c00ed1ee2b4
https://doi.org/10.2174/157018009788452474 -
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المؤلفون: Ronald E. White, Valerie Gerlach, Richard Morrison, Ann Thomas, K.-C. Cheng, Xiaoming Cui
المصدر: Biochemical Pharmacology. 76:680-689
مصطلحات موضوعية: Receptors, Steroid, Drug Evaluation, Preclinical, Retinoid X receptor, Pharmacology, Biology, Polymerase Chain Reaction, Biochemistry, Cell Line, Flutamide, chemistry.chemical_compound, Gene interaction, Genes, Reporter, Luciferases, Firefly, In vivo, Cytochrome P-450 CYP3A, Humans, DNA Primers, EC50, Pregnane X receptor, Base Sequence, CYP3A4, Pregnane X Receptor, Drug interaction, chemistry, Enzyme Induction, Hepatocytes
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5
المؤلفون: Weidong Pan, Prudence Bradley, Kevin X. Chen, Parekh Tejal N, Andrea Hart, Frank Bennett, Danial Prelusky, Srikanth Venkatraman, Robert Chase, Susan Bogdanowich-Knipp, Jianshe Kong, Bancha Vibulbhan, Viyyoor M. Girijavallabhan, Hendrata Siska, Rong Kong, Weiying Yang, Kuo-Chi Cheng, Ashit K. Ganguly, Nancy Butkiewicz, Ashok Arasappan, Yuhua Huang, Andrew Prongay, Bruce A. Malcolm, Xiang Liang, Rong Liu, Xiaoming Cui, Walter A. Korfmacher, Sony Agrawal, Wanli Wu, Zhuyan Guo, Stephane L. Bogen, Pike Russell E, Ronald E. White, Jesse Wong, Yi-Tsung Liu, Jean-Marc Brisson, John Pichardo, Anil K. Saksena, Pavlovsky Anastasia, Bahige M. Baroudy, F. George Njoroge, Vincent Madison, Patrick Pinto, Santhanam Bama, Raymond G. Lovey, Edwin Jao, Lisa Broske, Veljko Popov, Yunsheng Hsieh, Paul Ingravallo, Sumei Ruan, Piwinski John J
المصدر: Journal of Medicinal Chemistry. 49:6074-6086
مصطلحات موضوعية: Hepatitis, NS3, biology, Hepacivirus, Hepatitis C virus, Ribavirin, Hepatitis C, medicine.disease, biology.organism_classification, medicine.disease_cause, Virology, chemistry.chemical_compound, chemistry, Hepatocellular carcinoma, Drug Discovery, medicine, Molecular Medicine, Protease inhibitor (pharmacology)
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6
المؤلفون: Diana Montgomery, Cheng Li, Tong-tong Liu, Yunsheng Hsieh, Ronald E. White, K.-C. Cheng
المصدر: Journal of Pharmacological and Toxicological Methods. 53:215-218
مصطلحات موضوعية: Cell Culture Techniques, Administration, Oral, Hybrid Cells, Biology, Pharmacology, Toxicology, Xenobiotics, Rats, Sprague-Dawley, Pharmacokinetics, Predictive Value of Tests, In vivo, medicine, Animals, Humans, Cells, Cultured, In vitro, Rats, Bioavailability, Kinetics, Human hepatocyte, medicine.anatomical_structure, Caco-2, Area Under Curve, Hepatocyte, Hepatocytes, Linear Models, Biological Assay, Time curve, Caco-2 Cells
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7كتاب إلكتروني
نوع المادة: eBook.
الموضوعات: World War, 1939-1945--Naval operations, British, Americans--Great Britain--History--20th century, Sailors--United States--Biography
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8
المؤلفون: Xiaoming Cui, K.-C. Cheng, Ronald E. White, Yau Yi Lau, Elpida Sapidou
المصدر: Drug Metabolism and Disposition. 30:1446-1454
مصطلحات موضوعية: Metabolic Clearance Rate, Cell Culture Techniques, Pharmaceutical Science, Biology, Cryopreservation, Andrology, Dogs, Pharmacokinetics, In vivo, medicine, Animals, Humans, Incubation, Cells, Cultured, Pharmacology, Fissipedia, biology.organism_classification, In vitro, Rats, Macaca fascicularis, medicine.anatomical_structure, Cell culture, Hepatocyte, Immunology, Hepatocytes
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a1d35adf11379c92d12200d26372751c
https://doi.org/10.1124/dmd.30.12.1446 -
9
المؤلفون: Sunil Paliwal, Yan Xia, Diane Rindgen, Ronald E. White, Hong Kim, Gregory A. Reichard, Kathleen Cox, Amin A. Nomeir, David Hesk, Matthew Bryant, Jairam Palamanda, Feng Wenqing, Chan Tze-Ming
المصدر: Journal of Separation Science. 25:877-882
مصطلحات موضوعية: Chromatography, Chemistry, Metabolite, Filtration and Separation, Biological activity, Nuclear magnetic resonance spectroscopy, Tandem mass spectrometry, High-performance liquid chromatography, Analytical Chemistry, chemistry.chemical_compound, Pregnenolone, medicine, Microsome, Solid phase extraction, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::5b51bd25318b6a7ea044ccfe961c812e
https://doi.org/10.1002/1615-9314(20021001)25:14<877::aid-jssc877>3.0.co;2-w -
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المؤلفون: Vincent Madison, Ronald E. White, Li Xiao, Xiaoming Cui, K.-C. Cheng
المصدر: Drug Metabolism and Disposition. 30:951-956
مصطلحات موضوعية: Models, Molecular, Receptors, Steroid, Pyridines, Stereochemistry, Molecular Sequence Data, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Ligands, Calcitriol receptor, Pregnanediones, chemistry.chemical_compound, Humans, Amino Acid Sequence, Androstanols, Clotrimazole, Receptor, Constitutive Androstane Receptor, Pharmacology, Orphan receptor, Pregnane X receptor, Chemistry, Pregnane X Receptor, Ligand (biochemistry), Cell biology, Nuclear receptor, Docking (molecular), Receptors, Calcitriol, Androstane, Protein Binding, Transcription Factors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7dffd523dfccb2af10e3165850eba2b5
https://doi.org/10.1124/dmd.30.9.951