-
1
المؤلفون: Masahiro Fujita, Yu Wen Li, Joanne J. Bronson, Heidi Dulac, Robert Zaczek, Jeffrey A. Deskus, Robert B. Innis, Masao Imaizumi, Victor W. Pike, Rick L. Pieschl, Frederick T. Chin, Nicholas J. Lodge, John E. Macor, Sami S. Zoghbi, Thaddeus F. Molski, Douglas D. Dischino, Ronald J. Mattson
المصدر: Nuclear Medicine and Biology. 41:524-535
مصطلحات موضوعية: Male, Cancer Research, Cerebellum, medicine.medical_specialty, Biodistribution, Chemistry Techniques, Synthetic, Ligands, Receptors, Corticotropin-Releasing Hormone, Article, Internal medicine, medicine, Radioligand, Animals, Tissue Distribution, Radiology, Nuclear Medicine and imaging, Receptor, Radiochemistry, Chemistry, Brain, Human brain, Ligand (biochemistry), Macaca mulatta, In vitro, Rats, medicine.anatomical_structure, Endocrinology, Positron-Emission Tomography, Pyrazines, Molecular Medicine, Brainstem
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e6ef3db952927de40d265e3f67da6557
https://doi.org/10.1016/j .nucmedbio.2014.03.005 -
2
المؤلفون: Julia M. Nielsen, Jennifer McDonald, Dmitry Zuev, Megan Hayes, Eric Wexler, Joanne J. Bronson, Henry Wong, Yu-Wen Li, Nicholas J. Lodge, John E. Macor, Jeffrey A. Deskus, James E. Grace, Hong Huang, Gail K. Mattson, Mary Guaraldi, Derek J. Denhart, David C. Onthank, Vijay T. Ahuja, Heidi Dulac, Michael F. Parker, Larisa Zueva, Douglas D. Dischino, Ronald J. Mattson, Thaddeus F. Molski, Michael Azure, Jonathan L. Ditta, Richard A. Hartz
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:6651-6655
مصطلحات موضوعية: Fluorine Radioisotopes, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Medicinal chemistry, Imaging, Three-Dimensional, Drug Discovery, Radioligand, Animals, Tissue Distribution, Molecular Biology, Aniline Compounds, Molecular Structure, Chemistry, Organic Chemistry, Binding properties, Brain, Pet imaging, Metabolic stability, Rat brain, Rats, Positron-Emission Tomography, Pyrazines, Lipophilicity, Pyrazoles, Molecular Medicine
-
3
المؤلفون: Hong Huang, Nicholas J. Lodge, John E. Macor, Ronald J. Mattson, Edward S. Kozlowski, Gail K. Mattson, Xiaohua Stella Huang, Julia M. Nielsen, Qi Gao, Joanne J. Bronson, Dedong Wu, Dmitry Zuev, Larisa Zueva
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2484-2488
مصطلحات موضوعية: Nitrile, Bicyclic molecule, Triazines, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Crf1 receptor, Molecular Conformation, Pharmaceutical Science, Pet imaging, Crystallography, X-Ray, Ligand (biochemistry), Receptors, Corticotropin-Releasing Hormone, Biochemistry, Chemical synthesis, Molecular conformation, chemistry.chemical_compound, chemistry, Positron-Emission Tomography, Drug Discovery, Pyrazoles, Molecular Medicine, Amines, Molecular Biology
-
4
المؤلفون: Qi Gao, Brett R. Beno, Zhaoxing Meng, Jeffrey A. Deskus, Charles P. Sloan, Nicholas J. Lodge, John E. Macor, Matthew T. Taber, Melissa A. Lapaglia, Dalton King, Thaddeus F. Molski, Ronald J. Mattson, Edward S. Kozlowski, Gail K. Mattson
المصدر: Journal of Medicinal Chemistry. 53:7564-7572
مصطلحات موضوعية: Models, Molecular, Serotonin, Nitrile, Stereochemistry, Microdialysis, Molecular Conformation, Biological Availability, Cyclopentanes, Ring (chemistry), Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Side chain, Extracellular, Animals, Humans, Potency, Cerebral Cortex, Serotonin Plasma Membrane Transport Proteins, Indole test, Chemistry, Tryptamines, Rats, Molecular Medicine, Extracellular Space, Selective Serotonin Reuptake Inhibitors, Cis–trans isomerism
-
5
المؤلفون: Thaddeus F. Molski, Ronald J. Mattson, Gail K. Mattson, Qi Gao, Dedong Wu, Lawrence R. Marcin, Nicholas J. Lodge
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1027-1030
مصطلحات موضوعية: Indoles, Nitrile, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Ring (chemistry), Biochemistry, Chemical synthesis, Cell Line, Nitrone, chemistry.chemical_compound, Drug Discovery, Humans, Moiety, Molecular Biology, Serotonin Plasma Membrane Transport Proteins, chemistry.chemical_classification, Tetrahydroisoquinoline, Organic Chemistry, Tryptamines, Cycloaddition, chemistry, Molecular Medicine, Enantiomer, Protein Binding
-
6
المؤلفون: Yu-Wen Li, Harvey Wong, Allison B. Brenner, James E. Grace, Jianqing Li, Maria Rafalski, Nicholas J. Lodge, Macor John E, Ronald J. Mattson, Jonathan L. Ditta, Thaddeus F. Molski, Joanne J. Bronson, Vijay T. Ahuja, Robert Zaczek, Richard A. Hartz, Snjezana Lelas, Argyrios G. Arvanitis, Jeffrey A. Deskus, Kimberley A. Lentz, Richard E. Olson, Andrew P. Combs, William D. Schmitz, Eddy W. Yue, Derek J. Denhart
المصدر: Journal of Medicinal Chemistry. 52:4161-4172
مصطلحات موضوعية: Male, Metabolic Clearance Rate, Chemistry, Antagonist, Pharmacology, Receptors, Corticotropin-Releasing Hormone, Rats, Corticotropin-releasing hormone receptor 1, Bioavailability, Inhibitory Concentration 50, Biochemistry, Pharmacokinetics, In vivo, Oral administration, Pyrazines, Drug Discovery, Animals, Humans, Molecular Medicine, Receptor, IC50
-
7
المؤلفون: Rudolph G. Krause, Charles P. Sloan, Jingfang Qian-Cutrone, Thaddeus F. Molski, Joseph A. Cipollina, Gail K. Mattson, Matthew T. Taber, Qi Gao, Ronald J. Mattson, Jeffrey A. Deskus, James R. Epperson, Brett R. Beno, Baoqing Ma, Nicholas J. Lodge, Pierre Dextraze
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:3099-3104
مصطلحات موضوعية: Indoles, Nitrile, Pyridines, Stereochemistry, Microdialysis, Clinical Biochemistry, Molecular Conformation, Substituent, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Fluoxetine, Cyclohexenes, Drug Discovery, Animals, Humans, Serotonin Uptake Inhibitors, Molecular Biology, Serotonin transporter, Serotonin Plasma Membrane Transport Proteins, Indole test, biology, Organic Chemistry, Tryptamines, Rats, chemistry, biology.protein, Molecular Medicine, Serotonin, Reuptake inhibitor, Selective Serotonin Reuptake Inhibitors
-
8
المؤلفون: Gail K. Mattson, Charles P. Sloan, Matthew T. Taber, Brett R. Beno, Ronald J. Mattson, Melissa A. Cunningham, Qi Gao, Mendi A. Higgins, Nicholas J. Lodge, Thaddeus F. Molski, Jeffrey A. Deskus, Jonathan L. Ditta, Lawrence R. Marcin, John D. Catt, Derek J. Denhart
المصدر: Journal of Medicinal Chemistry. 48:6023-6034
مصطلحات موضوعية: Cyclopropanes, Models, Molecular, Steric effects, Indoles, Nitrile, Molecular model, Stereochemistry, Microdialysis, Serotonin reuptake inhibitor, Molecular Conformation, Crystallography, X-Ray, Cyclopropane, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Indole test, Stereoisomerism, Tryptamines, Frontal Lobe, Rats, chemistry, Receptors, Serotonin, Molecular Medicine, Serotonin, Enantiomer, Selective Serotonin Reuptake Inhibitors
-
9
المصدر: Journal of Labelled Compounds and Radiopharmaceuticals. 45:987-994
مصطلحات موضوعية: medicine.drug_class, Organic Chemistry, Ether, Carboxamide, Biochemistry, High-performance liquid chromatography, Chemical synthesis, Analytical Chemistry, Melatonergic, chemistry.chemical_compound, chemistry, Drug Discovery, medicine, Organic chemistry, Radiology, Nuclear Medicine and imaging, Trimethylstannane, Aliphatic compound, Spectroscopy, Thallium salt
-
10
المؤلفون: Charles P. Sloan, Qi Gao, Christopher C. Lockhart, Ronald J. Mattson, John D. Catt, Stella Huang
المصدر: The Journal of Organic Chemistry. 64:8004-8007
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Iodobenzene, Medicinal chemistry