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المؤلفون: Kenneth E. Carlson, Olafur S. Gudmundsson, Bruce A. Ellsworth, Philip M. Sher, Susan Harvey, Eva Zuvich, Michael Thomas, William J. Keim, Gang Wu, Helen E. Godonis, Paul Stetsko, Brian J. Murphy, Richard B. Sulsky, Guixue Yu, William R. Ewing, Mary Jane Cullen, Mary Ann Pelleymounter, Doree F. Sitkoff, Susan Johnghar, Zhengxiang Gu, Ximao Wu, James Devenny, Rose Ann F Baska, Asoka Ranasinghe, Ning Lee, Kamelia Behnia, Anthony V. Azzara, Kenneth W. Rohrbach, Gerry Everlof, Liya Kang, Natesan Murugesan, Yeheng Zhu, Yifan Yang
المصدر: Journal of Medicinal Chemistry. 56:9586-9600
مصطلحات موضوعية: Cannabinoid receptor, Drug discovery, Chemistry, medicine.medical_treatment, Antagonist, Triazoles, Pharmacology, Rats, Pyridazines, Structure-Activity Relationship, Cytochrome P-450 Enzyme System, Receptor, Cannabinoid, CB1, Pharmacokinetics, In vivo, Free fraction, Drug Discovery, medicine, Animals, Molecular Medicine, Structure–activity relationship, Cannabinoid, Half-Life, Protein Binding
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المؤلفون: Annapurna Pendri, Liya Kang, Kenneth E. Carlson, William R. Ewing, Jing Chen, Neil T. Burford, Chongqing Sun, Dharmpal S. Dodd, Mary Ellen Cvijic, Rose Ann F Baska, Samuel Gerritz
المصدر: ACS combinatorial science. 14(3)
مصطلحات موضوعية: Molecular Structure, Stereochemistry, medicine.medical_treatment, Aryl, General Chemistry, General Medicine, Pyrazole, Combinatorial chemistry, Amides, Acylation, chemistry.chemical_compound, Inhibitory Concentration 50, Solid-phase synthesis, chemistry, Receptor, Cannabinoid, CB1, Amide, Drug Discovery, medicine, Pyrazoles, Amine gas treating, Cannabinoid, Solid-Phase Synthesis Techniques, G protein-coupled receptor, Protein Binding
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المؤلفون: Kenneth E. Carlson, Yeheng Zhu, Yifan Yang, William R. Ewing, Rose Ann F Baska, Ying Wang, Bruce A. Ellsworth, Qi Huang, Samuel Gerritz, Susan Johnghar, Neil T. Burford, William N. Washburn, Mary Ann Pelleymounter, Chongqing Sun, Kamelia Behnia, Annapurna Pendri, Liya Kang, Mary Jane Cullen
المصدر: Bioorganicmedicinal chemistry letters. 17(14)
مصطلحات موضوعية: Pyrazine, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, Receptor, Cannabinoid, CB1, In vivo, Oral administration, Drug Discovery, medicine, Structure–activity relationship, Animals, Molecular Biology, ADME, Chemistry, Organic Chemistry, Amides, Pyrazinamide, Rats, Molecular Medicine
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المؤلفون: Maria T. Valentine, Natesan Murugesan, Yifan Yang, Leena Fadnis, W. Griffith Humphreys, Robert Zahler, Shih-Jung Lan, William R. Ewing, John E. Macor, Kenneth E. Carlson, Rose Ann F Baska, Kenneth E.J. Dickinson, Hossain Monshizadegan, Mark C. Kowala, John E. Tellew, Zhengxiang Gu, Sophie Beyer
المصدر: Journal of medicinal chemistry. 48(1)
مصطلحات موضوعية: Male, medicine.medical_specialty, medicine.drug_class, Endothelin A Receptor Antagonists, Administration, Oral, Biological Availability, Tetrazoles, Receptor, Angiotensin, Type 1, Structure-Activity Relationship, Irbesartan, Dogs, Internal medicine, Rats, Inbred SHR, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Receptor, Antihypertensive Agents, Sulfonamides, Angiotensin II receptor type 1, Chemistry, Angiotensin II, Biphenyl Compounds, Antagonist, Isoxazoles, Receptor antagonist, Rats, Macaca fascicularis, Endocrinology, Hypertension, cardiovascular system, Molecular Medicine, Angiotensin II Type 1 Receptor Blockers, medicine.drug
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المؤلفون: Natesan Murugesan, Mark H. Perrone, John E. Tellew, Mark C. Kowala, Jergen Baumann, Rose Ann F Baska, Yifan Yang, Zhengxiang Gu, Eileen Bird, Carol S. Ryan, Bridgette Kane, Kenneth E.J. Dickinson, Kenneth E. Carlson, Susan Arthur, Balkrushna C. Panchal, Sophie Beyer, Mary Giancarli, Pam Ferrer, Donglu Zhang, Leena Fadnis, John E. Macor, Hossain Monshizadegan, Joel C. Barrish, Nick C. Trippodo
المصدر: The Journal of pharmacology and experimental therapeutics. 309(1)
مصطلحات موضوعية: Male, medicine.medical_specialty, Angiotensin receptor, Vascular smooth muscle, medicine.drug_class, Endothelin A Receptor Antagonists, Tetrazoles, Blood Pressure, Pharmacology, Essential hypertension, Losartan, Receptor, Angiotensin, Type 1, Internal medicine, Rats, Inbred SHR, medicine, Animals, Humans, Desoxycorticosterone, Oxazoles, Antihypertensive Agents, Sulfonamides, Angiotensin II receptor type 1, Chemistry, Biphenyl Compounds, Sodium, Irbesartan, Receptor antagonist, medicine.disease, Receptor, Endothelin A, Angiotensin II, Rats, Disease Models, Animal, Endocrinology, Hypertension, Molecular Medicine, Calcium, Endothelin receptor, Angiotensin II Type 1 Receptor Blockers
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f0898471daf6b36f8b1af60fb680e492
https://pubmed.ncbi.nlm.nih.gov/14718594 -
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المؤلفون: Maria T. Valentine, Natesan Murugesan, John E. Tellew, Sophie Beyer, John E. Macor, Yifan Yang, Zhengxiang Gu, Cornelius Lyndon A M, Mark C. Kowala, Bridgette L. Kunst, Leena Fadnis, Carol S. Ryan, Hossain Monshizadegan, Kenneth E. Carlson, Rose Ann F Baska
المصدر: Bioorganicmedicinal chemistry letters. 13(6)
مصطلحات موضوعية: Endothelin Receptor Antagonists, Male, Angiotensin receptor, medicine.medical_specialty, Clinical Biochemistry, Pharmaceutical Science, Blood Pressure, Biochemistry, Receptor, Angiotensin, Type 1, Rats, Sprague-Dawley, Angiotensin Receptor Antagonists, Structure-Activity Relationship, Internal medicine, Drug Discovery, Renin–angiotensin system, medicine, Animals, Humans, Molecular Biology, Sulfonamides, Angiotensin II receptor type 1, Binding Sites, Chemistry, Organic Chemistry, Biphenyl Compounds, Antagonist, Imidazoles, Receptor, Endothelin A, Angiotensin II, Rats, Biphenyl compound, Endocrinology, Drug Design, Molecular Medicine, Indicators and Reagents, Caco-2 Cells, Endothelin receptor
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المؤلفون: John E. Tellew, Rose Ann F Baska, Cornelius Lyndon A M, Zhengxiang Gu, Kenneth E. Carlson, Richard A. Morrison, Maria T. Valentine, John E. Macor, Kenneth E.J. Dickinson, James R. Powell, Natesan Murugesan, Sophie Beyer, Yifan Yang, Balkrushna C. Panchal, Mark C. Kowala, Bridgette L. Kunst, Suzanne Moreland, Joel C. Barrish, Leena Fadnis, Hossain Monshizadegan, Saeho Chong
المصدر: Journal of medicinal chemistry. 45(18)
مصطلحات موضوعية: Endothelin Receptor Antagonists, Stereochemistry, Blood Pressure, CHO Cells, Crystallography, X-Ray, Chemical synthesis, Receptor, Angiotensin, Type 1, Angiotensin Receptor Antagonists, Radioligand Assay, Structure-Activity Relationship, Irbesartan, Cricetinae, Drug Discovery, medicine, Animals, Receptor, Antihypertensive Agents, Sulfonamides, Angiotensin II receptor type 1, Bicyclic molecule, Molecular Structure, Chemistry, Angiotensin II, Antagonist, Isoxazoles, Receptor, Endothelin A, Endothelin A Receptor Antagonists, Rats, Molecular Medicine, medicine.drug
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المؤلفون: Kenneth E.J. Dickinson, Robert Cohen, Catherine C Bryson, Rose Ann F Baska, Kirk Schroeder, Mark A. Smith, Nicholas J. Lodge
المصدر: European journal of pharmacology. 345(1)
مصطلحات موضوعية: medicine.medical_specialty, Patch-Clamp Techniques, Potassium Channels, Stereochemistry, Pyridines, Potassium, Vasodilator Agents, chemistry.chemical_element, Guanidines, Membrane Potentials, Adenosine Triphosphate, Internal medicine, medicine, Diazoxide, Potassium Channel Blockers, Animals, Patch clamp, Binding site, Cells, Cultured, Pharmacology, Membrane potential, Binding Sites, Sheep, Chemistry, Hyperpolarization (biology), Potassium channel, Electrophysiology, Kinetics, Endocrinology, Choroid Plexus, Choroid plexus, medicine.drug