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1
المؤلفون: Zhixiong Ye, Elizabeth T. Birzin, Meng-Hsin Chen, Louis Locco, Sheng-Shung Pong, Ravi P. Nargund, Rupa M. Parmar, Roy G. Smith, Ying-Duo Gao, Scott D. Feighner, Wanda W.-S. Chan, James M. Schaeffer, Arthur A. Patchett, Raman K. Bakshi, Allan D. Blake, Andrew D. Howard, Susan P. Rohrer
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:5-8
مصطلحات موضوعية: Models, Molecular, Agonist, Molecular model, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Receptors, Cell Surface, Carboxamide, Pharmacology, Biochemistry, Chemical synthesis, Receptors, G-Protein-Coupled, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Receptors, Ghrelin, Molecular Biology, Quinazolinone, Binding Sites, Human Growth Hormone, Chemistry, Organic Chemistry, In vitro, Rats, Kinetics, Drug Design, Quinazolines, Molecular Medicine, Secretagogue, Secretory Rate
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2
المؤلفون: James M. Schaeffer, Edward C. Hayes, Susan P. Rohrer, M. Dashkevicz, Allan D. Blake, Wanda W.-S. Chan, Rupa M. Parmar, Roy G. Smith
المصدر: Biochemical and Biophysical Research Communications. 263:276-280
مصطلحات موضوعية: Male, endocrine system, medicine.medical_specialty, Indoles, Growth-hormone-releasing hormone receptor, Somatotropic cell, Biophysics, Growth Hormone-Releasing Hormone, Biochemistry, Anterior pituitary, Pituitary Gland, Anterior, Thyrotropin-releasing hormone receptor, Internal medicine, medicine, Animals, Receptors, Somatostatin, Rats, Wistar, Molecular Biology, Dose-Response Relationship, Drug, Chemistry, Cell Biology, Growth hormone–releasing hormone, Amides, Growth hormone secretion, Rats, medicine.anatomical_structure, Somatostatin, Endocrinology, Growth Hormone, Corticotropic cell, hormones, hormone substitutes, and hormone antagonists
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3
المؤلفون: Steven M. Hutchins, James M. Schaeffer, Lihu Yang, Wanda W.-S. Chan, Ralph T. Mosley, Alex Pasternak, Min Shu, Sylvia J. Degrado, Scott C. Berk, Forrest Foor, Roy G. Smith, John M. Klopp, Sudha W. Mitra, Arthur A. Patchett, Sheng-Jian Cai, Kevin T. Chapman, Yusheng Xiong, Rupa M. Parmar, Dong-Ming Shen, Allan D. Blake, Elizabeth T. Birzin, Susan P. Rohrer, Edward C. Hayes
المصدر: Science. 282:737-740
مصطلحات موضوعية: endocrine system, medicine.medical_specialty, Molecular Sequence Data, Pharmacology, Biology, Ligands, Somatostatin Receptor Agonist, Cell Line, Islets of Langerhans, Mice, Pituitary Gland, Anterior, Cricetinae, Internal medicine, Insulin Secretion, medicine, Somatostatin receptor 3, Animals, Insulin, Somatostatin receptor 2, Somatostatin receptor 1, Amino Acid Sequence, Receptors, Somatostatin, Receptor, Cells, Cultured, Glucagon-like peptide 1 receptor, Multidisciplinary, Somatostatin receptor, Membrane Proteins, Glucagon, Amides, Rats, Endocrinology, Somatostatin, Models, Chemical, Drug Design, Growth Hormone, hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Roger M. Freidinger, Byron H. Arison, Roy G. Smith, Kevin T. Chapman, Kang Cheng, Arthur A. Patchett, Alexander Pasternak, Yanping Pan, Elizabeth T. Birzin, Rupa M. Parmar, Scott C. Berk, Maria A. de Souza Silva, Forrest Foor, Liangqin Guo, James M. Schaeffer, Tsuei-Ju Wu, Sudha W. Mitra, Bridgette S. Butler, Susan P. Rohrer, Edward C. Hayes, Lihu Yang, Ralph T. Mosley, Dennis J. Underwood
المصدر: Proceedings of the National Academy of Sciences. 95:10836-10841
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, Indoles, medicine.drug_class, CHO Cells, Biology, Insulin Antagonists, Mice, Cricetinae, Internal medicine, medicine, Somatostatin receptor 3, Animals, Humans, Insulin, Somatostatin receptor 2, Somatostatin receptor 1, Receptors, Somatostatin, Receptor, Multidisciplinary, Somatostatin receptor, Molecular Mimicry, Biological Sciences, Glucagon, Rats, Mice, Inbred C57BL, Endocrinology, Somatostatin, Growth Hormone, Benzimidazoles, Cyclase activity
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f2248ba0d424ebf80bd10e3290e6a51a
https://doi.org/10.1073/pnas.95.18.10836 -
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المؤلفون: Allan D. Blake, Rupa M. Parmar, Martin Köhler, James M. Schaeffer, Mathias Z. Strowski, Michael P. Dashkevicz, Hilary A. Wilkinson
المصدر: Neuroendocrinology. 75(6)
مصطلحات موضوعية: endocrine system, medicine.medical_specialty, Saccharomyces cerevisiae Proteins, Corticotropin-Releasing Hormone, Endocrinology, Diabetes and Metabolism, Adrenocorticotropic hormone, Binding, Competitive, Cell Line, Fungal Proteins, Iodine Radioisotopes, Cellular and Molecular Neuroscience, Corticotropin-releasing hormone, Radioligand Assay, fluids and secretions, Endocrinology, Adrenocorticotropic Hormone, Internal medicine, parasitic diseases, medicine, Cyclic AMP, Somatostatin receptor 2, Somatostatin receptor 1, Receptors, Somatostatin, Receptor, Endocrine and Autonomic Systems, Chemistry, Somatostatin receptor, fungi, GTPase-Activating Proteins, Somatostatin, Pituitary Gland, Somatostatin-28, Corticotropic cell, hormones, hormone substitutes, and hormone antagonists
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6
المصدر: Endocrinology. 141(1)
مصطلحات موضوعية: endocrine system, medicine.medical_specialty, Indoles, In Vitro Techniques, Naphthalenes, Glucagon, Insulin Antagonists, Islets of Langerhans, Mice, Endocrinology, Hormone Antagonists, Internal medicine, medicine, Somatostatin receptor 2, Animals, Receptors, Somatostatin, Glucagon-like peptide 1 receptor, Mice, Knockout, Somatostatin receptor, Chemistry, Pancreatic islets, Glucagon secretion, Amides, Stimulation, Chemical, Mice, Inbred C57BL, medicine.anatomical_structure, Somatostatin, Glucose, Somatostatin-28, Glucagon receptor family, hormones, hormone substitutes, and hormone antagonists
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::789f5e15be61584162f0a7eb40ce55a8
https://pubmed.ncbi.nlm.nih.gov/10614629 -
7
المؤلفون: Toshihiro Imaki, Yoko Kasagi, Michael P. Dashkevicz, Ping Yin, Ismail H. Zwain, Rupa M. Parmar, Armando Arroyo, Kensaku Sakae, Kengo Kawashima, Sun Mi Shin, James M. Schaeffer, Paula Amato, Anita C. Hansson, Inpyo Choi, Shiro Minami, Young Yang, Kun-yong Kim, Reiko Tokita, Tomoko Nakata, Hilary A. Wilkinson, Seung Hyun Han, Changmee Kim, Kwang Ho Pyun, Abba J. Kastin, Mathias Z. Strowski, Hyun Kim, Allan D. Blake, Samuel S.C. Yen, Martin Köhler, Jun Arita, Kjell Fuxe, Victoria Akerstrom
المصدر: Neuroendocrinology. 75:405-406
مصطلحات موضوعية: Cellular and Molecular Neuroscience, medicine.medical_specialty, Endocrinology, Traditional medicine, Endocrine and Autonomic Systems, business.industry, Endocrinology, Diabetes and Metabolism, Internal medicine, Medicine, business
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8
المؤلفون: Martin Köhler, Kun-yong Kim, Tomoko Nakata, Shiro Minami, Kjell Fuxe, Anita C. Hansson, Victoria Akerstrom, Hilary A. Wilkinson, Seung Hyun Han, Rupa M. Parmar, James M. Schaeffer, Armando Arroyo, Hyun Kim, Inpyo Choi, Mathias Z. Strowski, Kensaku Sakae, Yoko Kasagi, Abba J. Kastin, Kwang Ho Pyun, Paula Amato, Kengo Kawashima, Jun Arita, Allan D. Blake, Ismail H. Zwain, Toshihiro Imaki, Michael P. Dashkevicz, Young Yang, Changmee Kim, Samuel S.C. Yen, Ping Yin, Sun Mi Shin, Reiko Tokita
المصدر: Neuroendocrinology. 75:403-403
مصطلحات موضوعية: Cellular and Molecular Neuroscience, medicine.medical_specialty, Endocrinology, Index (economics), Endocrine and Autonomic Systems, Endocrinology, Diabetes and Metabolism, Internal medicine, medicine, Subject (documents), Medical physics, Psychology