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1دورية أكاديميةThe enzymatic activity of inositol hexakisphosphate kinase controls circulating phosphate in mammals
المؤلفون: Yusuke Moritoh, Shin-ichi Abe, Hiroki Akiyama, Akihiro Kobayashi, Ryokichi Koyama, Ryoma Hara, Shizuo Kasai, Masanori Watanabe
المصدر: Nature Communications, Vol 12, Iss 1, Pp 1-15 (2021)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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المؤلفون: Ryokichi Koyama, Mitsugi Ookawara, Yusuke Moritoh, Masanori Watanabe
المصدر: Molecular Pharmacology. 99:286-293
مصطلحات موضوعية: Blood Glucose, Male, 0301 basic medicine, Agonist, endocrine system, Pyridines, medicine.drug_class, medicine.medical_treatment, Allosteric regulation, CHO Cells, Glycemic Control, Pharmacology, Rats, Inbred WKY, Diabetes Mellitus, Experimental, Receptors, G-Protein-Coupled, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Piperidines, In vivo, Cricetinae, Free fatty acid receptor 1, Diabetes mellitus, medicine, Animals, Humans, Receptor, Dose-Response Relationship, Drug, business.industry, Insulin, medicine.disease, Rats, Dose–response relationship, 030104 developmental biology, Molecular Medicine, business, 030217 neurology & neurosurgery
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c81b58fb21dce5a8f6b01f184eae2ca1
https://doi.org/10.1124/molpharm.120.000168 -
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المؤلفون: Mitsugi Ookawara, Masanori Watanabe, Ryokichi Koyama, Satoshi Sasaki, Koji Watanabe, Yusuke Moritoh
المصدر: The FASEB Journal. 35
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Biochemistry, Allosteric regulation, Genetics, Glucose transporter, Fructose, Molecular Biology, Small molecule, Biotechnology
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4
المؤلفون: Ryokichi Koyama, Geza Ambrus-Aikelin, Darbi Witmer, Bi-Ching Sang, Yasunori Fukuda, Hidehisa Iwata, Hideyuki Nakagawa, Masaharu Nakayama, Yusuke Kamada
المصدر: ASSAY and Drug Development Technologies. 16:194-204
مصطلحات موضوعية: Orphan receptor, Sulfonamides, Reporter gene, Hydrocarbons, Fluorinated, Molecular Structure, Chemistry, Cholesterol binding, Drug Evaluation, Preclinical, Nuclear Receptor Subfamily 1, Group F, Member 3, Spodoptera, Pharmacology, Cholesterol, RAR-related orphan receptor gamma, Drug Discovery, Coactivator, Sf9 Cells, Animals, Humans, Th17 Cells, Molecular Medicine, Inverse agonist, lipids (amino acids, peptides, and proteins), Receptor, IC50
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59d9bc10dbf1390655dbeac60d89a052
https://doi.org/10.1089/adt.2018.852 -
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المؤلفون: Osamu Ujikawa, Yoko Morita, Kenichiro Shimokawa, Takayuki Hattori, Masahiro Ito, Tomoya Sameshima, Keiichiro Okuhira, Katsunori Nagai, Ikuo Fujimori, Yasuhiro Imaeda, Hiroshi Nara, Ryokichi Koyama, Mikihiko Naito, Youji Hayase, Nobuo Cho, Nobumichi Ohoka, Norihito Shibata, Osamu Sano
المصدر: Journal of Biological Chemistry. 293:6776-6790
مصطلحات موضوعية: 0301 basic medicine, Down-Regulation, Estrogen receptor, Antineoplastic Agents, X-Linked Inhibitor of Apoptosis Protein, Ligands, Inhibitor of apoptosis, Biochemistry, Mice, 03 medical and health sciences, 0302 clinical medicine, Ubiquitin, Animals, Humans, Molecular Biology, biology, Ligand, Chemistry, Estrogen Receptor alpha, Ubiquitination, Cell Biology, Xenograft Model Antitumor Assays, Cell biology, XIAP, Thiazoles, 030104 developmental biology, Proteasome, Protein Synthesis and Degradation, Apoptosis, 030220 oncology & carcinogenesis, Proteolysis, Cancer cell, MCF-7 Cells, biology.protein, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d71858240322a34c0d71fbf5734e371d
https://doi.org/10.1074/jbc.ra117.001091 -
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المؤلفون: Yuji Shimizu, Tomohiro Kawamoto, Ryokichi Koyama
المصدر: Biochemical Pharmacology. 140:105-114
مصطلحات موضوعية: 0301 basic medicine, Allosteric modulator, Pyridines, Recombinant Fusion Proteins, medicine.medical_treatment, media_common.quotation_subject, Green Fluorescent Proteins, Biology, Ligands, Second Messenger Systems, Biochemistry, Receptors, G-Protein-Coupled, 03 medical and health sciences, Allosteric Regulation, Downregulation and upregulation, Genes, Reporter, Homologous desensitization, Cyclic AMP, medicine, Humans, Tachyphylaxis, Internalization, Receptor, Protein Kinase Inhibitors, Rho-associated protein kinase, beta-Arrestins, Desensitization (medicine), G protein-coupled receptor, media_common, Feedback, Physiological, Pharmacology, Sulfonamides, rho-Associated Kinases, Amides, Molecular biology, Recombinant Proteins, Phenanthridines, Cell biology, Kinetics, Protein Transport, Zinc, HEK293 Cells, Pyrimidines, 030104 developmental biology, Gene Expression Regulation, Microscopy, Fluorescence
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المؤلفون: Nobumichi Ohoka, Norihito Shibata, Mikihiko Naito, Kenichiro Shimokawa, Nobuo Cho, Hiroshi Nara, Hirokazu Matsumoto, Osamu Sano, Ryokichi Koyama, Hisashi Fujita, Masahiro Ito, Katsunori Nagai, Yasuhiro Imaeda, Takayuki Hattori, Keiichiro Okuhira, Osamu Ujikawa, Mika Teratani
المصدر: Journal of Biological Chemistry. 292:4556-4570
مصطلحات موضوعية: 0301 basic medicine, BRD4, Gene knockdown, Estrogen receptor, Cell Biology, Biology, Inhibitor of apoptosis, Biochemistry, Cell biology, XIAP, Ubiquitin ligase, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Proteasome, Ubiquitin, Protein Synthesis and Degradation, 030220 oncology & carcinogenesis, biology.protein, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a81db1525450bb91feeaa74e7def011c
https://doi.org/10.1074/jbc.m116.768853 -
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المؤلفون: Naohiro Taya, Chien-Hung Chen, Tsuneo Oda, Bi-Ching Sang, Tomoya Yukawa, Takayuki Sato, Yoshi Nara, Noriko Uchiyama, Zenyu Shiokawa, Terufumi Takagi, Satoshi Yamamoto, Ayumu Sato, Ryokichi Koyama, Nobuyuki Negoro, Gyorgy Snell, Junya Shirai, Ryosuke Katsuyama, Takashi Imada, Yoshihiro Banno, Isaac Hoffman, Tetsuji Kawamoto, Mitsunori Kono, Robert J. Skene
المصدر: Journal of medicinal chemistry. 62(3)
مصطلحات موضوعية: Agonist, Drug Inverse Agonism, medicine.drug_class, Retinoic acid, Molecular Dynamics Simulation, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, RAR-related orphan receptor gamma, Drug Discovery, medicine, Inverse agonist, Structure–activity relationship, Animals, 030304 developmental biology, Orphan receptor, 0303 health sciences, Chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, 0104 chemical sciences, Cell biology, High-Throughput Screening Assays, 010404 medicinal & biomolecular chemistry, Design synthesis, Drug Design, Molecular Medicine, Th17 Cells
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المؤلفون: Yusuke Kamada, Masanori Miwa, Kotaro Sakamoto, Ryokichi Koyama, Akiyoshi Tani
المصدر: Biochemical and biophysical research communications. 503(3)
مصطلحات موضوعية: 0301 basic medicine, Vasoactive intestinal peptide, Biophysics, Peptide, Biosensing Techniques, CHO Cells, Ligands, Biochemistry, 03 medical and health sciences, Mice, Cricetulus, Peptide Library, Drug Discovery, Animals, Humans, Receptor, Molecular Biology, G protein-coupled receptor, chemistry.chemical_classification, Vasoactive intestinal peptide receptor, Cell Biology, Surface Plasmon Resonance, Cyclic peptide, Recombinant Proteins, Rats, 030104 developmental biology, chemistry, Pituitary Adenylate Cyclase-Activating Polypeptide, Receptors, Vasoactive Intestinal Peptide, Type II, VIPR1, VIPR2, Vasoactive Intestinal Peptide
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المؤلفون: Osamu Sano, Ryokichi Koyama, Osamu Ujikawa, Yoko Morita, Hiroshi Nara, Nobumichi Ohoka, Norihito Shibata, Mikihiko Naito, Takayuki Hattori, Nobuo Cho, Katsunori Nagai, Yasuhiro Imaeda
المصدر: Journal of medicinal chemistry. 61(2)
مصطلحات موضوعية: 0301 basic medicine, Male, Antineoplastic Agents, Chemistry Techniques, Synthetic, Protein degradation, Inhibitor of apoptosis, Ligands, Inhibitor of Apoptosis Proteins, 03 medical and health sciences, Prostate cancer, Structure-Activity Relationship, Ubiquitin, Cell Line, Tumor, Drug Discovery, medicine, Humans, Receptor, Cell Proliferation, biology, Chemistry, Prostatic Neoplasms, medicine.disease, Molecular biology, Cell biology, Androgen receptor, 030104 developmental biology, Apoptosis, A549 Cells, Receptors, Androgen, Proteolysis, biology.protein, Molecular Medicine, Drug Screening Assays, Antitumor, Protein ligand