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1
المؤلفون: Stefan Kavanagh, Julian A. Hudson, David S. Clarke, Alison Easter, Paul Schofield, Anne Ertan, Darren Mckerrecher, Hayley S. Brown, Suzanne S. Bowker, James S. Scott, Elizabeth A. Martin, David Laber, Philip A. MacFaul, Per H. Svensson, Joanne Teague, Andrew G. Leach, Kristin Goldberg, Katy J. Brocklehurst
المصدر: Journal of Medicinal Chemistry. 57:8984-8998
مصطلحات موضوعية: Male, hERG, Pharmacology, Receptors, G-Protein-Coupled, Sulfone, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Slice preparation, In vivo, Drug Discovery, Animals, Hypoglycemic Agents, Receptor, G protein-coupled receptor, Mice, Knockout, Oxadiazoles, biology, Ether-A-Go-Go Potassium Channels, In vitro, Mice, Inbred C57BL, Pyrimidines, Diabetes Mellitus, Type 2, chemistry, Toxicity, biology.protein, Molecular Medicine, Female, Epilepsy, Tonic-Clonic
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المؤلفون: Suzanne S. Bowker, Clive Green, Graeme R. Robb, Stephen Stokes, Nathaniel G. Martin, Anne Ertan, David G.A. Morgan, Christopher Sheldon, Alexander G. Dossetter, Robert D. M. Davies, David S. Clarke, Alastair J. H. Brown, William McCoull, Helen Pointon, Jane E. Moore, Mark L. Fenwick, Nicholas John Newcombe, Claire Newton, Jane L. Holmes, David J. Masters, Peter Barton, Jennifer Cameron
المصدر: Journal of Medicinal Chemistry. 57:6128-6140
مصطلحات موضوعية: Models, Molecular, medicine.medical_specialty, Drug Inverse Agonism, High-throughput screening, Pharmacology, Partial agonist, Structure-Activity Relationship, chemistry.chemical_compound, Internal medicine, Drug Discovery, medicine, Humans, Urea, Inverse agonist, Structure–activity relationship, Receptors, Ghrelin, Receptor, Dose-Response Relationship, Drug, Molecular Structure, digestive, oral, and skin physiology, Endocrinology, chemistry, Molecular Medicine, Ghrelin, Penetrant (biochemical), hormones, hormone substitutes, and hormone antagonists
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3دورية أكاديمية
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4
المؤلفون: W. Kleophas, B. Bieber, B. Robinson, J. Duttlinger, D. Fliser, G. Lonneman, L. Rump, R. Pisoni, F. Port, H. Reichel, R. Daniela, A. Ciocalteu, I. A. Checherita, I. Peride, D. M. Spataru, A. Niculae, K. Laetitia, K. Amna, D. Laurence, H.-A. Aoumeur, M. Flamant, J.-P. Haymann, E. Letavernier, E. Vidal-Petiot, J.-J. Boffa, F. Vrtovsnik, F. Bianco, G. Pessolano, M. Carraro, G. O. Panzetta, N. Ebert, J. Gaedeke, O. Jakob, M. Kuhlmann, P. Martus, M. Van der Giet, E. Scha ner, I. Khan, Y. Law, K. Turgutalp, O. Ozhan, E. Gok Oguz, A. Kiykim, C. Donadio, Z. N. Hatmi, M. Mahdavi-Mazdeh, E. Morales, V. Gutierrez-Millet, J. Rojas-Rivera, A. Huerta, E. Gutierrez, E. Gutierrez-Solis, N. Polanco, J. Caro, E. Gonza z, M. Praga, M. Marco Mayayo, J. Valdivielso, M. Marti z, E. Fernaez Giraez, G. Obrador, N. Olvera, D. Ortiz de la Pe, V. Gutie ez, A. Villa, B. Redal-Baigorri, K. Sombolos, D. Tsakiris, J. Boletis, D. Vlahakos, K. Siamopoulos, V. Vargiemezis, P. Nikolaidis, C. Iatrou, E. Dafnis, C. Argyropoulos, K. Xynos, D. Schock-Kusch, Y. Shulhevich, S. Geraci, J. Hesser, D. Stsepankou, S. Neudecker, S. Koenig, F. Hoecklin, J. Pill, N. Gretz, F. Schweda, A. Schreiber, K. Kudo, T. Konta, S. O. Choi, J. S. Kim, M. K. Kim, J. W. Yang, B. G. Han, P. Delanaye, E. Cavalier, I. Masson, M. Mehdi, M. Nicolas, B. Lambermont, B. Dubois, P. Damas, J.-M. Krzesinski, J. Morel, A. Lautrette, M. Christophe, A. Gagneux-Brunon, F. Anne, L. Fre (C)ric, S. Bevc, R. Ekart, R. Hojs, M. Gorenjak, L. Puklavec, N. Hashimoto, A. Suzuki, K. Mitsumoto, M. Shimizu, K. Niihata, A. Kawabata, Y. Sakaguchi, T. Hayashi, T. Shoji, N. Okada, Y. Tsubakihara, T. Hamano, C. Nakano, N. Fujii, Y. Obi, S. Mikami, K. Inoue, I. Matsui, Y. Isaka, H. Rakugi, V. Edvardsson, B. Siguron, M. Thorsteinsdottir, R. Palsson, J. Matsumoto, N. Miyazaki, I. Murata, G. Yoshida, K. Morishita, H. Ushikoshi, K. Nishigaki, S. Ogura, S. Minatoguchi, U. Werneke, M. Ott, E. Salander-Renberg, D. Taylor, B. Stegmayr, S. Surel, M. Wenzlova, G. Silva Junior, A. P. Vieira, A. Couto Bem, M. Alves, A. Torres, G. Meneses, A. Martins, A. Liborio, E. Daher, G. Gluhovschi, M. Modilca, L. Daminescu, C. Gluhovschi, S. Velciov, L. Petrica, F. Gadalean, C. Balgradean, H. H. Schmeiser, M. Kolesnyk, N. Stepanova, L. Surzhko, N. Stashevska, V. Filiopoulos, D. Hadjiyannakos, D. Arvanitis, K. Panagiotopoulos, D. Vlassopoulos, N. Kaesler, T. Schettgen, E. Magdeleyns, V. Brandenburg, C. Vermeer, J. Floege, T. Kr, O. Randone, M. Ferraresi, E. Aroasio, A. Depascale, S. Scognamiglio, V. Consiglio, G. B. Piccoli, L. V. Jensen, S. Lizakowski, P. Rutkowski, L. Tylicki, M. Renke, B. Sulikowska, R. Donderski, R. Bednarski, Z. Heleniak, M. Przybylska, J. Manitius, B. Rutkowski, L. Bobrova, N. Kozlovskaya, K. Kanayama, M. Hasegawa, F. Kitagawa, J. Ishii, Y. Yuzawa, K. Tanaka, K. Sakai, S. Hara, Y. Suzuki, Y. Tanaka, A. Aikawa, F. Hinoshita, N. Hamano, E. Sasaki, A. Kato, T. Katsuki, A. Katsuma, E. Imai, M. Shibata, M. Tada, T. Shimbo, Y. Kikuchi, S. Oka, T. Muramatsu, N. Yanagisawa, K. Fukutake, Y. Yamamoto, A. Ajisawa, K. Tsuchiya, K. Nitta, M. Ando, X. Liang, P. Wang, Z. Liu, Z. Zhao, V. Luyckx, S. Bowker, A. Miekle, E. Toth, R. Heguilen, A. Malvar, R. Hermes, L. Cohen, G. Muguerza, B. Lococo, A. Bernasconi, O. Loboda, I. Dudar, V. Krot, V. Alekseeva, M. Ichinose, N. Sasagawa, K. Toyama, A. Saito, Y. Kayamori, D. Kang, H. W. Kim, K. Yoshioka, M. Hara, K. Ohashi, A. Maksudova, T. Khalfina, A. Cuoghi, E. Bellei, M. Caiazzo, S. Bergamini, G. Palladino, E. Monari, A. Tomasi, E. Loiacono, R. Camilla, V. Dapr, L. Morando, R. Gallo, L. Peruzzi, M. Conrieri, M. Bianciotto, F. M. Bosetti, R. Coppo, L. DI Lullo, F. Floccari, R. Rivera, A. Granata, R. Faiola, C. Feliziani, A. Villani, M. Malaguti, A. Santoboni, K. Kyriaki, J. Droulias, M. Bogdanova, V. V. Rameev, A. H. Simonyan, L. V. Kozlovskaya, M. R. Altiparmak, S. Trabulus, N. Akalin, A. S. Yalin, A. Esenkaya, S. F. Yalin, K. Serdengeae(C), D. Arita, T. Cunha, J. Perez, M. Sakata, L. Arita, M. Nogueira, Z. Jara, N. Souza, D. Casarini, M. Metzger, M. Vallet, A. Karras, M. Froissart, B. Stengel, P. Houillier, K. Paul, D. Kretzschmar, A. Yilmaz, B. Ba hlein, S. Titze, H.-R. Figulla, G. Wolf, M. Busch, Y. Korotchaeva, N. Gordovskaya, L. Kozlovskaya, K. P. Ng, P. Sharma, S. Stringer, M. Jesky, M. Dutton, C. Ferro, P. Cockwell, S. J. Moon, S. C. Lee, S. Y. Yoon, J. E. Lee, S. J. Han, B. Anna, T. Kirsch, L. Svjetlana, P. Joon-Keun, B. Jan, K. Johanna, H. Haller, M. Haubitz, A. Smirnov, I. Kayukov, N. Rafrafi, O. Degtereva, V. Dobronravov, M. Koch, H. Stefan, G. Dika, M.-H. Antoine, C. Husson, J. Kos, M. Milic, M. Fucek, D. Cvoriocec, M.-F. Bourgeade, J. L. Nortier, B. Jelakovic, E. H. Nawal, M. Naoufal, M. Nabila, E. M. Fadwa, E. K. Salma, B. Nisrine, Z. Mohamed, M. Guislaine, B. Mohamed Gharbi, R. Benyounes, G. G. Sotila, R. Sorin, D. Irina Magdalena, C. Roxana, R. Claudia, F. Correa Barcellos, P. H. Hallal, M. Bohlke, F. Boscolo Del Vechio, A. Reges, I. Santos, G. Mielke, M. Fortes, B. Antunez, M. Laganovic, I. Vukovic Lela, S. Karanovic, J. Seric, V. Premuic, M. Fitrek, L. Fodor, T. Meljkovic Vrkic, V. Bansal, D. Hoppensteadt, J. Fareed
المصدر: Nephrology Dialysis Transplantation. 27:ii96-ii120
مصطلحات موضوعية: Transplantation, medicine.medical_specialty, Nephrology, business.industry, Medicine, Medical physics, Clinical nephrology, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d74085d4cdfbd41ad4b5e02e055f5d3c
https://doi.org/10.1093/ndt/gfs215 -
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المؤلفون: Peter William Rodney Caulkett, Scott Boyd, Clifford David Jones, Gordon S. Currie, Sarah Lackie, Emma Grange, Craig Johnstone, Barry R. Hayter, Harold Gaskin, Christopher D. Davies, Darren Mckerrecher, Rod B. Hargreaves, Mark L. Fenwick, Roger James, Rayner John Wall, Keith M. Johnson, Joanne V. Allen, Rolf Peter Walker, Suzanne S. Bowker
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:2103-2106
مصطلحات موضوعية: Clinical Biochemistry, Drug Evaluation, Preclinical, Enzyme Activators, Pharmaceutical Science, Biochemistry, Chemical synthesis, In vivo, Glucokinase, Drug Discovery, Animals, Rats, Wistar, Kinase activator, Molecular Biology, Biological evaluation, Activator (genetics), Chemistry, Organic Chemistry, Biological activity, Rats, Enzyme Activation, Thiazoles, Lipophilicity, Molecular Medicine, Female
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المؤلفون: James S. Scott, Nidhal Selmi, Joanne deSchoolmeester, Suzanne S. Bowker, Amanda Rees, Rachel M. Mayers, Derek Ogg, Paul Schofield, Elaine Kilgour, John G. Swales, Stefan Gerhardt, William McCoull, Martin J. Packer, David J. Hargreaves, Nicholas John Newcombe, John Revill, Adele Lloyd, Paul Robert Owen Whittamore
المصدر: Journal of medicinal chemistry. 55(12)
مصطلحات موضوعية: Male, Models, Molecular, Niacinamide, Stereochemistry, Protein Conformation, Carboxylic acid, Administration, Oral, Biological Availability, Substrate Specificity, Acetic acid, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Dogs, Piperidines, 11β-hydroxysteroid dehydrogenase type 1, Amide, 11-beta-Hydroxysteroid Dehydrogenase Type 1, Drug Discovery, Potency, Animals, Humans, Enzyme Inhibitors, chemistry.chemical_classification, biology, Chemistry, Drug discovery, Bioavailability, Rats, Nicotinic agonist, Biochemistry, biology.protein, Molecular Medicine, hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Graeme C. Moody, Alleyn T. Plowright, J. Matthew Wood, Matthew S. Addie, Scott Boyd, Paul D. Kemmitt, David Whalley, Chris Sheldon, Andrew V. Turnbull, Stephen Chapman, Andrew G. Leach, Pablo Morentin Gutierrez, Paul Schofield, Linda K. Buckett, William McCoull, Nicholas John Newcombe, Alan Martin Birch, Chloe Jenner, Martin J. Packer, Thorsten Nowak, Robert D. M. Davies, Susan Birtles, Steven Wang, Steve Stokes, Roger John Butlin, Suzanne S. Bowker, John Revill, Craig S. Donald, Clive Green
المصدر: Bioorganicmedicinal chemistry letters. 22(12)
مصطلحات موضوعية: Quantitative structure–activity relationship, High-throughput screening, Carboxylic acid, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Oxadiazole, Quantitative Structure-Activity Relationship, Ligands, Biochemistry, chemistry.chemical_compound, Mice, Dogs, In vivo, Drug Discovery, Diabetes Mellitus, Potency, Animals, Humans, Hypoglycemic Agents, Diacylglycerol O-Acyltransferase, Obesity, Enzyme Inhibitors, Molecular Biology, PK/PD models, chemistry.chemical_classification, Oxadiazoles, Chemistry, Organic Chemistry, Combinatorial chemistry, High-Throughput Screening Assays, Rats, Lipophilic efficiency, Drug Design, Molecular Medicine, Half-Life
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المؤلفون: A. J. Westphal, A. Allbrink, C. Allen, S. Bajt, R. Bastien, H. Bechtel, P. Bleuet, J. Borg, S. Bowker, F. Brenker, J. Bridges, D. E. Brownlee, M. Burchell, M. Burghammer, A. L. Butterworth, A. Campanile, P. Cloetens, G. Cody, T. Ferroir, K. Ferrari, C. Floss, G. J. Flynn, D. Frank, Z. Gainsforth, E. Grün, M. Harmer, P. Hoppe, A. Kearsley, S. Kulkarni, B. Lai, L. Lemelle, H. Leroux, R. Lettieri, W. Marchant, B. McCreadie, L. R. Nittler, R. Ogliore, F. Postberg, C. Rigamonti, S. A. Sandford, S. Schmitz, G. Silversmit, A. Simionovici, G. Sperry, R. Srama, F. Stadermann, T. Stephan, R. M. Stroud, J. Susini, S. Sutton, V. Thompson, R. Toucoulou, M. Trieloff, P. Tsou, A. Tsuchiyama, T. Tyliczszak, B. Vekemans, L. Vincze, J. Warren, T. Yahnke, D. Zevin, M. E. Zolensky, Melissa Denecke, Clive T. Walker
المصدر: AIP Conference Proceedings.
مصطلحات موضوعية: Interstellar medium, Physics, X-ray spectroscopy, Beamline, law, Infrared, X-ray fluorescence, Infrared cirrus, Astrophysics, Synchrotron, law.invention, Cosmic dust
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9دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
10دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل.