-
1دورية أكاديمية
المؤلفون: Florence Ecoeur, Jessica Weiss, Klemens Kaupmann, Samuel Hintermann, David Orain, Christine Guntermann
المصدر: Frontiers in Immunology, Vol 10 (2019)
مصطلحات موضوعية: retinoic acid receptor-related-orphan-receptor-gamma t, nuclear hormone receptor, T helper 17 differentiation, IL-17, autoimmunity, keratinocytes, Immunologic diseases. Allergy, RC581-607
وصف الملف: electronic resource
-
2دورية أكاديمية
المؤلفون: Ulf Guendisch, Jessica Weiss, Florence Ecoeur, Julia Christina Riker, Klemens Kaupmann, Joerg Kallen, Samuel Hintermann, David Orain, Janet Dawson, Andreas Billich, Christine Guntermann
المصدر: PLoS ONE, Vol 12, Iss 11, p e0188391 (2017)
وصف الملف: electronic resource
-
3دورية أكاديمية
المؤلفون: Francesca Montarolo, Chiara Raffaele, Simona Perga, Serena Martire, Annamaria Finardi, Roberto Furlan, Samuel Hintermann, Antonio Bertolotto
المصدر: PLoS ONE, Vol 9, Iss 9, p e108791 (2014)
وصف الملف: electronic resource
-
4
المؤلفون: Samuel Hintermann, Andreas Marzinzik, Johannes Ottl, Joerg Kallen, Therese-Marie Stachyra, Patrick C. Reid, Stephan Ruetz, Anselm F. L. Schneider, Christian P. R. Hackenberger, Christoph E. Dumelin, Sebastien Ripoche
المصدر: RSC Chemical Biology
مصطلحات موضوعية: chemistry.chemical_classification, biology, Chemistry, Stereochemistry, Drug discovery, Peptide, Ligand (biochemistry), Biochemistry, Genetics and Molecular Biology (miscellaneous), Biochemistry, Cyclic peptide, Chemistry (miscellaneous), biology.protein, Mdm2, Macrocyclic ligand, Pharmacophore, Molecular Biology, Intracellular
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b79c0089311703a726113d94f5b84104
http://europepmc.org/articles/PMC8637822 -
5
المؤلفون: Strang Ross Sinclair, Markus Streiff, Daniel J. McKay, Johannes Ottl, Andreas Billich, Claudia Betschart, Stephanie Harlfinger, Eloísa Jiménez-Núñez, Nigel Graham Cooke, Christine Guntermann, Markus Voegtle, Janet Dawson, Samuel Hintermann, Klemens Kaupmann, Rowan Stringer, Christian Beerli, Nathalie Gobeau, Juergen Wagner, Klemens Hoegenauer, Joerg Kallen, Peter Ertl
المصدر: Journal of Medicinal Chemistry. 62:10816-10832
مصطلحات موضوعية: chemistry.chemical_classification, Orphan receptor, 0303 health sciences, Chemistry, Carboxylic acid, Retinoic acid, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, Proinflammatory cytokine, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, In vivo, Lipophilic efficiency, RAR-related orphan receptor gamma, Drug Discovery, Molecular Medicine, 030304 developmental biology, ADME
-
6
المؤلفون: John Joslin, Jerome Giovannoni, John I. Manchester, Eugen Lounkine, Douglas S. Auld, Nikolas Fechner, Philipp Krastel, Caroline Engeloch, Jutta Blank, Manuel Schwarze, Ansgar Schuffenhauer, Nikolaus Stiefl, Johanna M. Jansen, Nadine Schneider, Lauren G. Monovich, Simona Cotesta, Michael Shultz, Samuel Hintermann, Daniel K. Baeschlin, Christoph Gaul, Anna Paola Pelliccioli
المصدر: Journal of medicinal chemistry. 63(23)
مصطلحات موضوعية: 0303 health sciences, Chemistry, Drug Evaluation, Preclinical, Structural diversity, Grid, computer.software_genre, 01 natural sciences, Small molecule, 0104 chemical sciences, Deck, High-Throughput Screening Assays, Small Molecule Libraries, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Ranking, Drug Design, Drug Discovery, Redundancy (engineering), Molecular Medicine, Data mining, computer, 030304 developmental biology
-
7
المؤلفون: Klemens, Hoegenauer, Joerg, Kallen, Eloísa, Jiménez-Núñez, Ross, Strang, Peter, Ertl, Nigel G, Cooke, Samuel, Hintermann, Markus, Voegtle, Claudia, Betschart, Daniel J J, McKay, Juergen, Wagner, Johannes, Ottl, Christian, Beerli, Andreas, Billich, Janet, Dawson, Klemens, Kaupmann, Markus, Streiff, Nathalie, Gobeau, Stephanie, Harlfinger, Rowan, Stringer, Christine, Guntermann
المصدر: Journal of medicinal chemistry. 62(23)
مصطلحات موضوعية: Male, Models, Molecular, Dose-Response Relationship, Drug, Molecular Structure, Imidazoles, Administration, Oral, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, Drug Design, Fluorescence Resonance Energy Transfer, Animals, Female, Hypersensitivity, Delayed, Half-Life
-
8
المؤلفون: Christine Guntermann, Janet Dawson, Anna Vulpetti, Andreas Billich, Rowan Stringer, Johannes Ottl, Samuel Hintermann, Henri Mattes, Eric Vangrevelinghe, Nigel Graham Cooke, Klemens Kaupmann, Romain M. Wolf, Juergen Wagner, Klemens Hoegenauer, Joerg Kallen, David Orain, David Carcache
المصدر: Journal of Medicinal Chemistry. 61:6724-6735
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Drug Inverse Agonism, Inflammation, 01 natural sciences, 03 medical and health sciences, Transcription (biology), In vivo, RAR-related orphan receptor gamma, Catalytic Domain, Drug Discovery, medicine, Animals, Inverse agonist, Transcription factor, 010405 organic chemistry, Drug discovery, Chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, 0104 chemical sciences, Cell biology, Disease Models, Animal, 030104 developmental biology, Molecular Medicine, Female, medicine.symptom
-
9
المؤلفون: Christine Guntermann, Juergen Wagner, David Orain, Andreas Billich, Joerg Kallen, Samuel Hintermann, Janet Dawson, Rowan Stringer, Henri Mattes, Klemens Kaupmann, David Carcache, Anna Vulpetti
المصدر: ChemMedChem. 11:2640-2648
مصطلحات موضوعية: 0301 basic medicine, Imidazopyridine, Drug Inverse Agonism, Pyridines, Receptors, Retinoic Acid, Stereochemistry, medicine.medical_treatment, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Biochemistry, Inhibitory Concentration 50, 03 medical and health sciences, Pharmacokinetics, RAR-related orphan receptor gamma, Drug Discovery, medicine, Animals, Humans, Potency, Inverse agonist, General Pharmacology, Toxicology and Pharmaceutics, Transcription factor, Cells, Cultured, Binding Sites, Molecular Structure, Chemistry, Interleukin-17, Organic Chemistry, Imidazoles, Nuclear Receptor Subfamily 1, Group F, Member 3, Triazoles, Rats, 030104 developmental biology, Cytokine, Molecular Medicine, Protein Binding
-
10
المؤلفون: Arndt Meyer, Murali Chebrolu, Christine E. Gee, Grit Laue, Markus Fendt, Laura H. Jacobson, Sangamesh Badiger, Samuel Hintermann, Chetan Pandit, Simona Cotesta, Claudia Betschart, Daniel Hoyer, Vinod D. Chaudhari, Dirk Behnke, Trixie Wagner
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:5555-5560
مصطلحات موضوعية: Pyridines, High-throughput screening, Clinical Biochemistry, Dual Orexin Receptor Antagonists, Administration, Oral, Pharmaceutical Science, Pharmacology, Crystallography, X-Ray, Doras, Biochemistry, Mice, Drug Discovery, Animals, Molecular Biology, G protein-coupled receptor, Molecular Structure, biology, Chemistry, Drug discovery, Orexin Receptor Antagonists, Organic Chemistry, biology.organism_classification, Orexin, Pyrazoles, Molecular Medicine, Administration, Intravenous, Protein Binding