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1
المؤلفون: Junliang Hao, James Beck, Xin Zhou, Gregory L. Lackner, Richard Johnston, Matt Reinhard, Paul Goldsmith, Sean Hollinshead, Veronique Dehlinger, Sandra A. Filla, Xu-shan Wang, Jeffery Richardson, Maria Posada, Mike Mohutsky, Doug Schober, Jason S. Katner, Qi Chen, Bingjie Hu, David M. Remick, David A. Coates, Brian M. Mathes, Mai K. Hawk, Kjell A. Svensson, Erik Hembre
المصدر: Journal of Medicinal Chemistry. 65:3786-3797
مصطلحات موضوعية: Neuroprotective Agents, Allosteric Regulation, Receptors, Dopamine D1, Drug Discovery, Cytochrome P-450 CYP3A, Cytochrome P-450 CYP3A Inhibitors, Humans, Molecular Medicine, Drug Interactions
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2
المؤلفون: Yao-Chang Xu, Brian Michael Mathes, John Mehnert Schaus, Qi Chen, Maria-Jesus Blanco, Suzanne E. Nutter, David L. Nelson, Deanna Piatt Zacherl, Sidney Xi Liang, Sandra Ann Filla, Wendy H. Gough, Cohen Michael Philip, Kevin John Hudziak, Bai-Ping Ying, Deyi Zhang, Joseph H. Krushinski, Daniel Timothy Kohlman, Frantz Victor, David B. Wainscott
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:4337-4341
مصطلحات موضوعية: chemistry.chemical_classification, Indole test, Ketone, Bicyclic molecule, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Receptor agonist activity, 5-HT1F receptor, Biochemistry, chemistry.chemical_compound, Amide, Drug Discovery, Molecular Medicine, Moiety, Molecular Biology
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3
المؤلفون: Brian M. Arnold, Miriam del Prado, Smriti Iyengar, Edward L. Mattiuz, Zhipei Wu, Mark A. Winter, David Bleakman, Ken H. Ho, Ann Marie L. Ogden, Paul L. Ornstein, Carrie K. Jones, Sandra Ann Filla, Brian Michael Mathes, Michael Gregory Bell, Douglas Richard Stack, Ana Maria Escribano, Thomas J. Bleisch, Ana I. Mateo, Kevin John Hudziak, Andrew Alt, Rosa Maria A. Simmons, Harlan E. Shannon, Robert E. Stratford, Jose A. Martinez-Perez, Esteban Dominguez, Ana M. Castaño
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:6459-6462
مصطلحات موضوعية: Molecular Sequence Data, Clinical Biochemistry, Administration, Oral, Pain, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Receptors, Kainic Acid, Oral administration, In vivo, Drug Discovery, Animals, Prodrugs, Amino Acid Sequence, Molecular Biology, Benzoic acid, chemistry.chemical_classification, Chemistry, Organic Chemistry, Haplorhini, Prodrug, Isoquinolines, Amino acid, Disease Models, Animal, Molecular Medicine
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4
المؤلفون: Gustavo Pascual, Smriti Iyengar, Gregory A. Stephenson, Laura J. Martin, Sandra Ann Filla, Craig E. Thomas, Susan K. Hemrick-Luecke, Kirk W. Johnson, Jikesh Arvind Shah, Eric George Tromiczak, Magnus Wilhelm Walter, Karsten Fynboe, Lance Allen Pfeifer, Mark A. Muhlhauser, Juan A. Rincón, Nicolas Dreyfus, Chunjin Ding, Jia Shaojuan, María Luz de la Puente, Beverly A. Heinz, Lee A. Phebus, Michael P. Johnson, Simon James Richards, Thomas J. Perun, Michael J. McCoy, Pilar Lopez, Hamideh Zarrinmayeh, Thierry Masquelin, Rosa Maria A. Simmons, Douglas Linn Gernert, Oscar de Frutos, Elizabeth M. Joshi, Denise Morrow, Wayne W. Weber, Anette M. Johansson, Linda K. Thompson, Eric P. Seest, Valentina O. Badescu, Javier Mendiola, Jason K. Myers, Patrick L. Love
المصدر: ACS Medicinal Chemistry Letters. 4:560-564
مصطلحات موضوعية: biology, business.industry, Organic Chemistry, Chronic pain, Pharmacology, Inhibitory postsynaptic potential, medicine.disease, Biochemistry, Norepinephrine reuptake inhibitor, Norepinephrine transporter, In vivo, Drug Discovery, medicine, biology.protein, Serotonin, Reuptake inhibitor, business, ADME
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5
المؤلفون: Deyi, Zhang, Maria-Jesus, Blanco, Bai-Ping, Ying, Daniel, Kohlman, Sidney X, Liang, Frantz, Victor, Qi, Chen, Joseph, Krushinski, Sandra A, Filla, Kevin J, Hudziak, Brian M, Mathes, Michael P, Cohen, DeAnna, Zacherl, David L G, Nelson, David B, Wainscott, Suzanne E, Nutter, Wendy H, Gough, John M, Schaus, Yao-Chang, Xu
المصدر: Bioorganicmedicinal chemistry letters. 25(19)
مصطلحات موضوعية: Structure-Activity Relationship, Dose-Response Relationship, Drug, Molecular Structure, Piperidines, Benzamides, Drug Discovery, Humans, Quantum Theory, Serotonin 5-HT1 Receptor Agonists, Receptors, Serotonin, 5-HT1
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6
المؤلفون: Edward L. Mattiuz, Ann Marie L. Ogden, Ana M. Castaño, Zhipei Wu, Robert E. Stratford, E. Dominguez, Thomas J. Bleisch, Brian Michael Mathes, Brian M. Arnold, David Bleakman, Smriti Iyengar, Rosa Maria A. Simmons, Harlan E. Shannon, Sandra Ann Filla, Jose A. Martinez-Perez, Douglas Richard Stack, Ana I. Mateo, Miriam del Prado, Kevin John Hudziak, Andrew Alt, Michael Gregory Bell, Carrie K. Jones, Paul L. Ornstein, Jennifer L. Buckmaster, Ana Maria Escribano, Mark A. Winter, Ken H. Ho
المصدر: Journal of Medicinal Chemistry. 48:4200-4203
مصطلحات موضوعية: Analgesic, Biological Availability, Pain, Kainate receptor, Pharmacology, Cell Line, Receptors, Kainic Acid, Drug Discovery, Animals, Humans, Receptors, AMPA, Amino Acids, Receptor, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, chemistry.chemical_classification, Analgesics, Chemistry, Glutamate receptor, Antagonist, Prodrug, Recombinant Proteins, Rats, Amino acid, Disease Models, Animal, Spinal Cord, Biochemistry, Hyperalgesia, Molecular Medicine, Licking
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7
المؤلفون: David B. Wainscott, John Mehnert Schaus, Wendy H. Gough, Yao-Chang Xu, Brian Michael Mathes, John M. Zgombick, Sandra Ann Filla, David L. Nelson, Suzanne E. Nutter, Kevin John Hudziak, Theresa Branchek
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:167-170
مصطلحات موضوعية: Indole test, Agonist, Bicyclic molecule, Pyridines, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, 5-HT1F receptor, Biochemistry, Chemical synthesis, Serotonin Receptor Agonists, chemistry.chemical_compound, chemistry, Receptors, Serotonin, Drug Discovery, medicine, Molecular Medicine, Bioisostere, Receptor, Molecular Biology, Protein Binding
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8
المؤلفون: John Mehnert Schaus, Lee A. Phebus, John M. Zgombick, David B. Wainscott, Kirk W. Johnson, Kathryn W. Schenck, Brian Michael Mathes, Marlene L. Cohen, David L. Nelson, Jon A. Erickson, Sandra Ann Filla, Theresa A Branchek
المصدر: Journal of Medicinal Chemistry. 46:3060-3071
مصطلحات موضوعية: Agonist, Pyrimidine, Polyunsaturated Alkamides, Pyridines, medicine.drug_class, Stereochemistry, Migraine Disorders, Administration, Oral, In Vitro Techniques, Chemical synthesis, Cell Line, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, medicine, Animals, Structure–activity relationship, Pyrroles, Saphenous Vein, Trigeminal Nerve, Receptor, 5-HT receptor, Bicyclic molecule, Chemistry, Blood Proteins, Bridged Bicyclo Compounds, Heterocyclic, Serotonin Receptor Agonists, Vasoconstriction, Receptors, Serotonin, Molecular Medicine, Rabbits, Acetamide
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9
المؤلفون: Ken H. Ho, Edward L. Mattiuz, Ann Marie L. Ogden, Brian Michael Mathes, Ana I. Mateo, David Bleakman, Kevin John Hudziak, Donna K. Dieckman, Sandra Ann Filla, Mark A. Winter, Thomas J. Bleisch, Ana Maria Escribano, Paul L. Ornstein, Kirk W. Johnson, Douglas Richard Stack, Amy Clemens-Smith, Miriam del Prado, Ana M. Castaño, Mary A. Katofiasc, Robert E. Stratford, E. Dominguez, Michael Gregory Bell, Lee A. Phebus, Jose A. Martinez-Perez
المصدر: Journal of Medicinal Chemistry. 45:4383-4386
مصطلحات موضوعية: Stereochemistry, Migraine Disorders, Carboxylic Acids, Administration, Oral, Biological Availability, Kainate receptor, Pharmacology, Cell Line, Radioligand Assay, Receptors, Kainic Acid, Drug Discovery, medicine, Animals, Humans, Prodrugs, Rats, Wistar, Receptor, Dose-Response Relationship, Drug, Chemistry, Antagonist, Glutamate receptor, Esters, Biological activity, Prodrug, Isoquinolines, Rats, Disease Models, Animal, Mechanism of action, Competitive antagonist, Acute Disease, Molecular Medicine, Calcium, medicine.symptom, Excitatory Amino Acid Antagonists
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10
المؤلفون: Satoru Masamune, Sandra A. Filla, Jinhua J. Song, Lihren Chen
المصدر: Tetrahedron Letters. 40:5449-5453
مصطلحات موضوعية: chemistry.chemical_compound, Natural product, chemistry, Aldol reaction, Stereochemistry, Organic Chemistry, Drug Discovery, Organic chemistry, Stereoselectivity, Discodermolide, Alkylation, Biochemistry