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المؤلفون: Sandra Johannsen, Robin M. Gierse, Aleksandra Olshanova, Ellie Smerznak, Christian Laggner, Lea Eschweiler, Zahra Adeli, Rawia Hamid, Alaa Alhayek, Norbert Reiling, Jörg Haupenthal, Anna K. H. Hirsch
المساهمون: Chemical Biology 2
المصدر: ChemMedChem, 18(11):e202200590. WILEY-V C H VERLAG GMBH
مصطلحات موضوعية: Pharmacology, Drug discovery, 2-C-methyl-D-erythritol 4-phosphate pathway, Organic Chemistry, inhibitors, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, 1-deoxy-D-xylulose 5-phosphate synthase, neural networks, Biochemistry
وصف الملف: application/pdf
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المؤلفون: Ravindra P. Jumde, Gwenaëlle Jézéquel, Margarida Saramago, Nicolas Frank, Sebastian Adam, Marta V. Cunha, Chantal Bader, Antonia P. Gunesch, Natalie M. Köhler, Sandra Johannsen, Thomas Pietschmann, Rute G. Matos, Rolf Müller, Cecilia M. Arraiano, Anna K. H. Hirsch
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3b23a97626810e53c4928ed251167a25
https://doi.org/10.26434/chemrxiv-2023-kpmj5 -
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المؤلفون: Di Zhu, Sandra Johannsen, Tiziana Masini, Céline Simonin, Jörg Haupenthal, Boris Illarionov, Anastasia Andreas, Mahendra Awale, Robin M. Gierse, Tridia van der Laan, Ramon van der Vlag, Rita Nasti, Mael Poizat, Eric Buhler, Norbert Reiling, Rolf Müller, Markus Fischer, Jean-Louis Reymond, Anna K. H. Hirsch
المساهمون: Stratingh Institute of Chemistry, Chemical Biology 2
المصدر: Chemical Science, 13(36), 10686-10698. ROYAL SOC CHEMISTRY
Zhu, Di; Johannsen, Sandra; Masini, Tiziana; Simonin, Céline; Haupenthal, Jörg; Illarionov, Boris; Andreas, Anastasia; Awale, Mahendra; Gierse, Robin M; van der Laan, Tridia; van der Vlag, Ramon; Nasti, Rita; Poizat, Mael; Buhler, Eric; Reiling, Norbert; Müller, Rolf; Fischer, Markus; Reymond, Jean-Louis; Hirsch, Anna K H (2022). Discovery of novel drug-like antitubercular hits targeting the MEP pathway enzyme DXPS by strategic application of ligand-based virtual screening. Chemical Science, 13(36), pp. 10686-10698. The Royal Society of Chemistry 10.1039/d2sc02371g <http://dx.doi.org/10.1039/d2sc02371g>مصطلحات موضوعية: DXPS, ligand-based virtual screening, Tuberculosis, MEP, 540 Chemie, 540 Chemistry, 570 Life sciences, biology, General Chemistry, 580 Plants (Botany), Settore CHIM/08 - Chimica Farmaceutica, 570 Biowissenschaften, Biologie
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d037a73a79e9b4607948d4bb961dcdb1
https://research.rug.nl/en/publications/47d91e4b-c3e0-48f1-b774-6f2c690412a0 -
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المؤلفون: Sandra Johannsen, Robin M. Gierse, Arne Krüger, Rachel L. Edwards, Vittoria Nanna, Anna Fontana, Di Zhu, Tizina Masini, Lais Pessanha de Carvalho, Mael Poizat, Bart Kieftenbelt, Dana M. Hodge, Sophie Alvarez, Daan Bunt, Kamila Anna Meissner, Edmarcia Elisa de Souza, Melloney Dröge, Bernard van Vliet, Jack de Hartog, Michael C. Hutter, Jana Held, Audrey R. Odom John, Carsten Wrenger, Anna K. H. Hirsch
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::968d2b347432557d44f960aef4313c60
https://doi.org/10.26434/chemrxiv-2022-npslc -
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المؤلفون: Alaa Alhayek, Christian Nehls, Philipp J. Neusens, Walid A. M. Elgaher, Zhoor Hamid, Ravindra P. Jumde, Jörg Haupenthal, Melissa Guardigni, Norbert Reiling, Di Zhu, Robin M. Gierse, Anna K. H. Hirsch, Sandra Johannsen
المساهمون: Chemical Biology 2, HIPS, Helmholtz-Institut für Pharmazeutische Forschung Saarland, Universitätscampus E8.1 66123 Saarbrücken, Germany.
المصدر: Chemical Science, 12(22), 7775-7785. ROYAL SOC CHEMISTRY
Chemical Science
Chemical science
Englandمصطلحات موضوعية: Chemistry, 010405 organic chemistry, Dynamic combinatorial chemistry, Anti infectives, General Chemistry, Computational biology, 010402 general chemistry, 01 natural sciences, 0104 chemical sciences, 1-deoxy-D-xylulose-5-phosphate synthase
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2113aa57d97261e800b50866f049b04b
https://research.rug.nl/en/publications/a2d48f55-2cb5-45ff-a034-9f6c9ad79496 -
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المؤلفون: Sandra Johannsen, Di Zhu, Alaa Alhayek, Melissa Guardigni, Robin M. Gierse, Jörg Haupenthal, Walid A. M. Elgaher, Ravindra P. Jumde, Zhoor Hamed, Anna K. H. Hirsch
المصدر: ChemRxiv
مصطلحات موضوعية: Chemistry, Drug discovery, Dynamic combinatorial chemistry, Anti infectives, Computational biology, Non-mevalonate pathway, 1-deoxy-D-xylulose-5-phosphate synthase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9f274e6ab3d8d6fca583c9ae37e69461
https://doi.org/10.26434/chemrxiv.12681761 -
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المؤلفون: Erik V. Van der Eycken, Upendra K. Sharma, Steven V. Ley, Lars Grunenberg, Joerg Sedelmeier, Fabio Mitsuo Lima, Sandra Johannsen, Debasmita Saha
المساهمون: Lima, Fabio [0000-0003-2127-9568], Ley, Steven [0000-0002-7816-0042], Apollo - University of Cambridge Repository
المصدر: Angewandte Chemie (International Ed. in English)
مصطلحات موضوعية: inorganic chemicals, boronic acids, 010405 organic chemistry, Communication, Library science, Lewis base catalysis, General Chemistry, General Medicine, 010402 general chemistry, 01 natural sciences, Catalysis, Communications, 0104 chemical sciences, 3. Good health, Scholarship, Political science, cross-coupling, synthetic methods, Organic chemistry, Christian ministry, Russian federation, Lewis acids and bases, Photoredox Catalysis
وصف الملف: application/pdf; Print-Electronic