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المؤلفون: Dejian Xie, Gillian Grafton, Alexander Roberts, Nicholas A. Moore, Jinkun Huang, Nicholas M. Barnes, Catherine A. Brady, Kristian Brock, Shuang Liu, Andrew D. Powell, Zania Stamataki, Omar S. Qureshi, A.J Cooper, Chunlin Chen, Peter R. Guzzo, Sargent Bruce J, David D. Manning
المصدر: Journal of Pharmacology and Experimental Therapeutics. 373:122-134
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, biology, Intrinsic activity, business.industry, medicine.disease, Symptomatic relief, Partial agonist, 5-HT3 receptor, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Alosetron, biology.protein, Molecular Medicine, Medicine, business, Receptor, 030217 neurology & neurosurgery, Carcinoid syndrome, Irritable bowel syndrome, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b618e2e0df8d6f7865236dcca51d463b
https://doi.org/10.1124/jpet.119.261008 -
2دورية أكاديمية
المؤلفون: Sargent, Bruce J, Henderson, Alan J
المصدر: In Current Opinion in Pharmacology 2011 11(1):52-58
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3دورية أكاديمية
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المصدر: Neurobiology of Disease, Vol 61, Iss, Pp 47-54 (2014)
مصطلحات موضوعية: Male, Melanin concentrating hormone, Indazoles, Pyridones, medicine.drug_class, Drug Evaluation, Preclinical, CSF, Pharmacology, Bioinformatics, Inflammatory bowel disease, lcsh:RC321-571, Mediator, Weight loss, Drug Discovery, Animals, Humans, Medicine, Obesity, Receptors, Pituitary Hormone, Receptor, lcsh:Neurosciences. Biological psychiatry. Neuropsychiatry, Clinical Trials as Topic, business.industry, Mechanism (biology), Antagonist, Receptor antagonist, medicine.disease, MCH, Rats, Neurology, Go/no go, Anti-Obesity Agents, medicine.symptom, business, MCH1, ALB-127158(a), Human
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المؤلفون: Alan J. Henderson, Sargent Bruce J
المصدر: Current Opinion in Pharmacology. 11:52-58
مصطلحات موضوعية: Pharmacology, Serotonin, medicine.medical_specialty, Mechanism (biology), Biology, Ligand (biochemistry), Serotonin Receptor Agonists, Endocrinology, Receptors, Serotonin, Internal medicine, Drug Discovery, Knockout mouse, medicine, Anorectic, Animals, Humans, Molecular Targeted Therapy, Obesity, Serotonin Antagonists, Antagonism, Receptor, 5-HT receptor
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المؤلفون: Marc L. Reitman, Cheng Guo, Theresa M. Kelly, Constantin Tamvakopoulos, Joseph M. Metzger, Tianying Jian, Howard Y. Chen, Arthur A. Patchett, Oksana C. Palyha, Alison M. Strack, Allan J. Goodman, Ravi P. Nargund, Peter H. Dobbelaar, Yanqing Kan, Mark Hadden, Larry Yet, Peter R. Guzzo, Qianping Peng, Linus S. Lin, Shuwen He, Lauren P. Shearman, Alan J. Henderson, Carina P. Tan, Sargent Bruce J, Xiao-Ming Guan, Scott D. Feighner, Iyassu K. Sebhat, Jie Pan, Jian Liu, Donald J. Marsh, Matthew J. Wyvratt, Andrew D. Howard, Megan Ruenz
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1913-1917
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Molecular Biology, Biphenyl, Chemistry, Drug discovery, fungi, Organic Chemistry, Imidazoles, Rats, Bombesin receptor, Bioavailability, Receptors, Bombesin, Molecular Medicine, Bombesin Receptor Subtype-3
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المؤلفون: Kevin S.J. Thompson, Sargent Bruce J, Sharon L. Smith, David J. Heal
المصدر: CNS Drug Reviews. 7:146-171
مصطلحات موضوعية: Migraine Disorders, medicine.medical_treatment, Pharmacology, Neuroprotection, Article, Mice, chemistry.chemical_compound, Epilepsy, Seizures, medicine, Animals, Humans, Pentylenetetrazol, Bicuculline, medicine.disease, Rats, Pyrimidines, Neuropsychology and Physiological Psychology, Anticonvulsant, chemistry, Cortical spreading depression, NMDA receptor, Anticonvulsants, Picrotoxin, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::790e4795689402b3305b84e3f171d72c
https://doi.org/10.1111/j .1527-3458.2001.tb00193.x -
8دورية أكاديمية
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المؤلفون: Min Hu, Snjezana Lelas, Michael Sinz, Yuri L. Khmelnitsky, Dennis Milanowski, Anne Payen-Fornicola, Matthew Isherwood, Dalton King, Nicholas Holman, Carla Hassler, Wenge Cui, Jonathan O’Connell, Yuh-Lin Yang, Ulhas Bhatt, Nicholas J. Lodge, Yu-Wen Li, Roy Haskell, John E. Macor, Sargent Bruce J, Kim A. Johnson, Linda Fleming, Stephen P. Adams, Vadim V. Mozhaev, Sarah M. Ebeltoft, Shuang Liu, Thaddeus F. Molski, Sambandam Aruna, Richard E. Olson, Congxiang Zha, Robert L. Bertekap, Bruce F. Molino, Wendy Clarke, Robert Zaczek, Anthony D. Pechulis, Michael Herr, Peter R. Guzzo, Larry Yet, Alicia Ng, Anitra F. Orie, Ian C. Cotterill, Kassoum Nacro
المصدر: ACS medicinal chemistry letters. 5(7)
مصطلحات موضوعية: biology, Chemistry, Serotonin reuptake inhibitor, Organic Chemistry, Dopamine reuptake inhibitor, Pharmacology, Biochemistry, Norepinephrine transporter, Norepinephrine reuptake inhibitor, Drug Discovery, biology.protein, Antidepressant, Reuptake inhibitor, Serotonin transporter, Dopamine transporter
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المصدر: Tetrahedron. 54:9603-9612
مصطلحات موضوعية: chemistry.chemical_classification, Aqueous solution, Tetrahydrate, Organic Chemistry, Decarbonylation, Salt (chemistry), Biochemistry, Enamine, chemistry.chemical_compound, chemistry, Reagent, Amide, Drug Discovery, Organic chemistry, Sodium perborate