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المؤلفون: Scott L. Dax, Mingde Xia, Dennis J. Stone, Xiaoqing Xu, Bin Zhu, Donald William Ludovici, Matthews Jay M, Mark A. Youngman, Tasha L. Hutchinson, Michael R. Brandt, Christopher M. Flores, Mary Lou Lubin, Mark J. Macielag, Raymond W. Colburn, Ning Qin, Manomi A. Tennakoon
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2234-2237
مصطلحات موضوعية: Clinical Biochemistry, Cell, Glycine, TRPM Cation Channels, Pharmaceutical Science, Stereoisomerism, Pyrimidinones, Pharmacology, Biochemistry, Structure-Activity Relationship, Transient receptor potential channel, In vivo, Drug Discovery, TRPM8, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, Behavior, Animal, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, In vitro, Rats, HEK293 Cells, medicine.anatomical_structure, Molecular Medicine, Antagonism
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2
المؤلفون: Vita Ozola, Edgars Suna, Andrejs Krasikovs, Scott L. Dax
المصدر: Synthesis. 45:683-693
مصطلحات موضوعية: Green chemistry, chemistry.chemical_classification, chemistry.chemical_compound, Iodoacetic acid, Chemistry, Reagent, Organic Chemistry, Organic chemistry, Catalysis, Flue-gas desulfurization, Amino acid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::dd0b0302fac790a7fa25707347984512
https://doi.org/10.1055/s-0032-1316849 -
3
المؤلفون: Andrew Peter Kennedy, Michael R. Van Scott, Ryan B. Gruber, Toshinori Hoshi, David Ritchie, Richard Woodward, Francis J. Golder, Robert L. Wardle, Courtney Ideo, Veljko Puskovic, Scott L. Dax, Santhosh M. Baby, Sean Peng, James C. Mannion, D. Euan MacIntyre
المصدر: Anesthesiology. 123(5)
مصطلحات موضوعية: Male, medicine.medical_specialty, Mean arterial pressure, Stimulation, Mice, Transgenic, Pharmacology, Rats, Sprague-Dawley, Mice, Internal medicine, Heart rate, medicine, Animals, Respiratory system, Large-Conductance Calcium-Activated Potassium Channel alpha Subunits, Carotid Body, business.industry, Triazines, Respiration, Carotid sinus, Rats, Analgesics, Opioid, Macaca fascicularis, Anesthesiology and Pain Medicine, medicine.anatomical_structure, Endocrinology, Opioid, Breathing, Respiratory Mechanics, Carotid body, Female, business, Respiratory Insufficiency, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::424cab7a7606da9f6d2cc754306754a3
https://pubmed.ncbi.nlm.nih.gov/26352381 -
4
المؤلفون: Ling Lin, Chaozhong Cai, Christopher M. Flores, Timothy P Coogan, Edmund K. LeGrand, Ellen E. Codd, Raymond W. Colburn, Angelique Leone, Charles Y. Wang, Mcdonnell Mark E, Scott L. Dax, Michael R. Brandt, Stewart Bryant, Bart DeCorte, James J. McNally, John R. Mabus, Sui-Po Zhang, John R. Carson, Michael Kemmerer, Dennis J. Stone, James M Lenhard, Michael K. McMillian, Kristen M. Chevalier, Judith Baker
المصدر: Toxicological Sciences. 117:493-504
مصطلحات موضوعية: Blood Glucose, Male, medicine.medical_specialty, Narcotic Antagonists, medicine.medical_treatment, Cyproheptadine, Cell Enlargement, Pharmacology, Osteochondrodysplasias, Toxicology, Rats, Sprague-Dawley, δ-opioid receptor, Mice, Dogs, Cell Line, Tumor, Insulin-Secreting Cells, Internal medicine, medicine, Animals, Insulin, Potency, Pancreas, chemistry.chemical_classification, Chemistry, High-Throughput Screening Assays, Rats, Diabetes Mellitus, Type 1, Endocrinology, Opioid, Hyperglycemia, Vacuoles, Toxicity, Female, Insulinoma, Serotonin Antagonists, Epiphyses, Hyperglycemic agent, medicine.drug, Tricyclic
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9776c107aa28aa0bdc15b9be77554703
https://doi.org/10.1093/toxsci/kfq200 -
5
المؤلفون: John R. Carson, Lou Anne Neilson, Ellen E. Codd, Jung Lee, Philip M. Pitis, Rebecca P. Martinez, Scott L. Dax, L. A. McKown, Wu-Nan Wu, Steven J. Coats, Sui-Po Zhang
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:2113-2116
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Analgesic, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Opioid, chemistry, In vivo, Amide, Drug Discovery, medicine, Molecular Medicine, Structure–activity relationship, Molecular Biology, medicine.drug
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6
المؤلفون: Rebecca P. Martinez, John R. Carson, Lou Anne Neilson, Steven J. Coats, Ellen E. Codd, Sui-Po Zhang, Jung Lee, Philip M. Pitis, Scott L. Dax
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:2109-2112
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Analgesic, Pharmaceutical Science, Stimulation, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Opioid receptor, Receptors, Opioid, delta, Drug Discovery, medicine, Molecular Biology, Chemistry, Organic Chemistry, General Medicine, Gtpγs binding, Analgesics, Opioid, Nociception, Opioid, Guanosine 5'-O-(3-Thiotriphosphate), Benzamides, Molecular Medicine, Selectivity, medicine.drug
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المؤلفون: Nadia Nasser, Adrienne E. Dubin, Sui Po Zhang, Scott L. Dax, Mcdonnell Mark E
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:531-534
مصطلحات موضوعية: Bicyclic molecule, Stereochemistry, Receptors, Drug, Organic Chemistry, Clinical Biochemistry, TRPV1, Antagonist, TRPV Cation Channels, Pharmaceutical Science, Naphthols, Amides, Biochemistry, Chemical synthesis, chemistry.chemical_compound, chemistry, Capsaicin, Amide, Drug Discovery, Urea, Humans, Molecular Medicine, Receptor, Molecular Biology, Protein Binding
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المؤلفون: Mark A. Youngman, James J. McNally, Scott L. Dax, Nicole M. Willard
المصدر: Synthetic Communications. 33:2215-2227
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Sodium cyanoborohydride, Organic Chemistry, Organic chemistry, Reductive amination, Medicinal chemistry, Ammonium acetate, Tetralones
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المؤلفون: Mcdonnell Mark E, Sui Po Zhang, Adrienne E. Dubin, Scott L. Dax
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:1189-1192
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Receptors, Drug, Clinical Biochemistry, Drug Evaluation, Preclinical, Resiniferatoxin, Pharmaceutical Science, In Vitro Techniques, Biochemistry, Chemical synthesis, Partial agonist, chemistry.chemical_compound, Drug Discovery, medicine, Humans, heterocyclic compounds, Phenols, Orthoester, Molecular Biology, Organic Chemistry, Biological activity, In vitro, chemistry, Molecular Medicine, Diterpenes, Iodine
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المؤلفون: Sandy J. Wilson, Scott L. Dax, Mcnally James J, Brian C. Zanoni, Allen B. Reitz, Cheryl P. Kordik, Chi Luo, Timothy W. Lovenberg
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2283-2286
مصطلحات موضوعية: Y5 Receptor, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Neuropeptide, Binding, Competitive, Biochemistry, Chemical synthesis, Cell Line, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Organic Chemistry, Neuropeptide Y receptor, In vitro, Receptors, Neuropeptide Y, Sulfonamide, chemistry, Drug Design, Pyrazoles, Molecular Medicine, Lead compound