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المؤلفون: Zhihong Huang, Jennifer Shaffer, Badry Bursulaya, Anna Galkin, Rie Kikkawa, Yelena Sarkisova, Su Hua, John Tellew, Yang Yang, Paul Vincent Rucker, Robert Epple, Jiqing Jiang, Nanxin Li, Chianelli Donatella, Jason Roland, Lintong Li, Sergio Briones, Casey J. N. Mathison, Valentina Molteni, Jacqueline Kinyamu-Akunda, Mu-Yun Gao, John Nelson, Christian C. Lee, Yun Feng Xie, Shailaja Kasibhatla, Chun Li
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Pyrimidine, biology, Kinase, Organic Chemistry, hERG, Cancer, Pharmacology, medicine.disease, Biochemistry, In vitro, chemistry.chemical_compound, Antitarget, chemistry, Tolerability, In vivo, Drug Discovery, biology.protein, medicine
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المؤلفون: Anhthu Dang, Deborah Knee, Cui Ying Wang, Feng Gao, Guoxun Liu, Sergio Briones, Michelle Coulson, Jessica Makofske, Keith Mansfield, May Liu, Tanya Mulvey, Emily K Meseck, Steve Woolfenden, Sean G Buchanan, David Steensma, Vasileios Askoxylakis
المصدر: Blood. 140:11564-11565
مصطلحات موضوعية: Immunology, Cell Biology, Hematology, Biochemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4d3e920fadb2ab0859e7a27380e4191b
https://doi.org/10.1182/blood-2022-159910 -
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المؤلفون: Badry Bursulaya, Nanxin Li, Yang Yang, Chianelli Donatella, John Nelson, Casey J. N. Mathison, Valentina Molteni, Sergio Briones, Chun Li, Shailaja Kasibhatla, Christian C. Lee, Jason Roland, Zhihong Huang, Jiqing Jiang, Anna Galkin, John Tellew, Robert Epple, Jacqueline Kinyamu-Akunda, Yelena Sarkisova, Mu-Yun Gao, Rie Kikkawa, Lintong Li, Su Hua, Paul Vincent Rucker, Jennifer Shaffer, Yun Feng Xie
المصدر: ACS Medicinal Chemistry Letters. 11:558-565
مصطلحات موضوعية: Pyrimidine, biology, 010405 organic chemistry, Chemistry, Kinase, business.industry, Organic Chemistry, Kinase insert domain receptor, medicine.disease, 01 natural sciences, Biochemistry, Receptor tyrosine kinase, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Text mining, Tolerability, In vivo, Drug Discovery, Cancer research, biology.protein, medicine, Adenocarcinoma, business
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المؤلفون: Carrie Richardson, Scott Armstrong, Sergio Briones, Sharath S. Hegde, Brian Horger, Sarah Jaw-Tsai
المصدر: Naunyn-Schmiedeberg's Archives of Pharmacology. 376:341-349
مصطلحات موضوعية: medicine.medical_specialty, Blood Pressure, Muscarinic Antagonists, Pharmacology, Rats, Sprague-Dawley, In vivo, Internal medicine, Muscarinic acetylcholine receptor, Bradycardia, medicine, Darifenacin, Animals, Infusions, Intravenous, Receptor, Methacholine Chloride, Receptor, Muscarinic M3, Receptor, Muscarinic M2, Dose-Response Relationship, Drug, Chemistry, Muscarinic acetylcholine receptor M3, General Medicine, Smooth muscle contraction, Rats, Disease Models, Animal, Endocrinology, Female, Methacholine, Tolterodine, medicine.drug
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المصدر: The FASEB Journal. 21
مصطلحات موضوعية: In vivo, Chemistry, Simple (abstract algebra), Muscarinic acetylcholine receptor, Genetics, Antagonist, Pharmacology, Molecular Biology, Biochemistry, Biotechnology