المؤلفون: Zyk NY; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Garanina AS; Laboratory of Biomedical Nanomaterials, National University of Science and Technology MISIS, 4 Leninskiy pr, Moscow 119049, Russia., Plotnikova EA; National Medical Research Radiological Centre of the Ministry of Health of the Russian Federation, 2 Botkinskiy proezd, 3, Moscow 125284, Russia., Ber AP; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Nimenko EA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Dashkova NS; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Uspenskaia AA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Shafikov RR; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia.; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow 117997, Russia., Skvortsov DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Petrov SA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Pankratov AA; National Medical Research Radiological Centre of the Ministry of Health of the Russian Federation, 2 Botkinskiy proezd, 3, Moscow 125284, Russia., Zyk NV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Majouga AG; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya sq. 9, Moscow 125047, Russia., Beloglazkina EK; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia., Machulkin AE; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russia.

المصدر: International journal of molecular sciences [Int J Mol Sci] 2023 Jul 11; Vol. 24 (14). Date of Electronic Publication: 2023 Jul 11.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

مواضيع طبية MeSH: Androgen Antagonists*/therapeutic use , Prostatic Neoplasms*/metabolism, Male ; Humans ; Cytotoxins/therapeutic use ; Prostate/pathology ; Ligands ; Cell Line, Tumor ; Glutamate Carboxypeptidase II/metabolism ; Antigens, Surface/metabolism

المؤلفون: Ivanenkov YA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia.; The Federal State Unitary Enterprise Dukhov Automatics Research Institute (VNIIA), 22. ul. Sushchevskaya, 127055 Moscow, Russia., Kukushkin ME; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Beloglazkina AA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Shafikov RR; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia.; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry RAS, GSP-7, Ulitsa Mklukho-Maklaya 16/10, 17997 Moscow, Russia.; A. N. Belozersky Research Institute of Physico-Chemical Biology MSU, Leninskye Gory, House 1, Building 40, 119992 Moscow, Russia., Barashkin AA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Ayginin AA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Serebryakova MS; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Majouga AG; College of New Materials and Nanotechnologies, National University of Science and Technology MISiS, 119049 Moscow, Russia., Skvortsov DA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Tafeenko VA; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia., Beloglazkina EK; Chemistry Department, Moscow State University, Leninskie Gory 1/3, 119991 Moscow, Russia.

المصدر: Molecules (Basel, Switzerland) [Molecules] 2023 Jan 30; Vol. 28 (3). Date of Electronic Publication: 2023 Jan 30.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE

مواضيع طبية MeSH: Antineoplastic Agents*/chemistry, Humans ; Animals ; Mice ; Structure-Activity Relationship ; Oxindoles/pharmacology ; Molecular Docking Simulation ; Mice, Nude ; HEK293 Cells ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Cell Line, Tumor ; Molecular Structure

المؤلفون: Zyk NY; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation. Electronic address: Zyknikola@gmail.com., Ber AP; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Nimenko EA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Shafikov RR; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow 117997, Russian Federation., Evteev SA; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russia., Petrov SA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Uspenskaya AA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Dashkova NS; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Ivanenkov YA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russia., Skvortsov DA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Beloglazkina EK; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Majouga AG; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow 125047, Russian Federation., Machulkin AE; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; RUDN University, Miklukho-Maklaya Str. 6, Moscow 117198, Russian Federation.

المصدر: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2022 Sep 01; Vol. 71, pp. 128840. Date of Electronic Publication: 2022 May 31.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

مواضيع طبية MeSH: Lysine* , Prostatic Neoplasms*, Antigens, Surface ; Cell Line, Tumor ; Glutamate Carboxypeptidase II ; Humans ; Ligands ; Male ; Nitrogen

المؤلفون: Machulkin AE; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation. Electronic address: alekseymachulkin@rambler.ru., Uspenskaya AA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Zyk NY; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Nimenko EA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Ber AP; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Petrov SA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Shafikov RR; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow, 117997, Russian Federation., Skvortsov DA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Faculty of Biology and Biotechnologies, Higher School of Economics, Myasnitskaya 13, Moscow, 101000, Russia., Smirnova GB; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia., Borisova YA; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia., Pokrovsky VS; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia; RUDN University, Miklukho-Maklaya Str.6, Moscow, 117198, Russian Federation., Kolmogorov VS; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Vaneev AN; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Ivanenkov YA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russia; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, Ufa, 450054, Russian Federation., Khudyakov AD; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Kovalev SV; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Erofeev AS; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Gorelkin PV; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Beloglazkina EK; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Zyk NV; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Khazanova ES; LLC Izvarino-Pharma, V. Vnukovskoe, Vnukovskoe Sh., 5th Km., Building 1, Moscow, 108817, Russian Federation., Majouga AG; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow, 125047, Russian Federation.

المصدر: European journal of medicinal chemistry [Eur J Med Chem] 2022 Jan 05; Vol. 227, pp. 113936. Date of Electronic Publication: 2021 Oct 23.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Docetaxel/*pharmacology , Prostate-Specific Antigen/*antagonists & inhibitors , Small Molecule Libraries/*pharmacology, Animals ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Docetaxel/chemical synthesis ; Docetaxel/chemistry ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Humans ; Male ; Mice ; Mice, Inbred ICR ; Molecular Structure ; Neoplasms, Experimental/drug therapy ; Neoplasms, Experimental/metabolism ; Neoplasms, Experimental/pathology ; Prostate-Specific Antigen/genetics ; Prostate-Specific Antigen/metabolism ; Rabbits ; Rats ; Rats, Wistar ; Small Molecule Libraries/chemical synthesis ; Small Molecule Libraries/chemistry ; Structure-Activity Relationship

المؤلفون: Machulkin AE; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Uspenskaya AA; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Zyk NU; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Nimenko EA; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Ber AP; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Petrov SA; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Polshakov VI; Center for Magnetic Tomography and Spectroscopy, Faculty of Fundamental Medicine, Lomonosov Moscow State University, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Shafikov RR; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation.; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow 117997, Russian Federation., Skvortsov DA; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Plotnikova EA; National Medical Research Radiological Centre of the Ministry of Health of the Russian Federation, 2 Botkinskiy Proezd, 3, Moscow 125284, Russian Federation., Pankratov AA; National Medical Research Radiological Centre of the Ministry of Health of the Russian Federation, 2 Botkinskiy Proezd, 3, Moscow 125284, Russian Federation., Smirnova GB; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye Shosse, Moscow 115478, Russian Federation., Borisova YA; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye Shosse, Moscow 115478, Russian Federation., Pokrovsky VS; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye Shosse, Moscow 115478, Russian Federation.; RUDN University, Miklukho-Maklaya Street 6, Moscow 117198, Russian Federation., Kolmogorov VS; National University of Science and Technology MISiS, 9 Leninskiy Prospekt, Moscow 119049, Russian Federation., Vaneev AN; National University of Science and Technology MISiS, 9 Leninskiy Prospekt, Moscow 119049, Russian Federation., Khudyakov AD; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Chepikova OE; Department of Biotechnology, Sirius University of Science and Technology, 1 Olympic Avenue, Sochi 354340, Russian Federation., Kovalev S; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Zamyatnin AA Jr; Department of Biotechnology, Sirius University of Science and Technology, 1 Olympic Avenue, Sochi 354340, Russian Federation.; Institute of Molecular Medicine, Sechenov First Moscow State Medical University, Trubetskaya Street 8-2, Moscow 119991, Russian Federation.; Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, GSP-1, Leninskie Gory, Moscow 119992, Russian Federation.; Faculty of Health and Medical Sciences, University of Surrey, Guildford GU2 7XH, U.K., Erofeev A; National University of Science and Technology MISiS, 9 Leninskiy Prospekt, Moscow 119049, Russian Federation., Gorelkin P; National University of Science and Technology MISiS, 9 Leninskiy Prospekt, Moscow 119049, Russian Federation., Beloglazkina EK; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Zyk NV; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation., Khazanova ES; LLC Izvarino-Pharma, v. Vnukovskoe, Vnukovskoe Shosse, Fifth km., Building 1, Moscow 108817, Russian Federation., Majouga AG; Chemistry Department, Lomonosov Moscow State University, Building 1/3, GSP-1, Leninskie Gory, Moscow 119991, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy Prospekt, Moscow 119049, Russian Federation.; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya Square 9, Moscow 125047, Russian Federation.

المصدر: Journal of medicinal chemistry [J Med Chem] 2021 Dec 09; Vol. 64 (23), pp. 17123-17145. Date of Electronic Publication: 2021 Nov 19.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Antigens, Surface/*chemistry , Coordination Complexes/*chemistry , Coordination Complexes/*pharmacology , Glutamate Carboxypeptidase II/*chemistry , Oligopeptides/*chemistry, Cell Line, Tumor ; Coordination Complexes/chemical synthesis ; Humans ; Male ; Microsomes, Liver/enzymology ; Microsomes, Liver/metabolism ; Prostatic Neoplasms/pathology ; Reactive Oxygen Species/metabolism ; Xenograft Model Antitumor Assays

المؤلفون: Machulkin AE; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Shafikov RR; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow 117997, Russian Federation., Uspenskaya AA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Petrov SA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Ber AP; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Skvortsov DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; Faculty of Biology and Biotechnologies, Higher School of Economics, Myasnitskaya 13, Moscow 101000, Russia., Nimenko EA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Zyk NU; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Smirnova GB; N.N. Blokhin Cancer Research Center, 24 Kashirskoye sh., Moscow 115478 , Russia., Pokrovsky VS; N.N. Blokhin Cancer Research Center, 24 Kashirskoye sh., Moscow 115478 , Russia.; RUDN University, Miklukho-Maklaya str. 6, Moscow 117198, Russian Federation., Abakumov MA; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation., Saltykova IV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Akhmirov RT; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya sq. 9, Moscow 125047, Russian Federation., Garanina AS; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation., Polshakov VI; Center for Magnetic Tomography and Spectroscopy, Faculty of Fundamental Medicine, M.V. Lomonosov Moscow State University, Moscow 119991, Russian Federation., Saveliev OY; Center for Magnetic Tomography and Spectroscopy, Faculty of Fundamental Medicine, M.V. Lomonosov Moscow State University, Moscow 119991, Russian Federation., Ivanenkov YA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region 141700, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation.; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow 127055, Russia.; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, Ufa 450054, Russian Federation., Aladinskaya AV; Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region 141700, Russian Federation., Finko AV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Yamansarov EU; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Krasnovskaya OO; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation., Erofeev AS; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation., Gorelkin PV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation., Dontsova OA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow 117997, Russian Federation., Beloglazkina EK; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Zyk NV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Khazanova ES; Izvarino Pharma LLC, v. Vnukovskoe, Vnukovskoe sh., 5th km., Building 1, Moscow 108817, Russian Federation., Majouga AG; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation.; National University of Science and Technology MISiS, 9 Leninskiy pr., Moscow 119049, Russian Federation.; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya sq. 9, Moscow 125047, Russian Federation.

المصدر: Journal of medicinal chemistry [J Med Chem] 2021 Apr 22; Vol. 64 (8), pp. 4532-4552. Date of Electronic Publication: 2021 Apr 06.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Ligands*, Antigens, Surface/*metabolism , Antineoplastic Agents/*metabolism , Fluorescent Dyes/*chemistry , Glutamate Carboxypeptidase II/*metabolism, Animals ; Antigens, Surface/chemistry ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/pharmacology ; Antineoplastic Agents/therapeutic use ; Cell Line, Tumor ; Cell Survival/drug effects ; Drug Screening Assays, Antitumor ; Glutamate Carboxypeptidase II/chemistry ; Humans ; Male ; Mice ; Mice, Nude ; Optical Imaging ; Prostatic Neoplasms/drug therapy ; Structure-Activity Relationship ; Tissue Distribution ; Transplantation, Heterologous

المؤلفون: Krasnovskaya OO; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia.; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Guk DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Naumov AE; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Nikitina VN; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Semkina AS; Department of Medical Nanobiotechnologies, Pirogov Russian National Research Medical University, Ostrovityanova 1, Moscow 117997, Russia.; Department of Basic and Applied Neurobiology, Serbsky National Medical Research Center for Psychiatry and Narcology, Kropotkinskiy 23, Moscow 119991, Russia., Vlasova KY; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Pokrovsky V; N.N. Blokhin National Medical Research Center of Oncology of the Ministry of Health of the Russian Federation, Kashirskoe Highway 23, Moscow 115478, Russia.; People's Friendship University, Moscow, Russia, Miklukho-Maklaya 6, Moscow 117198, Russia., Ryabaya OO; N.N. Blokhin National Medical Research Center of Oncology of the Ministry of Health of the Russian Federation, Kashirskoe Highway 23, Moscow 115478, Russia., Karshieva SS; N.N. Blokhin National Medical Research Center of Oncology of the Ministry of Health of the Russian Federation, Kashirskoe Highway 23, Moscow 115478, Russia., Skvortsov DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia.; Department of Biology and Biotechnologies, Higher School of Economics, Myasnitskaya 13, Moscow 101000, Russia., Zhirkina IV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Shafikov RR; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Gorelkin PV; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia., Vaneev AN; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia.; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Erofeev AS; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia., Mazur DM; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Tafeenko VA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Pergushov VI; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Melnikov MY; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Soldatov MA; The Smart Materials Research Institute Southern Federal University Sladkova, 178/24, Rostov-on-Don 344090, Russia., Shapovalov VV; The Smart Materials Research Institute Southern Federal University Sladkova, 178/24, Rostov-on-Don 344090, Russia., Soldatov AV; The Smart Materials Research Institute Southern Federal University Sladkova, 178/24, Rostov-on-Don 344090, Russia., Akasov RA; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia.; I.M. Sechenov First Moscow State Medical University, Trubetskaya 8-2, Moscow 119991, Russia., Gerasimov VM; Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow 125047, Russia., Sakharov DA; Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow 125047, Russia., Moiseeva AA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Zyk NV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Beloglazkina EK; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia., Majouga AG; Department of Materials Science of Semiconductors and Dielectrics, National University of Science and Technology MISIS, Leninskiy Prospect 4, Moscow 101000, Russia.; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russia.; Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow 125047, Russia.

المصدر: Journal of medicinal chemistry [J Med Chem] 2020 Nov 12; Vol. 63 (21), pp. 13031-13063. Date of Electronic Publication: 2020 Oct 20.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Coordination Complexes/*chemistry , Copper/*chemistry , Imidazoles/*chemistry, Antineoplastic Agents/chemistry ; Antineoplastic Agents/metabolism ; Antineoplastic Agents/pharmacology ; Apoptosis/drug effects ; Coordination Complexes/metabolism ; Coordination Complexes/pharmacology ; Crystallography, X-Ray ; DNA Damage/drug effects ; Humans ; Ligands ; MCF-7 Cells ; Models, Biological ; Molecular Conformation ; Oxidation-Reduction ; Reactive Oxygen Species/metabolism ; Spheroids, Cellular/drug effects ; Structure-Activity Relationship ; Telomerase/antagonists & inhibitors ; Telomerase/metabolism

المؤلفون: Machulkin AE; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, 450054 Ufa, Russian Federation. Electronic address: alekseymachulkin@rambler.ru., Skvortsov DA; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation. Electronic address: skvorratd@mail.ru., Ivanenkov YA; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region 141700, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy pr, Moscow 119049, Russian Federation; ChemDiv, San Diego, CA, USA; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, 450054 Ufa, Russian Federation., Ber AP; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Kavalchuk MV; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Aladinskaya AV; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region 141700, Russian Federation., Uspenskaya AA; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Shafikov RR; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Plotnikova EA; P. A. Herzen Moscow Oncology Research Institute, 3, 2th Botkinsky Driveway, Moscow 125284, Russian Federation., Yakubovskaya RI; P. A. Herzen Moscow Oncology Research Institute, 3, 2th Botkinsky Driveway, Moscow 125284, Russian Federation., Nimenko EA; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Zyk NU; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Beloglazkina EK; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Zyk NV; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Koteliansky VE; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation., Majouga AG; Lomonosov Moscow State University, Chemistry Dept., Leninskie gory, Building 1/3, GSP-1, Moscow 119991, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy pr, Moscow 119049, Russian Federation; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya sq. 9, Moscow 125047, Russian Federation.

المصدر: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2019 Aug 15; Vol. 29 (16), pp. 2229-2235. Date of Electronic Publication: 2019 Jun 20.

نوع المنشور: Letter; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

مواضيع طبية MeSH: Drug Delivery Systems/*methods , Paclitaxel/*chemical synthesis , Prostatic Neoplasms/*drug therapy, Animals ; Humans ; Male ; Mice

المؤلفون: Guk DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory 1/3, Moscow 119991, Russia., Krasnovskaya OO, Dashkova NS, Skvortsov DA, Rubtsova MP, Dyadchenko VP, Yudina ES, Kosarev MA, Soldatov AV, Shapovalov VV, Semkina AS, Vlasova KY, Pergushov VI, Shafikov RR, Moiseeva AA, Andreeva AV, Melnikov MY, Zyk NV, Majouga AG, Beloglazkina EK

المصدر: Dalton transactions (Cambridge, England : 2003) [Dalton Trans] 2019 Jan 02; Vol. 48 (2), pp. 752.

نوع المنشور: Journal Article; Published Erratum

بيانات الدورية: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101176026 Publication Model: Print Cited Medium: Internet ISSN: 1477-9234 (Electronic) Linking ISSN: 14779226 NLM ISO Abbreviation: Dalton Trans Subsets: PubMed not MEDLINE

المؤلفون: Guk DA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory 1/3, Moscow 119991, Russia., Krasnovskaya OO, Dashkova NS, Skvortsov DA, Rubtsova MP, Dyadchenko VP, Yudina ES, Kosarev MA, Soldatov AV, Shapovalov VV, Semkina AS, Vlasova KY, Pergushov VI, Shafikov RR, Moiseeva, Andreeva, Andreeva AA, Melnikov MY, Zyk NV, Majouga AG, Beloglazkina EK

المصدر: Dalton transactions (Cambridge, England : 2003) [Dalton Trans] 2018 Dec 11; Vol. 47 (48), pp. 17357-17366.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101176026 Publication Model: Print Cited Medium: Internet ISSN: 1477-9234 (Electronic) Linking ISSN: 14779226 NLM ISO Abbreviation: Dalton Trans Subsets: MEDLINE

مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Coordination Complexes/*pharmacology , Copper/*pharmacology , Enzyme Inhibitors/*pharmacology , Imidazoles/*pharmacology , Metallocenes/*pharmacology , Telomerase/*antagonists & inhibitors, Animals ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Apoptosis/drug effects ; Cattle ; Cell Line ; Cell Proliferation/drug effects ; Coordination Complexes/chemical synthesis ; Coordination Complexes/chemistry ; Copper/chemistry ; DNA Cleavage ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Enzyme Inhibitors/chemical synthesis ; Enzyme Inhibitors/chemistry ; HEK293 Cells ; Humans ; Imidazoles/chemical synthesis ; Imidazoles/chemistry ; Metallocenes/chemistry ; Molecular Structure ; Serum Albumin, Bovine/chemistry ; Structure-Activity Relationship ; Telomerase/metabolism