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1
المؤلفون: Ryotaku Inoue, Keiko Oshima, Shin-ichi Inaba, Takashi Kagari, Kaoru Tanaka-takanaka, Wataru Tomisato, Takaichi Shimozato, Takashi Izumi, Hiromi Doi-Komuro, Maki Goto, Hiroshi Yuita, Hisako Tanaka
المصدر: Biopharmaceutics & Drug Disposition. 37:561-573
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Sphingosine, Lymphocyte, Experimental autoimmune encephalomyelitis, Pharmaceutical Science, General Medicine, Biology, medicine.disease, 030226 pharmacology & pharmacy, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, medicine.anatomical_structure, Pharmacokinetics, chemistry, Free fraction, Oral administration, Pharmacodynamics, medicine, Pharmacology (medical), Active metabolite
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2
المؤلفون: Kiyoaki Yonesu, Maki Yamaguchi-Goto, Takashi Izumi, Hidetaka Sakurai, Shin-ichi Inaba, Kaoru Tanaka-takanaka, Kazuishi Kubota
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 48(3)
مصطلحات موضوعية: 0301 basic medicine, Male, Erythrocytes, Health, Toxicology and Mutagenesis, Morpholines, Fructose, Biology, Toxicology, Kidney, Biochemistry, Isozyme, Dephosphorylation, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Intestine, Small, Humans, Pyrroles, Enzyme Inhibitors, Phosphorylation, Pharmacology, chemistry.chemical_classification, General Medicine, Alkaline Phosphatase, Molecular biology, Amino Alcohols, Recombinant Proteins, Kinetics, Phosphotransferases (Alcohol Group Acceptor), Receptors, Lysosphingolipid, 030104 developmental biology, Enzyme, chemistry, Levamisole, 030220 oncology & carcinogenesis, Microsome, Microsomes, Liver, Alkaline phosphatase, Fructosamine-3-kinase, Female
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3
المؤلفون: Ikeda Takuya, Toshiyasu Takemoto, Yukiko Sekiguchi, Takashi Kagari, Takaichi Shimozato, Takeshi Fukuda, Taiji Goto, Yumi Kawase, Tsuyoshi Nakamura, Takashi Tsuji, Futoshi Nara, Keisuke Suzuki, Takashi Izumi, Takahide Nishi, Masakazu Tamura, Tomohiro Honda, Shin-ichi Inaba, Takako Kimura, Yumiko Mizuno, Chizuko Yahara
المصدر: Bioorganic & Medicinal Chemistry. 22:4246-4256
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Benzyl ether, chemistry, Docking (molecular), Oral administration, In vivo, Drug Discovery, Molecular Medicine, Homology modeling, Ethyl group, Selectivity, Receptor modulator, Molecular Biology
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4
المصدر: Molecular & Cellular Proteomics : MCP
مصطلحات موضوعية: Proteomics, Phosphatase, Biology, Kidney, Biochemistry, Isozyme, Analytical Chemistry, Sphingosine, Humans, Pyrroles, Molecular Biology, chemistry.chemical_classification, Fingolimod Hydrochloride, Research, ALPL, Biological activity, Alkaline Phosphatase, Amino Alcohols, Enzyme assay, Isoenzymes, Enzyme, chemistry, Propylene Glycols, biology.protein, Alkaline phosphatase, Immunosuppressive Agents
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f97067b6776a70308f917e6c7dfe84b6
http://europepmc.org/articles/PMC3734587 -
5
المؤلفون: Shin-Ichi, Inaba, Maki, Goto, Kaoru, Tanaka-Takanaka, Hisako, Tanaka, Wataru, Tomisato, Hiroshi, Yuita, Hiromi, Doi-Komuro, Ryotaku, Inoue, Keiko, Oshima, Takashi, Kagari, Takaichi, Shimozato, Takashi, Izumi
المصدر: Biopharmaceuticsdrug disposition. 37(9)
مصطلحات موضوعية: Male, Dose-Response Relationship, Drug, Administration, Oral, Amino Alcohols, Rats, Rats, Sprague-Dawley, Macaca fascicularis, Receptors, Lysosphingolipid, Species Specificity, Rats, Inbred Lew, Animals, Female, Pyrroles, Lymphocytes, Rats, Wistar
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6
المؤلفون: Nobuaki Watanabe, Shin-ichi Inaba, Chizuko Yahara, Kazuishi Kubota, Masakazu Tamura, Kiyoaki Yonesu, Futoshi Nara, Tomohiro Honda, Tatsuji Matsuoka
المصدر: The Journal of Biological Chemistry
مصطلحات موضوعية: Proteomics, Erythrocytes, Protein Purification, Morpholines, Immunology, Sphingosine kinase, Enzyme Purification, Fructose, Mitogen-activated protein kinase kinase, Biochemistry, MAP2K7, Mass Spectrometry (MS), Animals, Humans, Prodrugs, Pyrroles, Enzyme Inhibitors, Phosphorylation, Kinase activity, Sphingosine-1-Phosphate Receptors, Molecular Biology, biology, Cyclin-dependent kinase 2, Cyclin-dependent kinase 3, Cell Biology, Amino Alcohols, Protein kinase R, Rats, Phosphotransferases (Alcohol Group Acceptor), Receptors, Lysosphingolipid, HEK293 Cells, Enzymology, Immunosuppressor, biology.protein, Cyclin-dependent kinase 9
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6f6c4a8e90376aa653008ffe88252e7
https://doi.org/10.1074/jbc.m110.217299 -
7
المؤلفون: Wataru Tomisato, Keisuke Suzuki, Ryotaku Inoue, Yumi Kawase, Takashi Izumi, Keiko Oshima, Hiroshi Yuita, Takaichi Shimozato, Katsuyoshi Nakajima, Takahide Nishi, Shojiro Miyazaki, Futoshi Nara, Yukiko Iio, Takashi Kagari, Shin-ichi Inaba, Takashi Ohnuki, Toshiyasu Takemoto, Hiromi Doi
المصدر: ACS Medicinal Chemistry Letters. 2:368-372
مصطلحات موضوعية: Agonist, medicine.drug_class, business.industry, Multiple sclerosis, Lymphocyte, Organic Chemistry, Experimental autoimmune encephalomyelitis, Pharmacology, medicine.disease, Biochemistry, In vitro, medicine.anatomical_structure, Pharmacokinetics, In vivo, Peripheral blood lymphocyte, Drug Discovery, medicine, business
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8
المؤلفون: Hamim Zahir, Kenneth E. Truitt, James B. Moberly, Timothy J. Carrothers, Takaichi Shimozato, Shashank Rohatagi, Shin-ichi Inaba
المصدر: The Journal of Clinical Pharmacology. 49:50-62
مصطلحات موضوعية: Adult, CD4-Positive T-Lymphocytes, Male, Adolescent, Lymphocyte, Administration, Oral, Pharmacology, Biology, Models, Biological, Cohort Studies, Young Adult, chemistry.chemical_compound, Double-Blind Method, Pharmacokinetics, Sphingosine, medicine, Humans, Prodrugs, Pyrroles, Pharmacology (medical), Lymphocyte Count, Lymphocytes, Dosing, IC50, Active metabolite, PK/PD models, Dose-Response Relationship, Drug, Middle Aged, Amino Alcohols, Lymphocyte Subsets, Receptors, Lysosphingolipid, medicine.anatomical_structure, chemistry, Pharmacodynamics, Lysophospholipids
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9
المؤلفون: Tohru Takahashi, Akira Shinagawa, Kimihisa Ichikawa, Kazuishi Kubota, Takashi Izumi, Yumiko Fukushima, Hidetaka Sakurai, Shin-ichi Inaba, Mihoko Watanabe, Rika Nakano
المصدر: Pharmacology Research & Perspectives
مصطلحات موضوعية: chemistry.chemical_classification, FBPase inhibitor, biology, phosphoramidase, Carboxylesterase 1, bisamidate prodrug, Original Articles, Sphingomyelin phosphodiesterase, Prodrug, Biochemical purification, Cathepsin A, Esterase, Enzyme assay, drug metabolizing enzyme, Enzyme, Neurology, Biochemistry, chemistry, biology.protein, CS-917, General Pharmacology, Toxicology and Pharmaceutics, Histidine
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10
المؤلفون: Takashi Izumi, Maki Goto, Hisako Tanaka, Shin-ichi Inaba, Makoto Takahashi, Haruo Iwabuchi, Tomoko Ikeda
مصطلحات موضوعية: Male, Health, Toxicology and Mutagenesis, Metabolite, Administration, Oral, Pharmacology, Biology, Toxicology, Hydroxylation, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Feces, Pharmacokinetics, Oral administration, Animals, Pyrroles, Tissue Distribution, Phosphorylation, Active metabolite, Biotransformation, Sphingosine, General Medicine, Metabolism, Blood proteins, Amino Alcohols, Rats, Macaca fascicularis, Receptors, Lysosphingolipid, chemistry, Intestinal Absorption, Injections, Intravenous, Oxidation-Reduction, Algorithms, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::40f5565753aafdc646029efaf0e4f23e