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المؤلفون: Jon Hilden, Stephen D. Stamatis, Jeffrey S. Tan, Shobha N. Bhattachar
المصدر: Burger's Medicinal Chemistry and Drug Discovery
مصطلحات موضوعية: Chemistry, Pharmaceutics, Early phase, Neuroscience
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c260fddd98f2ee2abcaa44b6ef6c7dd2
https://doi.org/10.1002/0471266949.bmc263 -
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المؤلفون: Phenil J. Patel, Marieta Duvnjak Romic, Dipal Patel, Margaret S. Landis, Darren L. Reid, Shobha N. Bhattachar, Wenzhan Yang
المصدر: Drug Discovery Today. 26:713-723
مصطلحات موضوعية: 0301 basic medicine, Drug, Drug Industry, Computer science, media_common.quotation_subject, 03 medical and health sciences, Drug Delivery Systems, 0302 clinical medicine, Drug Development, Drug Discovery, Animals, Humans, Technology, Pharmaceutical, Pharmaceutical industry, media_common, Pharmacology, business.industry, Drug discovery, Target engagement, Drug Liberation, Safety profile, 030104 developmental biology, Tolerability, Risk analysis (engineering), Drug Design, 030220 oncology & carcinogenesis, Drug delivery, business, Dosing Frequency
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المؤلفون: Xueqian Gong, Karsten Boehnke, Carmen Baquero, Yue-Wei Qian, Gregory P. Donoho, Jason Manro, Robert T. Foreman, Carlos Marugán, Sonya C. Chapman, Yi Zeng, Phillip W Iversen, Jack A. Dempsey, Matthew Z. Dieter, David Anthony Barda, Henry James Robert, Michele Dowless, Shripad V. Bhagwat, Robert M. Campbell, Andrew Capen, Robert D. Van Horn, Amit Aggarwal, Mark S. Marshall, Darlene S. Barnard, Bharvin K. R. Patel, Louis Stancato, Huimin Bian, Li-Chun Chio, Sean Buchanan, Jian Du, Richard P. Beckmann, Christoph Reinhard, Ricardo Martinez, Gregory D. Plowman, Lei Yan, Shobha N. Bhattachar, Sarah M. Bogner, Maria Jose Lallena, Xiang S. Ye, Jennie L. Walgren, Yu-Hua Hui, Yue Webster, Emiko L. Kreklau, Raquel Torres, Yanzhu Yang, Bartley W. Halstead, Shaoyou Chu
المصدر: Molecular Cancer Therapeutics. 18:2207-2219
مصطلحات موضوعية: Male, 0301 basic medicine, Cancer Research, Aurora inhibitor, Aurora B kinase, Mitosis, Antineoplastic Agents, Apoptosis, macromolecular substances, Biology, 03 medical and health sciences, 0302 clinical medicine, Cell Line, Tumor, medicine, Humans, Kinase activity, Aurora Kinase A, Cell Proliferation, Cancer, medicine.disease, Spindle apparatus, enzymes and coenzymes (carbohydrates), 030104 developmental biology, Oncology, 030220 oncology & carcinogenesis, embryonic structures, Cancer cell, Cancer research, Female, biological phenomena, cell phenomena, and immunity, Cytokinesis, HeLa Cells
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7ea271aab24607f19770d2cdca75d5d3
https://doi.org/10.1158/1535-7163.mct-18-0529 -
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المؤلفون: Burkholder Timothy P, Maria-Carmen Fernandez, Gillig James Ronald, Lourdes Prieto, Miriam del Prado, Bo Tan, Genshi Zhao, Tao Wang, Robert L. Johnson, Yu-Hua Hui, Ken D. Roth, Shobha N. Bhattachar, Sean Buchanan, Xueqian Gong, Sandaruwan Geeganage, Robert L. Shepard, Ming-Shang Kuo, Colin F. Green, Lisa Kays, Wenjuan Wu, Sucai Dong
المصدر: Molecular Cancer Therapeutics. 16:2677-2688
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Retinal Pigment Epithelium, Pharmacology, Inhibitory postsynaptic potential, Niacin, Mice, 03 medical and health sciences, chemistry.chemical_compound, Biosynthesis, medicine, Animals, Humans, Nicotinamide Phosphoribosyltransferase, chemistry.chemical_classification, Chemistry, Cancer, Retinal, medicine.disease, 030104 developmental biology, Nicotinic agonist, Enzyme, Oncology, Cell culture, Cytokines, NAD+ kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f9736cf2bc7ba0f8a4694e69d5907932
https://doi.org/10.1158/1535-7163.mct-16-0674 -
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المؤلفون: Srinivasan Chandrasekhar, Bradley Condon, Matthew Allen Schiffler, Kuklish Steven Lee, Kim Euibong Jemes, Bryan H. Norman, John R. Rizzo, Jeremy Schulenburg York, Kristina M. Campanale, Stefan Jon Thibodeaux, Richard E. Rathmell, Michael J. Hickey, Christopher Groshong, Shobha N. Bhattachar, Norman Earle Hughes, Anita K. Harvey, John G. Luz, Stephen Antonysamy, Scott Alan Jones, Timothy Andrew Woods, Prashant V. Desai, Matthew J. Fisher, Xiao-Peng Yu, Thomas W. Seng
المصدر: Journal of Medicinal Chemistry. 59:194-205
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, medicine.medical_treatment, Biological Availability, Pharmacology, Structure-Activity Relationship, 03 medical and health sciences, Dogs, Microsomes, Drug Discovery, Cytochrome P-450 CYP3A, medicine, Animals, Cytochrome P-450 Enzyme Inhibitors, Humans, Structure–activity relationship, Potency, Cyclooxygenase Inhibitors, IC50, Prostaglandin-E Synthases, ADME, Analgesics, CYP3A4, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Imidazoles, Rats, Intramolecular Oxidoreductases, 030104 developmental biology, Biochemistry, Celecoxib, Molecular Medicine, Prostaglandin E
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المؤلفون: Shobha N. Bhattachar, Aktham Aburub, Xuan Ding, John P. Rose, David C. Sperry, Evelyn D. Lobo
المصدر: Journal of pharmaceutical sciences. 108(1)
مصطلحات موضوعية: Chemistry, Pharmaceutical, education, Pharmaceutical Science, Biological Availability, 02 engineering and technology, 021001 nanoscience & nanotechnology, 030226 pharmacology & pharmacy, Risk Assessment, Risk zone, Bioavailability, Biopharmaceutics, 03 medical and health sciences, 0302 clinical medicine, Pharmaceutical Preparations, Risk Factors, health services administration, Environmental health, Humans, 0210 nano-technology, Risk assessment, health care economics and organizations
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::837ee82826af2ac28174704431303d4f
https://pubmed.ncbi.nlm.nih.gov/30053554 -
7كتاب إلكتروني
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المصدر: AAPS PharmSciTech. 19(1)
مصطلحات موضوعية: Drug, Computer science, media_common.quotation_subject, Drug Compounding, Pharmacology toxicology, Pharmaceutical Science, Pharmacy, 02 engineering and technology, Aquatic Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, Ecology, Evolution, Behavior and Systematics, media_common, Drug compounding, Ecology, Drug discovery, business.industry, General Medicine, 021001 nanoscience & nanotechnology, Laboratory Personnel, Risk analysis (engineering), Pharmaceutical Preparations, Solubility, Drug Design, Drug delivery, Data delivery, 0210 nano-technology, business, Agronomy and Crop Science
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المؤلفون: David M. Bender, Shobha N. Bhattachar, Jeffrey S. Tan
المصدر: Translating Molecules into Medicines ISBN: 9783319500409
مصطلحات موضوعية: Biopharmaceutical, Computer science, Patient centricity, Biochemical engineering, Test plan, AKA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::36dd9ad80cb9573af22b4b5e714b362d
https://doi.org/10.1007/978-3-319-50042-3_7 -
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المؤلفون: David M. Bender, Daniel R. Mudra, Shobha N. Bhattachar, John Morrison
المصدر: AAPS Advances in the Pharmaceutical Sciences Series ISBN: 9783319500409
Translating Molecules into Medicinesمصطلحات موضوعية: business.industry, Medicine, business, Combinatorial chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d9503f5cdd20f18b5255c82a24474927
https://doi.org/10.1007/978-3-319-50042-3