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1
المؤلفون: Johann S. de Bono, Neil Pegg, Karen E. Knudsen, Matthew J. Schiewer, David Taddei, Amanda Swain, Jian Ning, Antje J. Neeb, Suzanne Carreira, Nina Tunariu, Rita Pereira, Ana Ferreira, Mateus Crespo, Susana Miranda, Veronica S. Gil, Gareth W. Harbottle, Don Smyth, Richard Brown, Silvia Paoletta, Jonathan Shannon, Stuart Onions, Jenny Worthington, Stuart Thomson, Jordan Lane, Amy Prosser, Meera Raja, Barbara Young, William West, Denisa Bogdan, Jan Rekowski, Bora Gurel, Ruth Riisnaes, Ines Figueiredo, Abhijit Pal, Saswati N. Chand, Christopher McNair, Wei Yuan, Nigel Brooks, Adam Sharp, Jonathan Welti
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2c73d8a93c6f4a3feb2612ceef314ced
https://doi.org/10.1158/2159-8290.c.6549379 -
2
المؤلفون: Johann S. de Bono, Neil Pegg, Karen E. Knudsen, Matthew J. Schiewer, David Taddei, Amanda Swain, Jian Ning, Antje J. Neeb, Suzanne Carreira, Nina Tunariu, Rita Pereira, Ana Ferreira, Mateus Crespo, Susana Miranda, Veronica S. Gil, Gareth W. Harbottle, Don Smyth, Richard Brown, Silvia Paoletta, Jonathan Shannon, Stuart Onions, Jenny Worthington, Stuart Thomson, Jordan Lane, Amy Prosser, Meera Raja, Barbara Young, William West, Denisa Bogdan, Jan Rekowski, Bora Gurel, Ruth Riisnaes, Ines Figueiredo, Abhijit Pal, Saswati N. Chand, Christopher McNair, Wei Yuan, Nigel Brooks, Adam Sharp, Jonathan Welti
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0d313da933b889d09a6fcaf5a2385ff7
https://doi.org/10.1158/2159-8290.22540441.v1 -
3دورية أكاديمية
المؤلفون: Kenneth A. Jacobson, Zhan-Guo Gao, Silvia Paoletta, Evgeny Kiselev, Saibal Chakraborty, P. Suresh Jayasekara, Ramachandran Balasubramanian, Dilip K. Tosh
المصدر: Computational and Structural Biotechnology Journal, Vol 13, Iss C, Pp 286-298 (2015)
مصطلحات موضوعية: GPCR, Medicinal chemistry, Purines, X-ray structures, Nucleosides, Nucleotides, Polypharmacology, Biotechnology, TP248.13-248.65
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Silvia Paoletta, Dilip K Tosh, Daniela Salvemini, Kenneth A Jacobson
المصدر: PLoS ONE, Vol 9, Iss 5, p e97858 (2014)
وصف الملف: electronic resource
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المؤلفون: Matthew J. Schiewer, Susana Miranda, William West, Suzanne Carreira, Stuart Thomson, Gareth W. Harbottle, Ana Ferreira, Stuart Thomas Onions, Donald Smyth, Nigel Brooks, Jonathan Shannon, Jonathan Welti, Nina Tunariu, Johann S. de Bono, Christopher McNair, Jenny Worthington, Wei Yuan, Karen E. Knudsen, Adam Sharp, Barbara Young, Amy Prosser, Jan Rekowski, Su C, Rita Pereira, Amanda Swain, Jian Ning, Abhijit Pal, Jordan Lane, Ruth Riisnaes, Bora Gurel, Ines Figueiredo, Mateus Crespo, Richard J. C. Brown, Saswati N. Chand, David Michel Adrien Taddei, Denisa Bogdan, Veronica Gil, Silvia Paoletta, Meera Raja, Neil Anthony Pegg, Antje Neeb
المصدر: Cancer discovery. 11(5)
مصطلحات موضوعية: 0301 basic medicine, Male, 03 medical and health sciences, Prostate cancer, Mice, 0302 clinical medicine, Cell Line, Tumor, Gene expression, Androgen Receptor Antagonists, Medicine, Animals, Humans, p300-CBP Transcription Factors, Oxazoles, Cell Proliferation, biology, Cell growth, business.industry, Alternative splicing, Imidazoles, Histone acetyltransferase, medicine.disease, Xenograft Model Antitumor Assays, Biomarker (cell), Bromodomain, Androgen receptor, Prostatic Neoplasms, Castration-Resistant, 030104 developmental biology, Oncology, 030220 oncology & carcinogenesis, biology.protein, Cancer research, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cfbe14e20a3d6b9fa6c1304e667e02ff
https://pubmed.ncbi.nlm.nih.gov/33947717 -
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المؤلفون: Tina C. Wan, Kenneth A. Jacobson, Lili Du, Zhan Guo Gao, Silvia Paoletta, Elizabeth T. Gizewski, Adriaan P. IJzerman, John A. Auchampach, Jacobus P. D. van Veldhoven, Samantha Barbour
المصدر: Purinergic Signalling. 14:59-71
مصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.drug_class, Allosteric regulation, 03 medical and health sciences, Cellular and Molecular Neuroscience, 0302 clinical medicine, medicine, Nucleoside, G protein-coupled receptor, Allosteric modulation, Molecular Biology, biology, Chemistry, Adenosine receptor, Cell Biology, Adenosine, Receptor–ligand kinetics, 030104 developmental biology, Allosteric enzyme, Mechanism of action, Biochemistry, 030220 oncology & carcinogenesis, biology.protein, medicine.symptom, medicine.drug
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المؤلفون: Sonja Kachler, Stefano Moro, Karl-Norbert Klotz, Kenneth A. Jacobson, Giampiero Spalluto, Giorgia Pastorin, Stephanie Federico, Silvia Paoletta, Enrico Margiotta
المساهمون: Federico, Stephanie, Margiotta, Enrico, Paoletta, Silvia, Kachler, Sonja, Klotz, Karl-Norbert, Jacobson, Kenneth A., Pastorin, Giorgia, Moro, Stefano, Spalluto, Giampiero
مصطلحات موضوعية: Pyrimidine, Stereochemistry, Pharmaceutical Science, Conjugated system, 01 natural sciences, Biochemistry, chemistry.chemical_compound, GPCR, Cell surface receptor, Drug Discovery, Moiety, adenosine receptor antagonist, SuMD, Receptor, Pharmacology, 010405 organic chemistry, Organic Chemistry, adenosine receptor antagonists, fluorescent ligands, Adenosine receptor, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Chemistry, chemistry, fluorescent ligand, Molecular Medicine, Pharmacophore, Linker
وصف الملف: STAMPA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6f942729e5c76c897b6059b172c5215
https://europepmc.org/articles/PMC6644567/ -
8
المؤلفون: Barbara Zieger, Eti Alessandra Femia, Christian Gachet, Marco Cattaneo, Gian Marco Podda, Philippe Ohlmann, Silvia Paoletta, Anna Lecchi, Arnaud Dupuis, Katharina Machura, Kenneth A. Jacobson
المصدر: Hämostaseologie. 36:279-283
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_specialty, P2Y receptor, Receptor expression, Hemorrhage, 030204 cardiovascular system & hematology, medicine.disease_cause, Polymorphism, Single Nucleotide, Article, 03 medical and health sciences, 0302 clinical medicine, P2Y12, Internal medicine, medicine, Humans, Genetic Predisposition to Disease, Platelet, Receptor, Mutation, Models, Genetic, business.industry, Models, Immunological, Hematology, Ligand (biochemistry), Adenosine, Receptors, Purinergic P2Y12, 030104 developmental biology, Endocrinology, Blood Platelet Disorders, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::08c80ff624acd04311c3f09b541b54f0
https://doi.org/10.5482/hamo-16-03-0010 -
9
المصدر: Journal of chemical information and modeling. 57(12)
مصطلحات موضوعية: Molecular Docking Simulation, Receptors, Purinergic P2Y1, Structure-Activity Relationship, Drug Discovery, Purinergic P2Y Receptor Antagonists, Humans, Purinergic P2Y Receptor Agonists, Molecular Dynamics Simulation, Ligands, Article, Protein Binding
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المؤلفون: Evgeny Kiselev, Kenneth A. Jacobson, Kevin Trujillo, Silvia Paoletta
المصدر: Bioorganic & Medicinal Chemistry. 23:4056-4064
مصطلحات موضوعية: Models, Molecular, Purinergic P2 Receptor Agonists, Molecular model, Stereochemistry, Ribose, Clinical Biochemistry, Pharmaceutical Science, Molecular Dynamics Simulation, Ligands, Biochemistry, Article, Phosphates, Nucleobase, Structure-Activity Relationship, Drug Discovery, Humans, Nucleotide, Homology modeling, Receptor, Molecular Biology, G protein-coupled receptor, chemistry.chemical_classification, Binding Sites, Receptors, Purinergic P2, Chemistry, Organic Chemistry, Molecular Docking Simulation, Glucose, Docking (molecular), Drug Design, Molecular Medicine, Uracil nucleotide