-
1دورية أكاديمية
المؤلفون: Logan Tillery, Kayleigh Barrett, Jenna Goldstein, Jared W Lassner, Bram Osterhout, Nathan L Tran, Lily Xu, Ryan M Young, Justin Craig, Ian Chun, David M Dranow, Jan Abendroth, Silvia L Delker, Douglas R Davies, Stephen J Mayclin, Brandy Calhoun, Madison J Bolejack, Bart Staker, Sandhya Subramanian, Isabelle Phan, Donald D Lorimer, Peter J Myler, Thomas E Edwards, Dennis E Kyle, Christopher A Rice, James C Morris, James W Leahy, Roman Manetsch, Lynn K Barrett, Craig L Smith, Wesley C Van Voorhis
المصدر: PLoS ONE, Vol 16, Iss 3, p e0241738 (2021)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1932-6203
-
2
المؤلفون: Sneha Basak, Yong Li, Suyuan Tao, Fereidoon Daryaee, Jonathan Merino, Chendi Gu, Silvia L. Delker, Jenny N. Phan, Thomas E. Edwards, Stephen G. Walker, Peter J. Tonge
المصدر: Journal of medicinal chemistry. 65(17)
مصطلحات موضوعية: Kinetics, Drug Discovery, Gram-Negative Bacteria, Pseudomonas aeruginosa, Molecular Medicine, Enzyme Inhibitors, Amidohydrolases, Anti-Bacterial Agents
-
3
المؤلفون: Philip P Chamberlain, Maria Wang, Yoshinori Hirano, Brian E. Cathers, Gilles Carmel, Toshio Hakoshima, Hiroshi Handa, Barbra Pagarigan, Emily Rychak, Yan J Ren, Barbara Chie-Leon, Silvia L. Delker, Laura G. Corral, Tomoyuki Mori, Takumi Ito, Thomas O. Daniel, Antonia Lopez-Girona, Karen Miller, Hideki Ando, Mariko Riley
المصدر: Nature Structural & Molecular Biology. 21:803-809
مصطلحات موضوعية: Protein Conformation, Ubiquitin-Protein Ligases, Molecular Sequence Data, Angiogenesis Inhibitors, Crystallography, X-Ray, Mice, DDB1, Ubiquitin, Structural Biology, medicine, Animals, Humans, Amino Acid Sequence, Lenalidomide, Molecular Biology, Adaptor Proteins, Signal Transducing, biology, Cereblon, Protein Cereblon, IKZF3, Protein Structure, Tertiary, Thalidomide, Ubiquitin ligase, DNA-Binding Proteins, Molecular Docking Simulation, Biochemistry, biology.protein, Cancer research, Sequence Alignment, Peptide Hydrolases, Protein Binding, medicine.drug
-
4
المؤلفون: Jan J. Mataka, Silvia L. Delker, Thomas L. Poulos, James M. Kraus, Kristin J. Labby, Richard B. Silverman, Huiying Li, Pavel Martásek, Haitao Ji, Linda J. Roman, Fengtian Xue
المصدر: Bioorganic & Medicinal Chemistry. 21:1333-1343
مصطلحات موضوعية: Cyclopropanes, Nitric Oxide Synthase Type III, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Nitric Oxide Synthase Type I, Crystallography, X-Ray, Biochemistry, Article, Mice, Structure-Activity Relationship, Enos, Drug Discovery, Animals, Structure–activity relationship, Enzyme Inhibitors, Binding site, Molecular Biology, Binding Sites, biology, Chemistry, Organic Chemistry, Oxidoreductase inhibitor, biology.organism_classification, Recombinant Proteins, In vitro, Enzyme assay, Protein Structure, Tertiary, Molecular Docking Simulation, biology.protein, Molecular Medicine
-
5
المؤلفون: Fengtian Xue, Richard B. Silverman, Kristin J. Labby, Pavel Martásek, Thomas L. Poulos, Haitao Ji, Guoyao Xia, Huiying Li, Linda J. Roman, James M. Kraus, Silvia L. Delker, Jan J. Mataka
المصدر: Journal of Medicinal Chemistry. 54:6399-6403
مصطلحات موضوعية: Models, Molecular, inorganic chemicals, Pyrrolidines, Nitric Oxide Synthase Type III, Stereochemistry, Stereoisomerism, Nitric Oxide Synthase Type I, Plasma protein binding, Crystallography, X-Ray, Endothelial NOS, Article, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, Catalytic Domain, Drug Discovery, Animals, Molecule, Structure–activity relationship, Molecular Structure, Oxidoreductase inhibitor, musculoskeletal system, Rats, body regions, nervous system, chemistry, cardiovascular system, Molecular Medicine, Protein Binding
-
6
المؤلفون: Linda J. Roman, Thomas L. Poulos, Pavel Martásek, Silvia L. Delker, Richard B. Silverman, Haitao Ji, Huiying Li
المصدر: Journal of Medicinal Chemistry. 53:7804-7824
مصطلحات موضوعية: Models, Molecular, Pyrrolidines, Protein Conformation, Stereochemistry, Aminopyridines, Stereoisomerism, Nitric Oxide Synthase Type I, Crystallography, X-Ray, Article, Structure-Activity Relationship, chemistry.chemical_compound, Oxidoreductase, Catalytic Domain, Drug Discovery, Animals, Structure–activity relationship, chemistry.chemical_classification, biology, Active site, Rats, Isoenzymes, Enzyme, chemistry, Drug Design, biology.protein, Alkoxy group, Molecular Medicine, Cattle, Selectivity, Protein Binding, 2-Aminopyridine
-
7
المؤلفون: Lindsay C. McDermott, Silvia L. Delker, Pamela J. Bjorkman, Anthony P. West, Malcolm W. Kennedy
المصدر: Journal of Structural Biology. 148:205-213
مصطلحات موضوعية: Models, Molecular, Glycosylation, Stereochemistry, Structural similarity, Polyethylene glycol, Crystal structure, Crystallography, X-Ray, Ligands, Protein Structure, Secondary, Polyethylene Glycols, chemistry.chemical_compound, Adipokines, Structural Biology, Humans, Molecule, Binding site, Fluorescent Dyes, Glycoproteins, Dansyl Compounds, chemistry.chemical_classification, Binding Sites, Fatty Acids, Ligand (biochemistry), Recombinant Proteins, Zinc, Crystallography, chemistry, Carrier Proteins, Peptides, Glycoprotein
-
8
المؤلفون: Richard B. Silverman, Carla Plaza, Soosung Kang, Qing Jing, Haitao Ji, Thomas L. Poulos, Huiying Li, He Huang, Silvia L. Delker, Joumana Jamal
المصدر: Biochemistry
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Protein Conformation, Endothelial NOS, 01 natural sciences, Biochemistry, Article, Conserved sequence, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, Protein structure, X-Ray Diffraction, Enos, Animals, Binding site, Tyrosine, Enzyme Inhibitors, Heme, Conserved Sequence, 030304 developmental biology, 0303 health sciences, Binding Sites, biology, Molecular Structure, 010405 organic chemistry, biology.organism_classification, 0104 chemical sciences, Rats, Nitric oxide synthase, Isoenzymes, chemistry, biology.protein, Cattle, Nitric Oxide Synthase, Crystallization
-
9
المؤلفون: Li Xu, Meg Mccarrick, Neil R. D'sidocky, Veronique Plantevin Krenitsky, Lisa Nadolny, Yoshitaka Satoh, April Bai, Sayee G. Hegde, Brian E. Cathers, Jonathan Wright, Ronald Albers, John Sapienza, Steven S. Clareen, David Giegel, Rachel Fan, Robert Hilgraf, Michael A. Shirley, Heather Raymon, Maria Celeridad, Leticia Ayala, Jason Katz, Philip P Chamberlain, Brent Benish, Brydon L. Bennett, Tracey Bodine, Mercedes Delgado, Sogole Bahmanyar, Mehran F. Moghaddam, Silvia L. Delker, Yang Tang, Kate Blease, Oleg Khatsenko, Jeff Lachowitzer, Jeff Muir
المصدر: Bioorganicmedicinal chemistry letters. 22(3)
مصطلحات موضوعية: Models, Molecular, Anti fibrotic, MAP Kinase Kinase 4, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Pharmacology, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, Dogs, Catalytic Domain, Drug Discovery, Potency, Structure–activity relationship, Animals, Enzyme Inhibitors, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Haplorhini, Multiple species, Cyclohexanols, Jnk inhibitor, Idiopathic Pulmonary Fibrosis, Rats, Enzyme Activation, Orally active, Plasma exposure, Purines, Molecular Medicine, Aminopurine
-
10
المؤلفون: Richard B. Silverman, Huiying Li, Linda J. Roman, Fengtian Xue, Jianguo Fang, Thomas L. Poulos, Silvia L. Delker, Pavel Martásek
المصدر: Journal of medicinal chemistry. 54(7)
مصطلحات موضوعية: Gene isoform, Models, Molecular, Cell Membrane Permeability, Membrane permeability, Stereochemistry, Protein Conformation, Aminopyridines, Nitric Oxide Synthase Type I, Article, chemistry.chemical_compound, Mice, Enos, Drug Discovery, Animals, Humans, Pterin, Enzyme Inhibitors, biology, Chemistry, HEK 293 cells, Substrate (chemistry), biology.organism_classification, Rats, Membrane, HEK293 Cells, Drug Design, Molecular Medicine, Cattle