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1
المؤلفون: Julian Blagg, Butrus Atrash, K. Boxall, Vassilios Bavetsias, Jessica Schmitt, Nathan J. Brown, Richard Bayliss, Sian Avery, Yolanda Pérez-Fuertes, Katherine Bush, Amar Joshi, Simon Crumpler, Spiros Linardopoulos, Rosemary Burke, Florence I. Raynaud, Chongbo Sun, Amir Faisal, Paul Workman, Alan T. Henley, Magda Kosmopoulou
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Gene isoform, Male, Indoles, Stereochemistry, Mutant, Aurora A kinase, macromolecular substances, Article, Protein–protein interaction, Substrate Specificity, chemistry.chemical_compound, Mice, Drug Stability, Catalytic Domain, Drug Discovery, Pyridine, Transferase, Animals, Aurora Kinase B, Humans, Protein Kinase Inhibitors, Aurora Kinase A, Chemistry, Wild type, Imidazoles, HCT116 Cells, Isoenzymes, Molecular Docking Simulation, enzymes and coenzymes (carbohydrates), Biochemistry, Drug Design, embryonic structures, Molecular Medicine, biological phenomena, cell phenomena, and immunity, Selectivity
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2
المؤلفون: Nathan J. Brown, Richard Bayliss, Jasmeen Oberoi, Mark W. Richards, Julian Blagg, Simon Crumpler
المصدر: Journal of Biological Chemistry. 285:39348-39358
مصطلحات موضوعية: Ubiquitin-Protein Ligases, Molecular Sequence Data, Antephase Checkpoint, Mitosis, Cell Cycle Proteins, Biology, Crystallography, X-Ray, Ligands, Biochemistry, chemistry.chemical_compound, Protein structure, CHFR, Humans, Amino Acid Sequence, Binding site, Poly-ADP-Ribose Binding Proteins, Molecular Biology, Zinc finger, Adenosine Diphosphate Ribose, Binding Sites, Adenosine diphosphate ribose, Temperature, Zinc Fingers, Cell Biology, Surface Plasmon Resonance, Neoplasm Proteins, Protein Structure, Tertiary, Cell biology, Adenosine Diphosphate, Zinc, chemistry, Structural biology, Protein Structure and Folding, Protein Binding, Binding domain
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa0137df5eb70aed56e60ad9bfb5b7de
https://doi.org/10.1074/jbc.m110.159855 -
3
المؤلفون: Edward McDonald, Simon Crumpler, Julian Blagg, Mark Pichowicz
المصدر: Tetrahedron. 66:2398-2403
مصطلحات موضوعية: Primary (chemistry), Nucleophilic aromatic substitution, Chemistry, Organic Chemistry, Drug Discovery, Nucleophilic substitution, Organic chemistry, Biochemistry, Chemical synthesis, Microwave assisted
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4
المؤلفون: Carl Berthelette, Florence Lee, Cheuk K. Lau, Kathy Macfarlane, Simon Crumpler
المصدر: Synlett. :2281-2286
مصطلحات موضوعية: chemistry.chemical_classification, chemistry, Stereochemistry, Organic Chemistry, Glycoside, Spongistatin 1
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::1287e257b637812aada1b705d5956c1e
https://doi.org/10.1055/s-2004-831334 -
5
المؤلفون: Magda Kosmopoulou, Alexis De Haven Brandon, Julian Blagg, Sian Avery, Spiros Linardopoulos, Richard Bayliss, Butrus Atrash, Simon Crumpler, Peter Sheldrake, Vassilios Bavetsias, Suzanne A. Eccles, Nathan J. Brown, Katherine Bush, Paul Workman, Melanie Valenti, Alan T. Henley, Andrew S. Moore, Gary Box, Amir Faisal, Florence I. Raynaud, Chongbo Sun
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Male, Models, Molecular, ERG1 Potassium Channel, Pyridines, Transplantation, Heterologous, Aurora inhibitor, Administration, Oral, Biological Availability, Antineoplastic Agents, Pharmacology, Protein Serine-Threonine Kinases, Article, Rats, Sprague-Dawley, Mice, Aurora kinase, fluids and secretions, Aurora Kinases, hemic and lymphatic diseases, Cell Line, Tumor, Drug Discovery, Animals, Aurora Kinase B, Humans, Aurora Kinase A, Mice, Inbred BALB C, Chemistry, Kinase, Imidazoles, Myeloid leukemia, hemic and immune systems, Ether-A-Go-Go Potassium Channels, Rats, Transplantation, Leukemia, Myeloid, Acute, fms-Like Tyrosine Kinase 3, Purines, Fms-Like Tyrosine Kinase 3, embryonic structures, Mutation, Microsomes, Liver, Molecular Medicine, Pyrazoles, Female, Drug Screening Assays, Antitumor, Neoplasm Transplantation
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6
المؤلفون: Paul Czodrowski, Andree Blaukat, Frank Stieber, Julian Blagg, Djordje Musil, Felix Rohdich, Simon Crumpler, Rosemary Burke, Michael Busch, Kai Schiemann, Sharon Gowan, Michel Calderini, Stephanie Simon, Richard Schneider, Suzanne A. Eccles, Robert TePoele, Maria-Jesus Ortiz-Ruiz, Oliver Poeschke, Trevor Clive Dale, Florence I. Raynaud, Klaus Urbahns, Olajumoke Adeniji-Popoola, Wolfgang Kaufmann, Daniel Schwarz, Klaus Schneider, Aurélie Mallinger, Rahul S. Samant, Christian Rink, Christina Esdar, Mark Stubbs, Dennis Waalboer, Paul Workman, Paul A. Clarke, Dirk Wienke
المصدر: Cancer Research. 76:3025-3025
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Kinase, Wnt signaling pathway, Cancer, Context (language use), Pharmacology, Biology, medicine.disease, MED12, 03 medical and health sciences, 030104 developmental biology, Mediator, Oncology, In vivo, medicine, Cyclin-dependent kinase 8
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::205048a11978c437f58e8b431a90eeaa
https://doi.org/10.1158/1538-7445.am2016-3025 -
7
المؤلفون: Edward McDonald, Julian Blagg, Simon Crumpler, Mark Pichowicz
المصدر: ChemInform. 41
مصطلحات موضوعية: Chemistry, General Medicine, Microwave assisted, Combinatorial chemistry
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8
المؤلفون: Kathy Macfarlane, Simon Crumpler, Carl Berthelette, Cheuk K. Lau, Florence Lee
المصدر: ChemInform. 36
مصطلحات موضوعية: Stereochemistry, Chemistry, General Medicine, Combinatorial chemistry, Spongistatin 1
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9
المؤلفون: C. Gustaf Saluste, Richard J. Whitby, Simon Crumpler, Mark Furber
المصدر: ChemInform. 36
مصطلحات موضوعية: Chemistry, chemistry.chemical_element, General Medicine, Combinatorial chemistry, Palladium, Catalysis
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10
المؤلفون: Mark Furber, Simon Crumpler, C. Gustaf Saluste, Richard J. Whitby
المصدر: Tetrahedron Letters. 45:6995-6996
مصطلحات موضوعية: inorganic chemicals, Ortho position, Aryl, Organic Chemistry, chemistry.chemical_element, Alcohol, Biochemistry, Amidine, chemistry.chemical_compound, chemistry, Yield (chemistry), Drug Discovery, Organic chemistry, Amine gas treating, Palladium