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1دورية أكاديمية
المؤلفون: Klara Livia Valko, Simon Teague, Charles Pudgeon
المصدر: ADMET and DMPK, Vol 6, Iss 3, Pp 267-268 (2018)
مصطلحات موضوعية: erratum, estimation of volume of distribution, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2
المؤلفون: Jayne E. Hastedt, Per Bäckman, Antonio Cabal, Andy Clark, Carsten Ehrhardt, Ben Forbes, Anthony J. Hickey, Guenther Hochhaus, Wenlei Jiang, Stavros Kassinos, Philip J. Kuehl, David Prime, Yoen-Ju Son, Simon Teague, Ulrika Tehler, Jennifer Wylie
المصدر: Molecular Pharmaceutics. 19:2032-2039
مصطلحات موضوعية: Pharmaceutical Preparations, Solubility, Administration, Inhalation, Drug Discovery, Administration, Oral, Pharmaceutical Science, Molecular Medicine, Permeability, Biopharmaceutics
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3
المؤلفون: Christopher R. Wellaway, Ian R. Baldwin, Paul Bamborough, Daniel Barker, Michelle A. Bartholomew, Chun-wa Chung, Birgit Dümpelfeld, John P. Evans, Neal J. Fazakerley, Paul Homes, Steven P. Keeling, Xiao Q. Lewell, Finlay W. McNab, Joanne Morley, Deborah Needham, Margarete Neu, Antoon J. M. van Oosterhout, Anshu Pal, Friedrich B. M. Reinhard, Francesco Rianjongdee, Craig M. Robertson, Paul Rowland, Rishi R. Shah, Emma B. Sherriff, Lisa A. Sloan, Simon Teague, Daniel A. Thomas, Natalie Wellaway, Justyna Wojno-Picon, James M. Woolven, Diane M. Coe
المصدر: Journal of Medicinal Chemistry. 65:633-664
مصطلحات موضوعية: Models, Molecular, Mice, Inbred BALB C, Binding Sites, Aldehyde Oxidase, Molecular Docking Simulation, Mice, Structure-Activity Relationship, Drug Delivery Systems, Liver, Drug Discovery, Quinazolines, Animals, Humans, Janus Kinase Inhibitors, Molecular Medicine, Administration, Intravenous, Female, Lung, Administration, Intranasal
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4
المؤلفون: Brian Farrer, Eve Robinson, Joseph Marchand, Ian S. Gilmore, Meredith Earl, Rasmus Havelund, Diane M. Coe, Doug Ball, Dave Hassall, Simon Teague, Heather Reid, Rebecca Terry, Paul Giffen, Peter S. Marshall
المصدر: The Analyst. 146:3378-3390
مصطلحات موضوعية: Drug, media_common.quotation_subject, Context (language use), Multimodal Imaging, 01 natural sciences, Biochemistry, Analytical Chemistry, Excipients, Delayed-Action Preparations, 03 medical and health sciences, Therapeutic index, Electrochemistry, Animals, Environmental Chemistry, Distribution (pharmacology), Medicine, Particle Size, Microparticle, Lung, Spectroscopy, 030304 developmental biology, media_common, 0303 health sciences, business.industry, 010401 analytical chemistry, Controlled release, Rats, 0104 chemical sciences, Drug delivery, business, Biomedical engineering
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5
المؤلفون: Joe Coyle, Lee William Page, Dave Clapham, Karen Affleck, Paul N. Mortenson, Jonathan P. Hutchinson, Ashley Paul Hancock, Melanie Leveridge, Joelle Le, Heather Hobbs, David Norton, Rachel McMenamin, Simon Teague, Emma Sherriff, Linda J. Russell, Sorif Uddin, Caroline Richardson, Anne Cleasby, Simon Teanby Hodgson, Philip J. Day, Martyn Frederickson, Gordon Saxty
المصدر: Med. Chem. Commun.. 5:134-141
مصطلحات موضوعية: Pharmacology, biology, Stereochemistry, Chemistry, Organic Chemistry, Fragment-based lead discovery, Pharmaceutical Science, Prostaglandin D2 synthase, Crystal structure, Ligand (biochemistry), Biochemistry, Small molecule, Protein structure, In vivo, Drug Discovery, biology.protein, Molecular Medicine, Molecule
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3f3850d001e5b02755bbbe21405c11b8
https://doi.org/10.1039/c3md00280b -
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المؤلفون: Simon Teague, Klára Valkó
المصدر: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences. 110
مصطلحات موضوعية: Drug, media_common.quotation_subject, Pharmaceutical Science, Biological Availability, Plasma protein binding, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, 0302 clinical medicine, Cytochrome P-450 Enzyme System, In vivo, Biomimetics, Albumins, Potency, Humans, Computer Simulation, Chromatography, High Pressure Liquid, Phospholipids, media_common, Whole blood, Volume of distribution, Dose-Response Relationship, Drug, Chemistry, Drug discovery, In vitro, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, Microsomes, Liver, Protein Binding
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المؤلفون: Simon Teague, Klára Valkó, Charles Pudgeon
المصدر: ADMET and DMPK
Volume 6
Issue 3
ADMET and DMPK, Vol 6, Iss 3, Pp 267-268 (2018)مصطلحات موضوعية: Drug discovery, Chemistry, lcsh:RM1-950, Medicine (miscellaneous), Plasma protein binding, In vitro, lcsh:Therapeutics. Pharmacology, IAM MB/PB technology, Chemistry (miscellaneous), In vivo, Biophysics, Distribution (pharmacology), Pharmacology (medical), Membrane binding, General Pharmacology, Toxicology and Pharmaceutics, erratum, estimation of volume of distribution
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::df0ef9ac1688af0f7fd088db136a1447
https://doi.org/10.5599/admet.568 -
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المؤلفون: Laurie J. Gordon, Gemma V. Puckey, Wyman Paul Adrian, David John Nash, Richard Blunt, Hugh J. Herdon, Simon Teague, Victoria Hadden, Stefano Fontana, Amanda Johns, Roderick A. Porter
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6176-6179
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Glycine, Pharmaceutical Science, Glycine Plasma Membrane Transport Proteins, Biochemistry, Glycine transporter, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, Animals, Humans, Structure–activity relationship, Solubility, Molecular Biology, Chemistry, Organic Chemistry, Combinatorial chemistry, Rats, Bioavailability, Lipophilicity, Molecular Medicine, Selectivity
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المؤلفون: Simon Teague, Klára Valkó, Charles Pidgeon
المصدر: ADMET and DMPK, Vol 5, Iss 1, Pp 14-38 (2017)
ADMET and DMPK
Volume 5
Issue 1مصطلحات موضوعية: Chromatography, Drug discovery, Chemistry, lcsh:RM1-950, 010401 analytical chemistry, Medicine (miscellaneous), Drug efficiency, Plasma protein binding, Biomimetic properties by HPLC, unbound volume of distribution, in vivo distribution, 01 natural sciences, In vitro, 0104 chemical sciences, 03 medical and health sciences, lcsh:Therapeutics. Pharmacology, 0302 clinical medicine, Biochemistry, Chemistry (miscellaneous), In vivo, Lipophilic efficiency, 030220 oncology & carcinogenesis, Potency, Pharmacology (medical), Membrane binding, volume of distribution, drug efficiency, membrane binding, protein binding, IAM, General Pharmacology, Toxicology and Pharmaceutics
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8dc8a261b9b179948e988cd3ca72293c
https://doi.org/10.5599/admet.5.1.373 -
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المؤلفون: Cristian Salvagno, James N.C. Kew, Caterina Virginio, Beatrice Oliosi, Simon Teague, Andrew P. Lightfoot, Anna Maria Capelli, Elisa Di Lenarda, Laura Castelletti
المصدر: Bioorganicmedicinal chemistry letters. 20(15)
مصطلحات موضوعية: Models, Molecular, Molecular model, Databases, Factual, alpha7 Nicotinic Acetylcholine Receptor, In silico, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Receptors, Nicotinic, complex mixtures, Biochemistry, Cell Line, Structure-Activity Relationship, Allosteric Regulation, mental disorders, Drug Discovery, Screening method, Structure–activity relationship, Animals, Humans, Molecular Biology, Virtual screening, Chemistry, Phenylurea Compounds, Organic Chemistry, Isoxazoles, Rats, nervous system, Microsomes, Liver, Molecular Medicine, Pharmacophore, α7 nachr, psychological phenomena and processes