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المؤلفون: Melanie Washington, Lisa E. Ranshaw, Philip Alan Skone, James A. Bull, David W. Brown, Ilaria Giordano, Richard Martyn Angell, Vipulkumar Kantibhai Patel, Smith Kathryn Jane, Anthony William James Cooper, Martin Sims, Emma Vickerstaff, John A. Christopher, Lucy Hind, Inder Bhamra, Paul Bamborough, Lynsey H. Fazal
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:4363-4368
مصطلحات موضوعية: Models, Molecular, Indazoles, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Carboxamide, Biochemistry, chemistry.chemical_compound, Pharmacokinetics, Drug Discovery, medicine, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Kinase, Organic Chemistry, Enzyme, Lymphocyte Specific Protein Tyrosine Kinase p56(lck), Enzyme inhibitor, biology.protein, Molecular Medicine, Amine gas treating, Tyrosine kinase
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المؤلفون: Jeremy John Payne, Geoff W. Mellor, Smith Kathryn Jane, Richard A. Williamson, Sebastien Andre Campos, Geoffrey J. Cutler, Caroline Whitworth, Mary A. Morse, Michael David Barker, Heather Hobbs, Rick P. C. Cousins, Duncan S. Holmes, Daniel Terence Tape, Paul Bamborough, John Martin Pritchard, John Liddle, Chris Ioannou
المصدر: Bioorganicmedicinal chemistry letters. 19(9)
مصطلحات موضوعية: Models, Molecular, Cellular activity, Indoles, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Tumor cells, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, Adenosine Triphosphate, Drug Discovery, Humans, Molecular Biology, Tumor necrosis factor α, chemistry.chemical_classification, Sulfonamides, Binding Sites, Molecular Structure, Kinase, Organic Chemistry, In vitro, Sulfonamide, I-kappa B Kinase, Enzyme, chemistry, Models, Chemical, Drug Design, Molecular Medicine, Protein Binding
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المؤلفون: Penny A. Smee, Stephen Sean Flack, Steve Ludbrook, Ann Louise Walker, Timothy Longstaff, Mark James Bamford, Paul Bamborough, Katherine Louise Jones, Chun-wa Chung, Rosannah Pearson, Tony D. Angell, Dramane I. Laine, Stuart G. Cockerill, Smith Kathryn Jane, Richard Martyn Angell, Don O. Somers
المصدر: Bioorganicmedicinal chemistry letters. 18(15)
مصطلحات موضوعية: Lipopolysaccharides, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, Naphthalenes, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Mitogen-Activated Protein Kinase 14, chemistry.chemical_compound, Structure-Activity Relationship, Amide, Drug Discovery, medicine, Transferase, Structure–activity relationship, Combinatorial Chemistry Techniques, Binding site, Amino Acids, Molecular Biology, Binding Sites, Molecular Structure, Kinase, Organic Chemistry, Biphenyl Compounds, Biological activity, Amides, chemistry, Drug Design, Molecular Medicine, Pyrazoles
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المؤلفون: Duncan S. Holmes, Ann Louise Walker, Katherine Louise Jones, Chris D. Edwards, Dramane I. Laine, Don O. Somers, Paul Bamborough, Smith Kathryn Jane, Shila Patel, Jacky B. Buckton, Suzanne J. deBoeck, Richard Martyn Angell, Penny A. Smee, Nicola Mary Aston, Stuart G. Cockerill
المصدر: Bioorganicmedicinal chemistry letters. 18(15)
مصطلحات موضوعية: Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Administration, Oral, Carboxamide, Crystallography, X-Ray, Biochemistry, Mitogen-Activated Protein Kinase 14, chemistry.chemical_compound, In vivo, Amide, Drug Discovery, medicine, Transferase, Animals, Combinatorial Chemistry Techniques, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, Biphenyl, biology, Molecular Structure, Chemistry, Organic Chemistry, Biphenyl Compounds, Rats, Disease Models, Animal, Enzyme, Mitogen-activated protein kinase, Benzamides, biology.protein, Molecular Medicine
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المؤلفون: Richard Martyn Angell, David W. Brown, Katherine Louise Jones, Smith Kathryn Jane, Ann Louise Walker, Penny A. Smee, Tim Longstaff, Paul Bamborough, Tony D. Angell, Stuart G. Cockerill, Chris D. Edwards, Don O. Somers, Murray J. B. Brown, Jacky B. Buckton, Malcolm Willson
المصدر: Bioorganicmedicinal chemistry letters. 18(1)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, p38 mitogen-activated protein kinases, Clinical Biochemistry, Biphenyl derivatives, Molecular Conformation, Pharmaceutical Science, Administration, Oral, Non-specific serine/threonine protein kinase, Crystallography, X-Ray, Biochemistry, p38 Mitogen-Activated Protein Kinases, Piperazines, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Amide, Drug Discovery, Animals, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, Biphenyl, Oxadiazoles, Organic Chemistry, Biphenyl Compounds, Amides, Arthritis, Experimental, Rats, Enzyme, chemistry, Molecular Medicine, Protein Binding