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1دورية أكاديمية
المؤلفون: Amélie Le Bihan, Ruben de Kanter, Iñigo Angulo-Barturen, Christoph Binkert, Christoph Boss, Reto Brun, Ralf Brunner, Stephan Buchmann, Jeremy Burrows, Koen J Dechering, Michael Delves, Sonja Ewerling, Santiago Ferrer, Christoph Fischli, Francisco Javier Gamo-Benito, Nina F Gnädig, Bibia Heidmann, María Belén Jiménez-Díaz, Didier Leroy, Maria Santos Martínez, Solange Meyer, Joerg J Moehrle, Caroline L Ng, Rintis Noviyanti, Andrea Ruecker, Laura María Sanz, Robert W Sauerwein, Christian Scheurer, Sarah Schleiferboeck, Robert Sinden, Christopher Snyder, Judith Straimer, Grennady Wirjanata, Jutta Marfurt, Ric N Price, Thomas Weller, Walter Fischli, David A Fidock, Martine Clozel, Sergio Wittlin
المصدر: PLoS Medicine, Vol 13, Iss 10, p e1002138 (2016)
مصطلحات موضوعية: Medicine
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Christoph Boss, Reto Brun, Walter Fischli, Christoph Binkert, Solange Meyer, Lars Prade, Luke Harris, Lionel Coppex, Corinna Grisostomi, Olivier Corminboeuf, Jean-Marc Bourgeois, Rocco Furnari, Sylvia Richard-Bildstein, Thomas Weller
المصدر: CHIMIA, Vol 58, Iss 9 (2004)
مصطلحات موضوعية: Aspartic proteases, Enzyme inhibitors, Malaria, Medicinal chemistry, Plasmepsin ii (pmii), Chemistry, QD1-999
وصف الملف: electronic resource
Relation: https://chimia.ch/chimia/article/view/3880; https://doaj.org/toc/0009-4293; https://doaj.org/toc/2673-2424
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المؤلفون: Christoph Binkert, Christoph Fischli, Christoph Boss, Solange Meyer, Sophie Racine, Romain Siegrist, Sergio Wittlin, Hamed Aissaoui, Claire-Lise Ciana, Ruben de Kanter, Léo Marx
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:658-662
مصطلحات موضوعية: Scaffold, Plasmodium berghei, Stereochemistry, Peptidomimetic, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Hydroxylamine, Mannich base, Amodiaquine, Biochemistry, Antimalarials, Inhibitory Concentration 50, Mice, chemistry.chemical_compound, In vivo, Drug Discovery, Ethylamines, medicine, Animals, Aspartic Acid Endopeptidases, Molecular Biology, Protease, Molecular Structure, Organic Chemistry, Combinatorial chemistry, Malaria, Disease Models, Animal, chemistry, Molecular Medicine, Amine gas treating, Pharmacophore, medicine.drug
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المؤلفون: W. Bernd Schweizer, François Diederich, Valentina Aureggi, Daniel Bur, Veronika Ehmke, Reto Brun, J. Wieland, Matthias Rottmann, Bruno Bernet, Céline Freymond, Solange Meyer, Bernhard Breit
المصدر: Chemistry - A European Journal. 19:155-164
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Plasmodium falciparum, Plasmepsin, Catalysis, Heptanes, Antimalarials, Bridged Bicyclo Compounds, Molecular recognition, Formaldehyde, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Cathepsin, chemistry.chemical_classification, Aza Compounds, biology, Chemistry, Organic Chemistry, Stereoisomerism, General Chemistry, biology.organism_classification, In vitro, Enzyme, Biochemistry, Selectivity, Hydroformylation
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المؤلفون: Julien Trollux, Aurelien Merot, Hamed Aissaoui, Christoph Binkert, Alexandre Flock, Stephane Delahaye, Christoph Fischli, Amélie Le Bihan, Christoph Boss, Aude Bauer, Reto Brun, Claire-Lise Ciana, Malory Girault, Sergio Wittlin, Sabrina Peixoto, Sophie Malrieu, Olivier Corminboeuf, Thomas Weller, Claire Hinder, Romain Siegrist, Saskia Mamzed, Claire Dollinger, Marie-Céline Frantz, Walter Fischli, Nolwenn Petit, Solange Meyer, Corinna Grisostomi, Astrid Friedli, Stephanie Bazire, Nathalie Amaral, Bibia Heidmann, Gael Jacob, Cédric Bürki
المصدر: ChemMedChem. 11(18)
مصطلحات موضوعية: 0301 basic medicine, Drug, Phenotypic screening, media_common.quotation_subject, Population, Plasmodium falciparum, Biology, Pharmacology, 01 natural sciences, Biochemistry, Piperazines, 03 medical and health sciences, Antimalarials, Structure-Activity Relationship, Parasitic Sensitivity Tests, Drug Discovery, medicine, General Pharmacology, Toxicology and Pharmaceutics, Artemisinin, education, media_common, education.field_of_study, Acrylamides, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Organic Chemistry, medicine.disease, 0104 chemical sciences, Malaria, 030104 developmental biology, Mechanism of action, Molecular Medicine, Classical pharmacology, medicine.symptom, Drug metabolism, medicine.drug
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المؤلفون: Thomas Weller, Jeremy N. Burrows, David A. Fidock, Sergio Wittlin, Rintis Noviyanti, Robert W. Sauerwein, Grennady Wirjanata, Robert E. Sinden, María Santos Martínez, Christoph Binkert, Christopher Snyder, Nina F. Gnädig, Stephan Buchmann, Ruben de Kanter, Andrea Ruecker, Christoph Fischli, Michael J. Delves, Joerg J. Moehrle, Iñigo Angulo-Barturen, Koen J. Dechering, Christian Scheurer, Francisco Javier Gamo Benito, Solange Meyer, Laura M. Sanz, Christoph Boss, Sarah Schleiferboeck, Martine Clozel, Sonja Ewerling, Caroline L. Ng, Reto Brun, María Belén Jiménez-Díaz, Didier Leroy, Jutta Marfurt, Santiago Ferrer, Walter Fischli, Amélie Le Bihan, Judith Straimer, Bibia Heidmann, Ric N. Price, Ralf Brunner
المساهمون: Medicines for Malaria Venture
المصدر: Plos Medicine, 13, e1002138
Plos Medicine, 13, 10, pp. e1002138
PLoS Medicine
PLoS Medicine, Vol 13, Iss 10, p e1002138 (2016)مصطلحات موضوعية: 0301 basic medicine, Plasmodium, Physiology, Plasmodium berghei, Plasmodium vivax, lnfectious Diseases and Global Health Radboud Institute for Molecular Life Sciences [Radboudumc 4], Pharmacology, Gametocytes, Piperazines, Mice, Animal Cells, Mice, Inbred NOD, Medicine and Health Sciences, Artemisinin, GeneralLiterature_REFERENCE(e.g.,dictionaries,encyclopedias,glossaries), Protozoans, biology, Pharmaceutics, Malarial Parasites, Drugs, General Medicine, 11 Medical And Health Sciences, Animal Models, Hematology, Artemisinins, 3. Good health, Body Fluids, Blood, Medicine, Female, Cellular Types, Anatomy, Multidrug Resistance-Associated Proteins, medicine.drug, Research Article, Combination therapy, 030106 microbiology, Plasmodium falciparum, Cmax, Mouse Models, Microbial Sensitivity Tests, Research and Analysis Methods, 03 medical and health sciences, Antimalarials, Model Organisms, Dose Prediction Methods, General & Internal Medicine, Parasite Groups, parasitic diseases, medicine, Gametocyte, Parasitic Diseases, Animals, Humans, Acrylamides, Dose-Response Relationship, Drug, Organisms, Biology and Life Sciences, Cell Biology, biology.organism_classification, Tropical Diseases, Parasitic Protozoans, Malaria, Germ Cells, Pharmacodynamics, Parasitology, Apicomplexa
وصف الملف: application/pdf
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المؤلفون: Marc Iglarz, Josiane Rein, Solange Meyer, Martine Clozel, Daniel Bur, Thomas Weller, Stephan Buchmann, Martin Bolli, Markus Rey, Christoph Binkert, Patrick Hess, Alexander Treiber, Walter Fischli, Christoph Boss
المصدر: Journal of Medicinal Chemistry. 55:7849-7861
مصطلحات موضوعية: Endothelin A Receptor Antagonists, Stereochemistry, Endothelin B Receptor Antagonists, Administration, Oral, CHO Cells, Pharmacology, chemistry.chemical_compound, Cricetulus, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Antihypertensive Agents, Sulfamide, Macitentan, Sulfonamides, Rats, Inbred Dahl, Endothelin receptor antagonist, Bosentan, Rats, Pyrimidines, chemistry, Molecular Medicine, Endothelin receptor, medicine.drug
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المؤلفون: Petros Papastogiannidis, Hamed Aissaoui, Olivier Corminboeuf, Ralf Brunner, Romain Siegrist, Sergio Wittlin, Bibia Heidmann, Richard W. D. Welford, Stephane Delahaye, Marcel Kaiser, Christoph Boss, Christoph Binkert, Jolanda Kamber, Reto Brun, Zbynek Bozdech, Till S. Voss, Christoph Fischli, Solange Meyer
المساهمون: School of Biological Sciences
المصدر: The Journal of infectious diseases
مصطلحات موضوعية: Artemisinins, Erythrocytes, Microarray, Plasmodium berghei, Biological Availability, Drug resistance, Pharmacology, Parasitemia, Piperazines, Cell Line, Antimalarials, Inhibitory Concentration 50, Mice, 03 medical and health sciences, Chloroquine, parasitic diseases, medicine, Animals, Immunology and Allergy, Antimalarial Agent, 030304 developmental biology, 0303 health sciences, biology, 030306 microbiology, Plasmodium falciparum, medicine.disease, biology.organism_classification, In vitro, Malaria, Rats, 3. Good health, Infectious Diseases, medicine.drug
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a757029cd53bed4e8ee4209460271056
http://www.jid.oxfordjournals.org/cgi/pmidlookup?view=long&pmid=22732921 -
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المؤلفون: Christoph Fäh, Solange Meyer, Leo A. Hardegger, Daniel Bur, Roland Mathys, François Diederich
المصدر: European Journal of Organic Chemistry. 2010:4617-4629
مصطلحات موضوعية: chemistry.chemical_classification, Ketone, biology, Stereochemistry, Organic Chemistry, Absolute configuration, Diastereomer, Plasmepsin, Active site, Chemical synthesis, Chiral resolution, Alicyclic compound, chemistry, biology.protein, Physical and Theoretical Chemistry
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المؤلفون: W. Bernd Schweizer, Leo A. Hardegger, Lukas Baitsch, François Diederich, Solange Meyer, Christoph Fäh, Daniel Bur
المصدر: ORGANIC & BIOMOLECULAR CHEMISTRY
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Peptidomimetic, Stereochemistry, Molecular Conformation, Protonation, Crystallography, X-Ray, Biochemistry, Alicyclic compound, Antimalarials, Plasmepsin II, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Physical and Theoretical Chemistry, chemistry.chemical_classification, Organic Chemistry, Water, Biological activity, Fluorine, Ketones, Ligand (biochemistry), Malaria, Enzyme, chemistry, Hydrate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ee0be6418f105599d5f992f1328b569b