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1
المؤلفون: Heather Finlay, Claudia Generaux, Carrie Xu, Chiuwa E. Luk, Ruth R. Wexler, Ji Jiang, James A. Johnson, Michael Galella, Jeffrey S. Bostwick, William A. Schumacher, Tao Wang, Monique Phillips, Soong-Hoon Kim, Yan He, Joelle M. Onorato, Peter S. Gargalovic, Xue-Qing Chen, David A. Gordon
المصدر: Journal of medicinal chemistry. 64(6)
مصطلحات موضوعية: Cardiac function curve, Agonist, Male, Models, Molecular, medicine.drug_class, Pyridones, Endogeny, Pharmacology, 01 natural sciences, Rats, Sprague-Dawley, 03 medical and health sciences, Dogs, Drug Discovery, medicine, Animals, Humans, Receptor, 030304 developmental biology, Apelin receptor, 0303 health sciences, Apelin Receptors, Chemistry, Haplorhini, medicine.disease, 0104 chemical sciences, Rats, 010404 medicinal & biomolecular chemistry, Heart failure, Molecular Medicine, Intercellular Signaling Peptides and Proteins
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2
المؤلفون: David S. Taylor, Lei Zhao, Leonard P. Adam, David A. Gordon, Michael Basso, Alice Ye Chen, Eddie C.-K. Liu, Ji Jiang, Christian Caporuscio, Zulan Pi, James A. Johnson, Soong-Hoon Kim, Heather Finlay, John Lloyd, Joelle M. Onorato, Gregory A. Locke, George O. Tora, Ruth R. Wexler, Todd Kirshgessner, Lynn M. Abell, Xiaohong Yin, Hao Lu, Richard Yang, Sarah C. Traeger, Monique Phillips, Kamelia Behnia, Carol S. Ryan
المصدر: Journal of medicinal chemistry. 63(4)
مصطلحات موضوعية: Endothelial lipase, Male, Oxadiazoles, Molecular Structure, Chemistry, Cholesterol, Transgene, Reverse cholesterol transport, Cholesterol, HDL, Lipase, Pharmacology, Ketones, Small molecule, Mice, Inbred C57BL, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Drug Discovery, Molecular Medicine, Animals, lipids (amino acids, peptides, and proteins), Efflux, Enzyme Inhibitors, Lipoprotein
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المؤلفون: Lynn M. Abell, Brandon Parkhurst, Lei Zhao, Richard Yang, David A. Gordon, Jennifer X. Qiao, Soong-Hoon Kim, Xue-Qing Chen, Joelle M. Onorato, David S. Taylor, Hao Lu, Michael Basso, Alice Ye Chen, Kamelia Behnia, Heather Finlay, Xiaohong Yin, Leonard P. Adam, Ji Jiang, Gregory A. Locke, George O. Tora, Zulan Pi, Monique Phillips, Christian Caporuscio, Ruth R. Wexler, Eddie C.-K. Liu, James A. Johnson
المصدر: Bioorganicmedicinal chemistry letters. 29(15)
مصطلحات موضوعية: Endothelial lipase, biology, 010405 organic chemistry, Cholesterol, Organic Chemistry, Clinical Biochemistry, Reverse cholesterol transport, Pharmaceutical Science, Pharmacology, 01 natural sciences, Biochemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, High-density lipoprotein, chemistry, Benzothiazole, Drug Discovery, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), Hepatic lipase, Lipase, Molecular Biology, IC50
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المؤلفون: Yufen Zhao, Ashvinikumar V. Gavai, Saulnier Mark G, Demartino Michael P, Claude A. Quesnelle, Brian E. Fink, Libing Chen, Patrice Gill, David B. Frennesson, Soong-Hoon Kim, Phil S. Baran
المصدر: Synlett. 27:2254-2258
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Succinic acid, Stereochemistry, Organic Chemistry, Intermolecular force, Diastereomer, Organic chemistry, 010402 general chemistry, 01 natural sciences, 0104 chemical sciences
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a1ab4c496ef40e73dd1968f7daf87048
https://doi.org/10.1055/s-0035-1561636 -
5
المؤلفون: Eddie C.-K. Liu, James A. Johnson, Lynn M. Abell, Leonard P. Adam, Xue-Qing Chen, Christian Caporuscio, Heather Finlay, Jennifer X. Qiao, Brandon Parkhurst, David S. Taylor, Monique Phillips, Soong-Hoon Kim, Ji Jiang, Joelle M. Onorato, Gregory A. Locke, David A. Gordon, Michael Basso, Alice Ye Chen, George O. Tora, Xiaohong Yin, Ruth R. Wexler, Zulan Pi, Richard Yang, Kamelia Behnia, Lei Zhao, Hao Lu
المصدر: Bioorganic & Medicinal Chemistry Letters. 29:2525
مصطلحات موضوعية: Endothelial lipase, chemistry.chemical_compound, Benzothiazole, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Identification (biology), Molecular Biology, Biochemistry
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6Synthesis, Chromatographic Purification, and Isolation of Epothilone–Folic Acid Conjugate BMS-753493
المؤلفون: Riccardo E. Frigerio, Soong-Hoon Kim, Xujin Lu, Wei Wang, Nuria de Mas, Bing-Shiou Yang, Kevin P. Girard, Olav Lyngberg, Zhenrong Guo, Victor W. Rosso, Zerene A. Manaloto, Gokhale Madhushree Yeshwant, Mark S. Bolgar, Luca Parlanti, Ajit B. Thakur, Germano D'arasmo, Konstantinos Dambalas, Guido Ströhlein
المصدر: Organic Process Research & Development. 15:797-809
مصطلحات موضوعية: Active ingredient, Chromatography, Aqueous solution, Chemistry, Precipitation (chemistry), Organic Chemistry, Epothilone, Decomposition, chemistry.chemical_compound, Adsorption, Zwitterion, medicine, Physical and Theoretical Chemistry, medicine.drug, Conjugate
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7
المؤلفون: Johnni Gullo-Brown, Michael A. Poss, Wayne Vaccaro, Tram N. Huynh, Stephanie Barbosa, Carolyn S. Ricca, Mark E. Salvati, Veeraswamy Manne, Zhong Chen, Kenneth J. Leavitt, Soong-Hoon Kim, David R. Tortolani, Donna D. Wei
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:628-632
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Acylation, Clinical Biochemistry, Substituent, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Pyrroles, Amines, Enzyme Inhibitors, skin and connective tissue diseases, Molecular Biology, Mitogen-Activated Protein Kinase Kinases, chemistry.chemical_classification, Aniline Compounds, biology, Chemistry, MEK inhibitor, fungi, Organic Chemistry, Aromatic amine, Rats, Pyridazines, body regions, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Amine gas treating
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المؤلفون: Bruce M. Rankin, William J. Pitts, William J. Metzler, Kenneth J. Leavitt, Andrew T. Pudzianowski, Wayne Vaccaro, Richard Liu, Patricia A. McDonnell, Joseph Barbosa, Soong-Hoon Kim
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1101-1106
مصطلحات موضوعية: Models, Molecular, Drug, Matrix metalloproteinase inhibitor, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, Matrix Metalloproteinase Inhibitors, Matrix metalloproteinase, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Matrix Metalloproteinase 13, Osteoarthritis, Drug Discovery, medicine, Humans, Structure–activity relationship, Computer Simulation, Spiro Compounds, Enzyme Inhibitors, Molecular Biology, media_common, chemistry.chemical_classification, biology, Organic Chemistry, General Medicine, In vitro, Kinetics, Enzyme, chemistry, Enzyme inhibitor, Drug Design, Barbiturates, biology.protein, Collagenase, Computer-Aided Design, Structure based, Molecular Medicine, medicine.drug
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المؤلفون: Craig R. Fairchild, Robert M. Borzilleri, James A. Johnson, Soong-Hoon Kim, Byron H. Long, Gregory D. Vite, Alicia Regueiro-Ren, Xiaoping Zheng, Francis Y. Lee
المصدر: Organic Letters. 3:2693-2696
مصطلحات موضوعية: Epothilones, Stereochemistry, Aziridines, Organic Chemistry, Epoxide, Antineoplastic Agents, Biological activity, Epothilone, Aziridine, Biochemistry, Tubulin binding, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, medicine, Epoxy Compounds, Structure–activity relationship, Moiety, Physical and Theoretical Chemistry, medicine.drug
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المؤلفون: Craig R. Fairchild, John D. Dimarco, Robert M. Borzilleri, Soong-Hoon Kim, Jack Z. Gougoutas, Francis Y. Lee, James A. Johnson, Gregory D. Vite, Robert J. Schmidt, and Byron H. Long, Xiaoping Zheng
المصدر: Journal of the American Chemical Society. 122:8890-8897
مصطلحات موضوعية: Epothilones, Total synthesis, General Chemistry, Epothilone, Biochemistry, Combinatorial chemistry, Semisynthesis, Catalysis, chemistry.chemical_compound, Colloid and Surface Chemistry, chemistry, Lactam, medicine, Nucleophilic substitution, Stereoselectivity, Azide, medicine.drug