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1دورية أكاديمية
المؤلفون: Gwladys Rivière, Saoussen Oueslati, Maud Gayral, Jean-Bernard Créchet, Naïma Nhiri, Eric Jacquet, Jean-Christophe Cintrat, François Giraud, Carine van Heijenoort, Ewen Lescop, Stéphanie Pethe, Bogdan I. Iorga, Thierry Naas, Eric Guittet, Nelly Morellet
المصدر: ACS Omega, Vol 5, Iss 18, Pp 10466-10480 (2020)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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2
المؤلفون: Charles Skarbek, Hichem Maslah, Marie-Aude Plamont, Stéphanie Pethe, Catherine Gourson, Thomas Le Saux, Ludovic Jullien, Raphaël Labruère
المصدر: Angewandte Chemie. 133:24245-24249
مصطلحات موضوعية: Phenanthridine, Molecular Structure, Chemistry, Cell Survival, Biological activity, Antineoplastic Agents, General Chemistry, Drug action, General Medicine, Prodrug, Combinatorial chemistry, Catalysis, KB Cells, Phenanthridines, chemistry.chemical_compound, Drug Development, Cyclization, Cancer cell, Cytotoxic T cell, Humans, Prodrugs, Bioorthogonal chemistry, Drug Screening Assays, Antitumor, Cytotoxicity, Cell Proliferation
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3
المؤلفون: Anaïs Espinosa, Estelle Rascol, Marta Abellán Flos, Charles Skarbek, Pascale Lieben, Eva Bannerman, Alba Diez Martinez, Stéphanie Pethe, Pierre Benoit, Sylvie Nélieu, Raphaël Labruère
المصدر: Chemosphere. 306:135616
مصطلحات موضوعية: Photolysis, Environmental Engineering, Drinking Water, Health, Toxicology and Mutagenesis, Public Health, Environmental and Occupational Health, General Medicine, General Chemistry, Wastewater, Pollution, Methotrexate, Pharmaceutical Preparations, Environmental Chemistry, Environmental Pollutants, Ecosystem, Water Pollutants, Chemical, Ethers
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4
المؤلفون: Raphaël Labruère, Hichem Maslah, Stéphanie Pethe
المصدر: Future medicinal chemistry. 13(10)
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Reactive oxygen species, 2019-20 coronavirus outbreak, Coronavirus disease 2019 (COVID-19), Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2), Antineoplastic Agents, Prodrug, Anticancer chemotherapy, Boronic Acids, Reactive Nitrogen Species, Cancer treatment, chemistry.chemical_compound, chemistry, Neoplasms, Drug Discovery, Tumor Microenvironment, Molecular Medicine, Humans, Prodrugs, Reactive Oxygen Species, Boronic acid
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5
المؤلفون: Raphaël Labruère, Philippe M. Loiseau, Stéphanie Pethe, Elodie Jagu, Sébastien Pomel, Alba Diez-Martinez, Estelle Rascol
المصدر: European Journal of Medicinal Chemistry. 150:655-666
مصطلحات موضوعية: 0301 basic medicine, Spermidine, Stereochemistry, Trypanosoma brucei gambiense, Antiprotozoal Agents, Leishmania donovani, 010402 general chemistry, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Parasitic Sensitivity Tests, parasitic diseases, Drug Discovery, Biological evaluation, Pharmacology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, biology, Organic Chemistry, General Medicine, biology.organism_classification, 0104 chemical sciences, 030104 developmental biology, Enzyme, chemistry, Trypanothione reductase, Polyamine
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6
المصدر: European Journal of Medicinal Chemistry. 139:982-1015
مصطلحات موضوعية: 0301 basic medicine, 030106 microbiology, Antiprotozoal Agents, Spermine, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Parasitic Sensitivity Tests, In vivo, Drug Discovery, Polyamines, Animals, Humans, Kinetoplastida, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, General Medicine, In vitro, Spermidine, 030104 developmental biology, Biochemistry, chemistry, Putrescine, Polyamine, Polyamine metabolism, Conjugate
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7
المؤلفون: Charles Skarbek, Thi Hang Au, Thi Thu Ha Vu, Stéphanie Pethe, Giang Vo-Thanh, Thi Phuong Hoa Nguyen, Raphaël Labruère, Jean-Pierre Baltaze
المصدر: Tetrahedron. 92:132248
مصطلحات موضوعية: chemistry.chemical_classification, Aqueous solution, Ketone, 010405 organic chemistry, Chemistry, Stereochemistry, Organic Chemistry, Biological activity, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Bioavailability, Cell culture, Yield (chemistry), Drug Discovery, Cancer cell, Michael reaction
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8
المؤلفون: Jean-Christophe Cintrat, Philippe M. Loiseau, Raphaël Labruère, Sébastien Pomel, Stéphanie Pethe, Elodie Jagu
المساهمون: Biomolécules : Conception, Isolement, Synthèse (BioCIS), Institut de Chimie du CNRS (INC)-Université Paris-Saclay-Centre National de la Recherche Scientifique (CNRS)-CY Cergy Paris Université (CY)
المصدر: Bioorganic & Medicinal Chemistry Letters
Bioorganic & Medicinal Chemistry Letters, 2019, 29, pp.1710-1713. ⟨10.1016/j.bmcl.2019.05.030⟩مصطلحات موضوعية: Clinical Biochemistry, Leishmania donovani, Pharmaceutical Science, Spermine, 01 natural sciences, Biochemistry, chemistry.chemical_compound, parasitic diseases, Drug Discovery, Polyamines, [CHIM]Chemical Sciences, Animals, Molecular Biology, IC50, Fluorescent Dyes, biology, Polyamine transport, 010405 organic chemistry, Organic Chemistry, Biological Transport, biology.organism_classification, Fluorescence, 3. Good health, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Molecular Medicine, Conjugate
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9
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10
المؤلفون: Charles Skarbek, Hichem Maslah, Raphaël Labruère, Stéphanie Pethe
المساهمون: Institut de Chimie Moléculaire et des Matériaux d'Orsay (ICMMO), Institut de Chimie du CNRS (INC)-Université Paris-Saclay-Centre National de la Recherche Scientifique (CNRS)
المصدر: European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 2020, 207, pp.112670-. ⟨10.1016/j.ejmech.2020.112670⟩مصطلحات موضوعية: Boron Compounds, Antineoplastic Agents, medicine.disease_cause, Anticancer chemotherapy, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Neoplasms, Drug Discovery, Boron containing, Tumor Microenvironment, medicine, Animals, Humans, [CHIM]Chemical Sciences, Prodrugs, 030304 developmental biology, Pharmacology, chemistry.chemical_classification, 0303 health sciences, Tumor microenvironment, Reactive oxygen species, 010405 organic chemistry, Chemistry, Organic Chemistry, General Medicine, Anticancer prodrugs, Prodrug, 0104 chemical sciences, Oxidative Stress, Cancer research, Reactive Oxygen Species, Oxidative stress, Boronic acid