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1
المؤلفون: Deepak Dalvie, Yong Wang, Theodore O. Johnson, Michael Siu, Cripps Stephan James, Klaus Ruprecht Dress, Jacqui Elizabeth Hoffman, Taylor Wendy Dianne, Stanley William Kupchinsky, Ping Kang, Sue Zhou, Jacques Ermolieff, Andrea Fanjul, Sajiv Krishnan Nair, Arturo Castro, Jennifer E. Vogel, Jean Joo Matthews, Amy LaPaglia, Cheng Hengmiao, Paul A. Rejto, Christopher Ronald Smith, Martin Paul Edwards, Natilie Hosea
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2344-2348
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Aminopyridines, Pharmaceutical Science, Dehydrogenase, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, 11β-hydroxysteroid dehydrogenase type 1, 11-beta-Hydroxysteroid Dehydrogenase Type 1, Drug Discovery, Humans, Structure–activity relationship, Molecular Biology, Sulfonamides, biology, Chemistry, Organic Chemistry, HEK 293 cells, Glutathione, HEK293 Cells, Reactive metabolite, Risk-benefit analysis, biology.protein, Molecular Medicine
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2
المؤلفون: Skalitzky Donald James, Karen A. Maegley, Stanley William Kupchinsky, Pei Pei Kung, Anne Ekker, Laura Anne Bloom, Leslie A. Kuhn, Peter W. Rose, Jerry J. Meng, Zehnder Luke Raymond, M. Catherine Johnson
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:2829-2833
مصطلحات موضوعية: chemistry.chemical_classification, 5'-deoxy-5'-methylthioadenosine phosphorylase, Molecular Structure, biology, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Substrate (chemistry), Biochemistry, Chemical synthesis, In vitro, Substrate Specificity, Enzyme, Purine-Nucleoside Phosphorylase, chemistry, Design synthesis, Drug Design, Drug Discovery, Glycosyltransferase, biology.protein, Humans, Molecular Medicine, Molecular Biology, Biological evaluation
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3
المؤلفون: Kristin Kelly, Christopher John Helal, Tate Bonnie Frances, Mavis Diane Adam, Zhijun Kang, Marcia F. Peterson, Thomas G. Gant, Christopher B. Cooper, Michael K. Ahlijanian, Stanley William Kupchinsky, John C. Lucas, Frank S. Menniti, Sanner Mark Allen
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:5521-5525
مصطلحات موضوعية: Cyclin E, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Nerve Tissue Proteins, Isobutyramide, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Aminothiazole, Alzheimer Disease, Drug Discovery, CDC2-CDC28 Kinases, Protein kinase A, Molecular Biology, Molecular Structure, biology, Kinase, Cyclin-dependent kinase 5, Cyclin-Dependent Kinase 2, Organic Chemistry, Cyclin-dependent kinase 2, Cyclin-Dependent Kinase 5, Amides, Cyclin-Dependent Kinases, Thiazoles, nervous system, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine