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1دورية أكاديمية
المؤلفون: Valentin Wydra, Stefan Gerstenecker, Dieter Schollmeyer, Stanislav Andreev, Teodor Dimitrov, Ricardo Augusto Massarico Serafim, Stefan Laufer, Matthias Gehringer
المصدر: Molbank, Vol 2021, Iss 1, p M1181 (2021)
مصطلحات موضوعية: 3-nitropyridines, nucleophilic aromatic substitution, Buchwald–Hartwig arylamination, protein kinase inhibitors, covalent inhibitors, Inorganic chemistry, QD146-197
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Stefan Gerstenecker, Lisa Haarer, Martin Schröder, Mark Kudolo, Martin P. Schwalm, Valentin Wydra, Ricardo A. M. Serafim, Apirat Chaikuad, Stefan Knapp, Stefan Laufer, Matthias Gehringer
المصدر: Cancers, Vol 13, Iss 20, p 5133 (2021)
مصطلحات موضوعية: protein kinases, chemical probes, S6K2, p70S6K2, p70S6Kb, RPS6KB2, Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Michael Forster, Xiaojun Julia Liang, Martin Schröder, Stefan Gerstenecker, Apirat Chaikuad, Stefan Knapp, Stefan Laufer, Matthias Gehringer
المصدر: International Journal of Molecular Sciences, Vol 21, Iss 23, p 9269 (2020)
مصطلحات موضوعية: tyrosine kinases, bone marrow tyrosine kinase on chromosome X, Bruton’s tyrosine kinase, Janus kinase 3, covalent inhibitors, chemical probes, Biology (General), QH301-705.5, Chemistry, QD1-999
وصف الملف: electronic resource
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4
المؤلفون: Ricardo A. M. Serafim, André da Silva Santiago, Martin P. Schwalm, Zexi Hu, Caio V. dos Reis, Jessica E. Takarada, Priscila Mezzomo, Katlin B. Massirer, Mark Kudolo, Stefan Gerstenecker, Apirat Chaikuad, Lars Zender, Stefan Knapp, Stefan Laufer, Rafael M. Couñago, Matthias Gehringer
المصدر: Journal of Medicinal Chemistry. 65:3173-3192
مصطلحات موضوعية: Male, Models, Molecular, Antineoplastic Agents, Cell Cycle Proteins, Triple Negative Breast Neoplasms, In Vitro Techniques, Protein Serine-Threonine Kinases, Protein-Tyrosine Kinases, Crystallography, X-Ray, Mass Spectrometry, Mice, Cell Line, Tumor, Drug Design, Drug Discovery, Microsomes, Liver, Animals, Humans, Molecular Medicine, Female, Drug Screening Assays, Antitumor, Protein Kinase Inhibitors
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5
المؤلفون: Katlin B. Massirer, Priscila Mezzomo, Mark Kudolo, A.S. Santiago, Apirat Chaikuad, Caio V. dos Reis, Matthias Gehringer, Rafael M. Couñago, Jessica Takarada, Ricardo A. M. Serafim, Stefan Knapp, Martin P. Schwalm, Stefan Laufer, Stefan Gerstenecker
مصطلحات موضوعية: Chromosome segregation, Spindle checkpoint, Chemistry, Covalent bond, Kinase, Context (language use), Mitosis, Monopolar spindle, Cysteine, Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b037609509dc018037dcddecb4ee07df
https://doi.org/10.26434/chemrxiv.14601264 -
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المؤلفون: Ricardo A. M. Serafim, Matthias Gehringer, Stanislav Andreev, Teodor Dimitrov, Stefan Gerstenecker, Valentin Wydra, Dieter Schollmeyer, Stefan Laufer
المصدر: Molbank, Vol 2021, Iss M1181, p M1181 (2021)
مصطلحات موضوعية: Imine, nucleophilic aromatic substitution, Infrared spectroscopy, 01 natural sciences, Biochemistry, Medicinal chemistry, 03 medical and health sciences, chemistry.chemical_compound, Buchwald–Hartwig arylamination, Nucleophilic aromatic substitution, Benzophenone, lcsh:Inorganic chemistry, Physical and Theoretical Chemistry, 030304 developmental biology, 0303 health sciences, 010405 organic chemistry, Chemistry, Organic Chemistry, Regioselectivity, Nuclear magnetic resonance spectroscopy, lcsh:QD146-197, 0104 chemical sciences, 3-nitropyridines, protein kinase inhibitors, covalent inhibitors, Amine gas treating, Two-dimensional nuclear magnetic resonance spectroscopy
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7
المؤلفون: Chelsey Collins-Kautz, Gerhard Klebe, Stefan Gerstenecker, Björn Wagner, Andreas Heine, K. Ngo
المصدر: Journal of medicinal chemistry. 63(6)
مصطلحات موضوعية: Proteases, Pyridines, Protonation, Calorimetry, Crystallography, X-Ray, Ligands, 01 natural sciences, Antithrombins, Serine, 03 medical and health sciences, Thrombin, Drug Discovery, medicine, Animals, Humans, Trypsin, 030304 developmental biology, 0303 health sciences, Binding Sites, Chemistry, Substrate (chemistry), Water, Dipeptides, Ligand (biochemistry), 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Biochemistry, Molecular Medicine, Thermodynamics, Cattle, Protons, Selectivity, Trypsin Inhibitors, circulatory and respiratory physiology, medicine.drug, Protein Binding