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1دورية أكاديمية
المؤلفون: Stefanie Kickinger, Maria E. K. Lie, Akihiro Suemasa, Anas Al-Khawaja, Koichi Fujiwara, Mizuki Watanabe, Kristine S. Wilhelmsen, Christina B. Falk-Petersen, Bente Frølund, Satoshi Shuto, Gerhard F. Ecker, Petrine Wellendorph
المصدر: Frontiers in Chemistry, Vol 9 (2021)
مصطلحات موضوعية: SLC6 neurotransmitter transporters, competitive inhibition, binding mode analysis, computational chemistry, bicyclo-GABA, BGT1, Chemistry, QD1-999
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Vojtech Dvorak, Tabea Wiedmer, Alvaro Ingles-Prieto, Patrick Altermatt, Helena Batoulis, Felix Bärenz, Eckhard Bender, Daniela Digles, Franz Dürrenberger, Laura H. Heitman, Adriaan P. IJzerman, Douglas B. Kell, Stefanie Kickinger, Daniel Körzö, Philipp Leippe, Thomas Licher, Vania Manolova, Riccardo Rizzetto, Francesca Sassone, Lia Scarabottolo, Avner Schlessinger, Vanessa Schneider, Hubert J. Sijben, Anna-Lena Steck, Hanna Sundström, Sara Tremolada, Maria Wilhelm, Marina Wright Muelas, Diana Zindel, Claire M. Steppan, Giulio Superti-Furga
المصدر: Frontiers in Pharmacology, Vol 12 (2021)
مصطلحات موضوعية: solute carrier, cell-based assay, drug discovery, chemical screening, transporters, SLC, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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المؤلفون: Mette H. Poulsen, Feng Xue, Svetlana R. Maurya, Stefanie Kickinger, Samuel Usher, Petrine Wellendorph, Alicia Lundby, Stephan A. Pless
المصدر: Biophysical Journal. 122:249a
مصطلحات موضوعية: Biophysics
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المؤلفون: Stefanie Kickinger, Jennifer Hemmerich, Gerhard F. Ecker, Stefan Kubicek, Bettina Gürtl, Charles-Hugues Lardeau, Adrián César-Razquin, Giulio Superti-Furga, Richard Kumaran Kandasamy, Kristaps Klavins, Vitaly Sedlyarov, Alvaro Ingles-Prieto, Giuseppe Fiume, Sabrina Lindinger, Felix Kartnig, Konstantinos Papakostas, Anna Koren, Enrico Girardi, Justyna Konecka
المصدر: Nature chemical biology
Nature Chemical Biologyمصطلحات موضوعية: Cisplatin, 0303 health sciences, Chemistry, 030302 biochemistry & molecular biology, Transporter, Cell Biology, Chemical space, Transmembrane protein, Article, 3. Good health, 03 medical and health sciences, Biochemistry, medicine, Cytotoxic T cell, Artemisinin, Molecular Biology, Gene, 030304 developmental biology, Genetic screen, medicine.drug
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المؤلفون: Alvaro Ingles-Prieto, Douglas B. Kell, Laura H. Heitman, Daniela Digles, Stefanie Kickinger, Patrick Altermatt, Diana Zindel, Adriaan P. IJzerman, Vanessa Schneider, Daniel Körzö, Maria Wilhelm, Tabea Wiedmer, Helena Batoulis, Sara Tremolada, Giulio Superti-Furga, Anna Lena Steck, Marina Wright Muelas, Thomas Licher, Eckhard Bender, Vojtech Dvorak, Hubert J. Sijben, Avner Schlessinger, Franz Dürrenberger, Francesca Sassone, Vania Manolova, Riccardo Rizzetto, Philipp Leippe, Lia Scarabottolo, Felix Bärenz, Hanna Sundström, Claire M. Steppan
المصدر: Frontiers in Pharmacology
Dvorak, V, Wiedmer, T, Ingles-Prieto, A, Altermatt, P, Batoulis, H, Bärenz, F, Bender, E, Digles, D, Dürrenberger, F, Heitman, L H, IJzerman, A P, Kell, D B, Kickinger, S, Körzö, D, Leippe, P, Licher, T, Manolova, V, Rizzetto, R, Sassone, F, Scarabottolo, L, Schlessinger, A, Schneider, V, Sijben, H J, Steck, A L, Sundström, H, Tremolada, S, Wilhelm, M, Wright Muelas, M, Zindel, D, Steppan, C M & Superti-Furga, G 2021, ' An Overview of Cell-Based Assay Platforms for the Solute Carrier Family of Transporters ', Frontiers in Pharmacology, vol. 12, 722889 . https://doi.org/10.3389/fphar.2021.722889
Frontiers in Pharmacology, 12, 722889
Frontiers in pharmacology
Frontiers in Pharmacology, Vol 12 (2021)مصطلحات موضوعية: chemical screening, solute carrier, SLC, Druggability, cell-based assay, RM1-950, Computational biology, Review, transporters, Biology, drug discovery, 03 medical and health sciences, 0302 clinical medicine, Pharmacology (medical), 030304 developmental biology, Pharmacology, 0303 health sciences, Drug discovery, Chemical screening, Cellular Assay, Transporter, SUPERFAMILY, Solute carrier, 3. Good health, Solute carrier family, Transporters, Cell-based assay, Therapeutics. Pharmacology, 030217 neurology & neurosurgery, Cell based
وصف الملف: application/pdf; application/zip
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8c538438b273fae113d94d4db91b031c
https://phaidra.univie.ac.at/o:1603733 -
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المؤلفون: Arne Schousboe, Rasmus P. Clausen, Stefanie Kickinger, Jonas Skovgaard-Petersen, Maria E. K. Lie, Gerhard F. Ecker, Petrine Wellendorph, H. Steve White
المصدر: Lie, M E K, Kickinger, S, Skovgaard-Petersen, J, Ecker, G F, Clausen, R P, Schousboe, A, White, H S & Wellendorph, P 2020, ' Pharmacological Characterization of a Betaine/GABA Transporter 1 (BGT1) Inhibitor Displaying an Unusual Biphasic Inhibition Profile and Anti-seizure Effects ', Neurochemical Research, vol. 45, pp. 1551–1565 . https://doi.org/10.1007/s11064-020-03017-y
Neurochemical Researchمصطلحات موضوعية: 0301 basic medicine, Male, GABA Plasma Membrane Transport Proteins, Tiagabine, Mice, Transgenic, GABA uptake, CHO Cells, Pharmacology, Biochemistry, Epilepsy, Reflex, Protein Structure, Secondary, GABA transporter 1, 03 medical and health sciences, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Mice, 0302 clinical medicine, Betaine, Cricetulus, Seizures, medicine, GABA transporter, Animals, Humans, Q299L, Binding site, Original Paper, Epilepsy, biology, General Medicine, Cyclohexanecarboxylic acid, 030104 developmental biology, HEK293 Cells, Treatment Outcome, chemistry, Acoustic Stimulation, GAT1, Docking (molecular), Cell culture, biology.protein, Anticonvulsants, Homology modelling, 030217 neurology & neurosurgery, medicine.drug, Protein Binding
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3be1e5b0f009359dee573c6df3162134
https://curis.ku.dk/portal/da/publications/pharmacological-characterization-of-a-betainegaba-transporter-1-bgt1-inhibitor-displaying-an-unusual-biphasic-inhibition-profile-and-antiseizure-effects(f58627b3-6c59-4d36-ad00-48d86bf6a034).html -
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المؤلفون: Anas Al-Khawaja, Stine B. Vogensen, Hans Bräuner-Osborne, Jonas Skovgaard-Petersen, Rasmus P. Clausen, Stefanie Kickinger, Petrine Wellendorph, Arne Schousboe, Rebekka Löffler, Karsten K. Madsen, Gerhard F. Ecker, Emil Rosenthal, Lars N. Jorgensen, Nrupa Borkar
المصدر: Journal of Medicinal Chemistry. 60:8834-8846
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, GABA Plasma Membrane Transport Proteins, Stereochemistry, Allosteric regulation, GABA transporter 1, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Betaine, Piperidines, Drug Discovery, Radioligand, Humans, Structure–activity relationship, Homology modeling, Binding site, Serotonin Plasma Membrane Transport Proteins, biology, Chimera, Chemistry, 030104 developmental biology, Biochemistry, Docking (molecular), Benzamides, biology.protein, Molecular Medicine, GABA Uptake Inhibitors, Carrier Proteins, Allosteric Site
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المؤلفون: Charles-Hugues Lardeau, Stefanie Kickinger, Giulio Superti-Furga, Justyna Konecka, Giuseppe Fiume, Gerhard F. Ecker, Felix Kartnig, Anna Ringler, Sabrina Lindinger, Konstantinos Papakostas, Richard Kumaran Kandasamy, Enrico Girardi, Adrián César-Razquin, Alvaro Ingles-Prieto, Jennifer Hemmerich, Stefan Kubicek
مصطلحات موضوعية: Drug, 0303 health sciences, Cas9, media_common.quotation_subject, Cell, Transporter, Biology, Transmembrane protein, 3. Good health, 03 medical and health sciences, 0302 clinical medicine, medicine.anatomical_structure, Biochemistry, 030220 oncology & carcinogenesis, medicine, CRISPR, Cytotoxic T cell, 030304 developmental biology, media_common, Genetic screen
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9be34aa8b3f8d867e33780030c389a9d
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المؤلفون: Stefanie Kickinger, Maria Damgaard, Anas Al-Khawaja, Rebekka Löffler, Gerhard F. Ecker, Maria E. K. Lie, Bente Frølund, Petrine Wellendorph, Anne S. Haugaard, Francesco Bavo
المصدر: Biophysical Journal. 118:130a
مصطلحات موضوعية: biology, Biochemistry, Chemistry, Biophysics, biology.protein, Subtype selectivity, GABA transporter
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المؤلفون: Bente Frølund, Stefanie Kickinger, Petrine Wellendorph, Eva Hellsberg, Arne Schousboe, Gerhard F. Ecker
المصدر: Neuropharmacology. 161:107644
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Neurotransmitter transporter, GABA Plasma Membrane Transport Proteins, Synaptic cleft, Brain, Transporter, Biology, medicine.disease, Solute carrier family, GABA transporter 1, 03 medical and health sciences, Cellular and Molecular Neuroscience, Epilepsy, 030104 developmental biology, 0302 clinical medicine, medicine, biology.protein, Animals, Humans, GABAergic, GABA transporter, Neuroscience, 030217 neurology & neurosurgery