-
1
المؤلفون: Stephen Hindley, Paul M. O'Neill, Eghbaleh Asadollahy, Karen Rimmer, Alison E. Shone, Gemma L. Nixon, James L. Maggs, Stephen A. Ward, Richard A. Brigandi, Martin Bates, Patrick G. Bray, P. A. Winstanley, Paul A. Stocks, Jill Davies, Silvia Parapini, Livia Vivas, Domingo Gargallo, Stephanie L. Gresham, Hollie Lander, Giancarlo A. Biagini, B. Kevin Park, Donatella Taramelli, Ramesh Bambal, Federico M. Gomez-de-las-Heras, Charles B. Davis, Charlotte Hall, Neil G. Berry, Phil Roberts, Deborah Stanford
المصدر: Journal of Medicinal Chemistry. 52:1828-1844
مصطلحات موضوعية: Male, Cell Survival, Plasmodium berghei, Stereochemistry, Plasmodium falciparum, Drug Resistance, Amodiaquine, In Vitro Techniques, Chemical synthesis, Antimalarials, Mice, Structure-Activity Relationship, Dogs, Parasitic Sensitivity Tests, In vivo, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Rats, Wistar, ADME, Chemistry, Chloroquine, Biological activity, Haplorhini, Plasmodium yoelii, In vitro, Malaria, Rats, Bioavailability, Aminoquinolines, Hepatocytes, Molecular Medicine, Female, medicine.drug
-
2
المؤلفون: Stephanie L. Gresham, P. Roberts, Federico M. Gomez-de-las-Heras, Charles B. Davis, Timothy K. Hart, Ron M. Lawrence, Neil G. Berry, Paul M. O'Neill, Domingo Gargallo, B. Kevin Park, Stephen Hindley, Patrick G. Bray, Giancarlo A. Biagini, James L. Maggs, Amira Mukhtar, Peter Gibbons, P. A. Winstanley, Richard A. Brigandi, Paul A. Stocks, Alison E. Shone, Ramesh Bambal, Martin Bates, Richard P. Bonar-Law, Stephen A. Ward
المصدر: Journal of Medicinal Chemistry. 52:1408-1415
مصطلحات موضوعية: Models, Molecular, Benzylamines, Plasmodium berghei, Plasmodium falciparum, Industry standard, Drug Evaluation, Preclinical, Drug Resistance, Heme, Amodiaquine, Pharmacology, Antimalarials, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Chloroquine, Drug Discovery, medicine, Animals, Cytochrome P-450 Enzyme Inhibitors, Humans, Tert butyl, biology, Safety pharmacology, Haplorhini, Plasmodium yoelii, biology.organism_classification, Malaria, Rats, chemistry, 4-Aminoquinoline, Aminoquinolines, Molecular Medicine, Female, medicine.drug
-
3
المؤلفون: B. Kevin Park, Paul M. O'Neill, Dauda S. Kapu, Stephen Hindley, Paul A. Stocks, Jill Davies, Matthew D. Pugh, Patrick G. Bray, Stephen A. Ward
المصدر: Tetrahedron Letters. 44:8135-8138
مصطلحات موضوعية: chemistry.chemical_classification, Total harmonic distortion, Ketone, Chemistry, Organic Chemistry, Enantioselective synthesis, chemistry.chemical_element, General Medicine, Medicinal chemistry, Biochemistry, Catalysis, Cyclic Alkenes, Yield (chemistry), Drug Discovery, Organic chemistry, Cobalt
-
4
المؤلفون: Paul M. O'Neill, Jill Davies, Stephen A. Ward, Stephen Hindley, B. Kevin Park, Natalie L. Searle, Richard C. Storr, Patrick G. Bray
المصدر: Journal of Medicinal Chemistry. 45:1052-1063
مصطلحات موضوعية: Male, Tertiary amine, Plasmodium berghei, Stereochemistry, medicine.medical_treatment, Plasmodium falciparum, Dihydroartemisinin, Heterocyclic Compounds, 4 or More Rings, Chemical synthesis, Piperazines, Antimalarials, Mice, chemistry.chemical_compound, Drug Discovery, Food vacuole, medicine, Animals, Artemether, Artemisinin, biology, Chemistry, biology.organism_classification, Artemisinins, Malaria, Artesunate, Molecular Medicine, Sesquiterpenes, medicine.drug
-
5
المؤلفون: J. L. Maggs, Andrew V. Stachulski, Stephen A. Ward, Paul M. O'Neill, Feodor Scheinmann, Stephen Hindley, Stanley M. Roberts, Laurence P. D. Bishop, and Gary H. Posner, Alison Miller, B. Kevin Park
المصدر: Journal of Medicinal Chemistry. 44:58-68
مصطلحات موضوعية: Male, Free Radicals, Plasmodium berghei, Stereochemistry, medicine.medical_treatment, Plasmodium falciparum, Dihydroartemisinin, Crystallography, X-Ray, Antimalarials, Mice, Structure-Activity Relationship, In vivo, parasitic diseases, Drug Discovery, medicine, Animals, Bile, Ferrous Compounds, Artemether, Rats, Wistar, Artemisinin, Chemical decomposition, biology, Chemistry, Phenyl Ethers, Electron Spin Resonance Spectroscopy, Stereoisomerism, Plasmodium yoelii, biology.organism_classification, Combinatorial chemistry, Artemisinins, In vitro, Malaria, Rats, Molecular Medicine, Stereoselectivity, Sesquiterpenes, medicine.drug
-
6
المؤلفون: Patrick G. Bray, Paul M. O'Neill, Stephen Hindley, Ruth H Hughes, James L. Maggs, Jamie F. Bickley, Stephen A. Ward, P. A. Winstanley, Paul A. Stocks, Richard C. Storr, Amira Mukhtar, Ian A. O'Neil, Laura E. Randle, B. Kevin Park
المصدر: Journal of medicinal chemistry. 46(23)
مصطلحات موضوعية: Male, Stereochemistry, Metabolite, Plasmodium falciparum, Glucuronidation, Amodiaquine, Crystallography, X-Ray, chemistry.chemical_compound, Antimalarials, Structure-Activity Relationship, Chloroquine, In vivo, Drug Discovery, medicine, Animals, Rats, Wistar, biology, Chemistry, Biological activity, Plasmodium yoelii, biology.organism_classification, Malaria, Rats, 4-Aminoquinoline, Aminoquinolines, Molecular Medicine, medicine.drug
-
7دورية أكاديمية
المؤلفون: Paul M. O’Neill, Alison E. Shone, Deborah Stanford, Gemma Nixon, Eghbaleh Asadollahy, B. Kevin Park, James L. Maggs, Phil Roberts, Paul A. Stocks, Giancarlo Biagini, Patrick G. Bray, Jill Davies, Neil Berry, Charlotte Hall, Karen Rimmer, Peter A. Winstanley, Stephen Hindley, Ramesh B. Bambal, Charles B. Davis, Martin Bates
المصدر: Journal of Medicinal Chemistry; Apr2009, Vol. 52 Issue 7, p1828-1844, 17p
-
8دورية أكاديمية
المؤلفون: Paul M. OâNeill, B. Kevin Park, Alison E. Shone, James L. Maggs, Phillip Roberts, Paul A. Stocks, Giancarlo A. Biagini, Patrick G. Bray, Peter Gibbons, Neil Berry, Peter A. Winstanley, Amira Mukhtar, Richard Bonar-Law, Stephen Hindley, Ramesh B. Bambal, Charles B. Davis, Martin Bates, Timothy K. Hart, Stephanie L. Gresham, Ron M. Lawrence
المصدر: Journal of Medicinal Chemistry; Mar2009, Vol. 52 Issue 5, p1408-1415, 8p