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1
المؤلفون: Jennifer E, Davoren, Michelle, Garnsey, Betty, Pettersen, Michael A, Brodney, Jeremy R, Edgerton, Jean-Philippe, Fortin, Sarah, Grimwood, Anthony R, Harris, Stephen, Jenkinson, Terry, Kenakin, John T, Lazzaro, Che-Wah, Lee, Susan M, Lotarski, Lisa, Nottebaum, Steven V, O'Neil, Michael, Popiolek, Simeon, Ramsey, Stefanus J, Steyn, Catherine A, Thorn, Lei, Zhang, Damien, Webb
المصدر: Journal of medicinal chemistry. 60(15)
مصطلحات موضوعية: Diarrhea, Male, Lactams, Vomiting, Scopolamine, Isoindoles, Structure-Activity Relationship, Dogs, Allosteric Regulation, Piperidines, Seizures, Thiadiazoles, Animals, Humans, Donepezil, Rats, Wistar, Oxazoles, Sulfonamides, Receptor, Muscarinic M1, Mice, Inbred C57BL, Amphetamine, Drug Design, Indans, Microsomes, Liver, Ataxia, Female
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2
المؤلفون: Steven V. O’Neil, Biswanath De, Christopher D. Ellis, Charles A. Cruze, Mark William Baize, Thomas P. Demuth, Laufersweiler Michael Christopher, Maria Buchalova, Wei Lu, Richard L. Wang, Marina Belkin, Amy N. Fancher, Maureen K. Suchanek, John August Wos, David Lindsey Soper, William P. Schwecke, Kofi A. Oppong, Yili Wang
المصدر: Bioorganic & Medicinal Chemistry. 15:1311-1322
مصطلحات موضوعية: Male, Models, Molecular, Peptidomimetic, Stereochemistry, Interleukin-1beta, Clinical Biochemistry, Molecular Conformation, Biological Availability, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Structure-Activity Relationship, Viral Proteins, chemistry.chemical_compound, Drug Discovery, Animals, Caprolactam, Enzyme Inhibitors, Molecular Biology, Serpins, chemistry.chemical_classification, Dipeptide, Molecular Structure, biology, Organic Chemistry, Active site, Hydrogen Bonding, Caspase Inhibitors, Enzyme assay, Rats, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
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3
المؤلفون: Thomas P. Demuth, Maria E. Petrey, Maria Kontoyianni, Laufersweiler Michael Christopher, Matthew Pokross, Yili Wang, R.L. Walter, Jeffrey Tupper Roesgen, Eloise C. Richardson, Artem G. Evdokimov, Marlene Mekel, Georgios Sabatakos, Corey R. Hopkins, Steven V. O’Neil
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:5659-5663
مصطلحات موضوعية: Indoles, Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Peroxisome proliferator-activated receptor, Biochemistry, Chemical synthesis, Mice, chemistry.chemical_compound, Drug Discovery, Animals, Receptor, Imide, Molecular Biology, chemistry.chemical_classification, Indole test, Sulfonyl, Bicyclic molecule, Chemistry, Organic Chemistry, 3T3 Cells, Amides, PPAR gamma, Drug Design, Osteoporosis, Molecular Medicine
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4
المؤلفون: David Lindsey Soper, John August Wos, Kofi A. Oppong, Richard L. Wang, Biswanath De, Laufersweiler Michael Christopher, Thomas P. Demuth, Wei Lu, Steven V. O’Neil, Maureen K. Suchanek, Christopher D. Ellis, Amy N. Fancher, Yili Wang
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4728-4732
مصطلحات موضوعية: Models, Molecular, Thiazepines, Peptidomimetic, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Thiazepine, Enzyme Inhibitors, Molecular Biology, IC50, chemistry.chemical_classification, Molecular Structure, biology, Caspase 1, Organic Chemistry, Caspase Inhibitors, In vitro, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
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5
المؤلفون: Amy N. Fancher, Mark William Baize, Thomas P. Demuth, Kofi A. Oppong, Yili Wang, David Lindsey Soper, Steven V. O’Neil, Richard L. Wang, Wei Lu, Christopher D. Ellis, Maureen K. Suchanek, John August Wos, Gregory K. Bosch, Laufersweiler Michael Christopher, Biswanath De
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:5434-5438
مصطلحات موضوعية: Models, Molecular, Peptidomimetic, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Ring (chemistry), Metathesis, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Biomimetics, Drug Discovery, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Dipeptide, Bicyclic molecule, Chemistry, Organic Chemistry, Bridged Bicyclo Compounds, Heterocyclic, Caspase Inhibitors, Lactam, Molecular Medicine, Indicators and Reagents, Lactone
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6
المؤلفون: Mark William Baize, Thomas P. Demuth, Yili Wang, Steven V. O’Neil, Maureen K. Suchanek, John August Wos, David Lindsey Soper, Wei Lu, Laufersweiler Michael Christopher, Kofi A. Oppong, Christopher D. Ellis, Amy N. Fancher, Richard L. Wang
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:4322-4326
مصطلحات موضوعية: Peptidomimetic, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Pyrimidinones, Biochemistry, Chemical synthesis, Monocytes, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Immunologic Factors, Pyrroles, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Dipeptide, biology, Molecular Mimicry, Organic Chemistry, Dipeptides, Caspase Inhibitors, Enzyme binding, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Heterocyclic Compounds, 3-Ring, Tricyclic
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7
المصدر: Collection of Czechoslovak Chemical Communications. 65:490-510
مصطلحات موضوعية: Claisen rearrangement, Birch reduction, Stereochemistry, Chemistry, Dihydroxylation, Enantioselective synthesis, Iodolactonization, Regioselectivity, Total synthesis, General Chemistry, Stereocenter
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::42378c1b9ae6eeb2e50621ba5f930172
https://doi.org/10.1135/cccc20000490 -
8
المؤلفون: David G. Young, Qingbei Zeng, Steven V. O'Neil, Nathalie Guillo, Leo A. Paquette
المصدر: Synlett. 1999:1857-1866
مصطلحات موضوعية: Deprotonation, Aldol reaction, Chemistry, Organic Chemistry, Alkoxy group, Regioselectivity, Medicinal chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a68f9547bc2460562a447a1ebdfb5b32
https://doi.org/10.1055/s-1999-2959 -
9
المؤلفون: Steven V. O'Neil, Barry B. Snider, Nha Huu Vo
المصدر: The Journal of Organic Chemistry. 63:4732-4740
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Erinacine, Organic chemistry, Allocyathin B2
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10
المؤلفون: Steven V. O'Neil, Barry B. Snider
المصدر: Tetrahedron. 51:12983-12994
مصطلحات موضوعية: Formal synthesis, Chemistry, Organic Chemistry, Drug Discovery, Organic chemistry, Oxidative phosphorylation, Biochemistry, Radical cyclization