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1
المؤلفون: David E. Gloriam, Rebekka Löffler, Frederik Rostrup, Petrine Wellendorph, Bente Frølund, Christina Birkedahl Falk-Petersen, Kasper Harpsøe, Stine Buchleithner
المصدر: Molecular Pharmacology. 100:46-56
مصطلحات موضوعية: Pharmacology, Diazepam binding, GABAA receptor, Chemistry, Docking (molecular), Stereochemistry, Allosteric regulation, Functional selectivity, Molecular Medicine, Ligand-gated ion channel, Binding site, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b61e1339ce2ac4e170729ea407919188
https://doi.org/10.1124/molpharm.121.000266 -
2
المؤلفون: Tanja Schirmeister, David E. Gloriam, Stine Buchleithner, Christina Birkedahl Falk-Petersen, Sascha Jung, Frederik Rostrup, Petrine Wellendorph, Kasper Harpso E, Irene Conforti, Bente Fro Lund
المصدر: Journal of Medicinal Chemistry. 64:4730-4743
مصطلحات موضوعية: Imidazopyridine, Allosteric modulator, Pyridines, Stereochemistry, Allosteric regulation, Ligands, 01 natural sciences, Aminobutyric acid, Structure-Activity Relationship, 03 medical and health sciences, Allosteric Regulation, Drug Discovery, Humans, Potency, Receptor, 030304 developmental biology, Membrane potential, 0303 health sciences, Binding Sites, Chemistry, Receptors, GABA-A, 0104 chemical sciences, Molecular Docking Simulation, Protein Subunits, 010404 medicinal & biomolecular chemistry, HEK293 Cells, Drug Design, Molecular Medicine, Plate reader
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3
المؤلفون: Christina B, Falk-Petersen, Frederik, Rostrup, Rebekka, Löffler, Stine, Buchleithner, Kasper, Harpsøe, David E, Gloriam, Bente, Frølund, Petrine, Wellendorph
المصدر: Molecular pharmacology. 100(1)
مصطلحات موضوعية: Models, Molecular, Binding Sites, Diazepam, Imidazoles, Molecular Conformation, Receptors, GABA-A, Molecular Docking Simulation, HEK293 Cells, Allosteric Regulation, Protein Domains, Multiprotein Complexes, Benzamides, Mutagenesis, Site-Directed, Humans, Etomidate, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::c837e23849f8f58d6be669f190f31e85
https://pubmed.ncbi.nlm.nih.gov/33990405 -
4
المؤلفون: Kasper Harpsøe, Christina Birkedahl Falk-Petersen, Rebekka Löffler, David E. Gloriam, Petrine Wellendorph, Frederik Rostrup, Stine Buchleithner, Bente Frølund
مصطلحات موضوعية: Transmembrane domain, Diazepam binding, Docking (molecular), Stereochemistry, GABAA receptor, Chemistry, Allosteric regulation, Functional selectivity, Binding site, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::acdb2ee1ddc3df8b270b203444a0df85
https://doi.org/10.1101/2021.01.21.427670 -
5
المؤلفون: David E. Gloriam, Tanja Schirmeister, Christina Birkedahl Falk-Petersen, Stine Buchleithner, Kasper Harpsøe, Frederik Rostrup, Petrine Wellendorph, Sascha Jung, Bente Frølund, Irene Conforti
مصطلحات موضوعية: Membrane potential, Imidazopyridine, GABAA receptor, Chemistry, Biophysics, Potency, Binding site, Receptor, Aminobutyric acid, Plate reader
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::baf5e25f7f3f2a9f11633076a277c398
https://doi.org/10.26434/chemrxiv.13395416.v1