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المؤلفون: Sho Sato, Andy Sykes, Stuart Stafford, Yoshihiko Tagawa, Rosa Fradley, Shyam Bechar, Eimear Howley, Tomoki Yoneyama, Toshal Patel, Toshiya Moriwaki, Satoru Asahi
المصدر: Pharmaceutical Research
مصطلحات موضوعية: D-Amino-Acid Oxidase, Male, Kinetics, D-amino acid oxidase, Pharmaceutical Science, PK/PD, multilayer quantitative model, Blood–brain barrier, Mice, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, medicine, Animals, Pharmacology (medical), 030304 developmental biology, TAK-831, Pharmacology, 0303 health sciences, Oxidase test, Dose-Response Relationship, Drug, Chemistry, Organic Chemistry, Brain, D-amino acid oxidase inhibitor, Quantitative model, Receptor–ligand kinetics, Mice, Inbred C57BL, medicine.anatomical_structure, Pharmacodynamics, Schizophrenia, Biophysics, Molecular Medicine, target occupancy, 030217 neurology & neurosurgery, Research Paper, Biotechnology
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المؤلفون: K. Real, Matt Barnes, Richard J. Davenport, Helen M. Cox, Robert Newman, Stuart Stafford, Helen Heffron, Johannes Grosse, Sarah Forbes, Gareth Coope
المصدر: Diabetes. 64:3763-3771
مصطلحات موضوعية: Agonist, endocrine system, medicine.medical_specialty, medicine.drug_class, Endocrinology, Diabetes and Metabolism, media_common.quotation_subject, Appetite, Mice, Obese, Receptors, Cell Surface, Enteroendocrine cell, Biology, Dipeptidyl peptidase, Impaired glucose tolerance, Eating, Mice, Glucagon-Like Peptide 1, Internal medicine, Glucose Intolerance, Free fatty acid receptor 2, Internal Medicine, medicine, Animals, Peptide YY, Obesity, Intestinal Mucosa, Gastrointestinal Transit, Cells, Cultured, media_common, digestive, oral, and skin physiology, medicine.disease, Intestines, Endocrinology, Decreased glucose tolerance, hormones, hormone substitutes, and hormone antagonists
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9691959fca26e3bb88814cbebc62e29c
https://doi.org/10.2337/db15-0481 -
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المؤلفون: Richard J. Davenport, Sarah Bousba, Mathew Leveridge, David Harrison, Junji Matsui, Taku Sakurai, Louise Dickson, Kazumasa Ogawa, Matt Barnes, Stephen Robert Mack, Johannes Grosse, Parmar Alka, Laura Parton, Jennifer Cameron, Andy Sykes, Stuart Stafford
المصدر: European Journal of Pharmacology. 727:1-7
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, Mice, 129 Strain, Side effect, medicine.drug_class, Adipose Tissue, White, Lipolysis, White adipose tissue, GPR81, Biology, Transfection, Receptors, G-Protein-Coupled, Mice, Structure-Activity Relationship, In vivo, 3T3-L1 Cells, Internal medicine, Drug Discovery, Adipocytes, Flushing, medicine, Animals, Structure–activity relationship, Lactic Acid, Receptor, Hypolipidemic Agents, Mice, Knockout, Pharmacology, Dose-Response Relationship, Drug, High-Throughput Screening Assays, Mice, Inbred C57BL, Thiazoles, Endocrinology, Injections, Intraperitoneal