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1
المؤلفون: Hilary A. Wilkinson, Chun Cheng, Susan P. Rohrer, Kwok-lam Karen Hong, Michael Chisamore, Stephen E. Alves
المصدر: Biomarkers
مصطلحات موضوعية: endocrine, steroid nuclear receptor, Health, Toxicology and Mutagenesis, Clinical Biochemistry, Serum protein, Estrogen receptor, Biochemistry, Mice, Animals, Estrogen Receptor beta, RNA, Messenger, Estrogen receptor beta, Oligonucleotide Array Sequence Analysis, Mice, Knockout, Membrane Glycoproteins, Estradiol, biology, Gene Expression Profiling, Binding protein, Uterus, Estrogen Receptor alpha, Blood Proteins, Molecular biology, Rats, Gene expression profiling, Gene Expression Regulation, Liver, Nuclear receptor, Cancer research, biology.protein, Biomarker (medicine), Female, Carrier Proteins, Estrogen receptor alpha, Lipopolysaccharide binding protein, Biomarkers, Acute-Phase Proteins, Research Article
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2
المؤلفون: Susan P. Rohrer, Sheng Jian Cai, James Schaeffer, Elizabeth T. Birzin, J. Don Chen, Osvaldo A. Flores, Paul Zuck, Ralph T. Mosley, Michael J. Chisamore, Hilary A. Wilkinson, Gregory O'Donnell
المصدر: Drug Development Research. 69:203-218
مصطلحات موضوعية: Estrogen-related receptor, Estrogen-related receptor alpha, Nuclear receptor, Biochemistry, Docking (molecular), Drug Discovery, Coactivator, Estrogen receptor, Homology modeling, Biology, Receptor
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3
المؤلفون: Susan P. Rohrer, Edward C. Hayes, Paula M.D. Fitzgerald, Yi Tien Yang, Carolyn DaSilva, Lee-Yuh Pai, Elizabeth T. Birzin, Frank P. DiNinno, Milton L. Hammond, Ralph T. Mosley, Wanda Chan, Liangqin Guo, James M. Schaeffer, Kevin D. Dykstra, Bryan Kraker
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:2322-2328
مصطلحات موضوعية: Indoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Estrogen receptor, Breast Neoplasms, Ligands, Biochemistry, Bazedoxifene, Inhibitory Concentration 50, Cell Line, Tumor, Drug Discovery, medicine, Humans, Molecular Biology, Estrogen receptor beta, Indole test, Chemistry, Uterus, Organic Chemistry, Estrogen Antagonists, Estrogen Receptor alpha, Antagonist, Cancer cell, Molecular Medicine, Female, Estrogen receptor alpha, Linker, medicine.drug
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4
المؤلفون: Donald M. Sperbeck, Elizabeth T. Birzin, Dann L. Parker, Robert R. Wilkening, Katalin Frisch, Dongfang Meng, Lawrence F. Colwell, Ronald W. Ratcliffe, Stefan Nilsson, Milton L. Hammond, Susan P. Rohrer, Sherrie Lambert, Ann-Gerd Thorsell, Mark L. Greenlee
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4652-4656
مصطلحات موضوعية: Agonist, medicine.medical_specialty, medicine.drug_class, Clinical Biochemistry, Triazole, Pharmaceutical Science, Ligands, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Internal medicine, Drug Discovery, polycyclic compounds, medicine, Animals, Estrogen Receptor beta, Humans, Structure–activity relationship, Selective receptor modulator, Molecular Biology, reproductive and urinary physiology, Estrogen receptor beta, Fluorenes, Molecular Structure, Chemistry, Organic Chemistry, Rats, Bioavailability, Endocrinology, Selective estrogen receptor modulator, Molecular Medicine, Bioisostere, Azo Compounds, hormones, hormone substitutes, and hormone antagonists
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5
المؤلفون: Milton L. Hammond, Elizabeth T. Birzin, Wanying Sun, Lovji D. Cama, Louis Locco, Ralph T. Mosley, Susan P. Rohrer, Sudha Warrier
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:1468-1472
مصطلحات موضوعية: Agonist, Molecular model, Stereochemistry, medicine.drug_class, Fluoroimmunoassay, Clinical Biochemistry, Pharmaceutical Science, Ligands, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, Coactivator, Benzene Derivatives, Tumor Cells, Cultured, polycyclic compounds, medicine, Estrogen Receptor beta, Humans, Structure–activity relationship, Benzopyrans, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Chemistry, Organic Chemistry, Estrogen Receptor alpha, General Medicine, Selective estrogen receptor modulator, Molecular Medicine, Selectivity, hormones, hormone substitutes, and hormone antagonists, Lactone
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6
المؤلفون: Nandini Sharma, Consuelo Tudela, Milton L. Hammond, Fang Chen, Jerry D. Morgan, Timothy A. Blizzard, Susan P. Rohrer, Mark A. Holmes, Ralph Troy Mosley, Wanda Chan, Bryan Kraker, Candido Gude, Marina Mojena, Kristin Knecht, Qin Su, Paula M.D. Fitzgerald, Elizabeth T. Birzin
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:834-838
مصطلحات موضوعية: Androstenediol, Models, Molecular, Selective Estrogen Receptor Modulators, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Estrogen receptor, Crystallography, X-Ray, Ligands, Biochemistry, Chemical synthesis, Steroid, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Estrogen Receptor beta, Humans, Molecular Biology, Chemistry, Organic Chemistry, Stereoisomerism, In vitro, Selective estrogen receptor modulator, Molecular Medicine
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7
المؤلفون: Lee-Yuh Pai, Carolyn DaSilva, Yi Tien Yang, Elizabeth T. Birzin, Ralph T. Mosley, Timothy A. Blizzard, Jerry D. Morgan, Frank P. DiNinno, Edward C. Hayes, Susan P. Rohrer, Milton L. Hammond, Wanda Chan
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:5124-5128
مصطلحات موضوعية: Selective Estrogen Receptor Modulators, Ligand, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Estrogen Receptor alpha, Antagonist, Pharmaceutical Science, Estrogen receptor, Tumor cells, Ligands, Biochemistry, Rats, Oxathiins, Drug Discovery, Side chain, Animals, Molecular Medicine, Dihydrobenzoxathiin, Molecular Biology
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8
المؤلفون: Donald B. Kimmel, Lee Yuh Pai, Carolyn DaSilva, Paula M.D. Fitzgerald, Nandini Sharma, Alfred A. Reszka, Wanda Chan, Milton L. Hammond, Elizabeth T. Birzin, Yi Tien Yang, Lawrence F. Colwell, Susan Li, Hilary A. Wilkinson, Sharon Adamski, Qiang Tan, Jerry D. Morgan, Leonard P. Freedman, Edward C. Hayes, James M. Schaeffer, John E. Fisher, Susan P. Rohrer, Timothy A. Blizzard, Frank P. DiNinno, Sudha Warrier, Joel B. Yudkovitz
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1675-1681
مصطلحات موضوعية: Selective Estrogen Receptor Modulators, medicine.medical_specialty, Clinical Biochemistry, Gene Expression, Pharmaceutical Science, Estrogen receptor, Ligands, Biochemistry, Bone resorption, Cell Line, Rats, Sprague-Dawley, Structure-Activity Relationship, In vivo, Internal medicine, Drug Discovery, medicine, Animals, Humans, Chromans, Molecular Biology, Binding Sites, Molecular Structure, Chemistry, Cell growth, Uterus, Organic Chemistry, Estrogen Receptor alpha, Organ Size, Antiestrogen, Rats, Resorption, Endocrinology, Models, Chemical, Molecular Medicine, Female, Signal transduction, Estrogen receptor alpha, Protein Binding
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9
المؤلفون: Wanda Chan, Elizabeth T. Birzin, Lee-Yuh Pai, James M. Schaeffer, Edward C. Hayes, Carolyn DaSilva, Susan P. Rohrer, Yi Tien Yang, Frank P. DiNinno, Milton L. Hammond, Jian Liu, Ralph T. Mosley
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:715-718
مصطلحات موضوعية: Models, Molecular, Gene isoform, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Estrogen receptor, Ligands, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Humans, Protein Isoforms, Chromans, Molecular Biology, Cell Proliferation, Estradiol, Bicyclic molecule, Ligand, Chemistry, Uterus, Organic Chemistry, Estrogen Receptor alpha, Biological activity, Lasofoxifene, Molecular Medicine, Female, Selectivity, Protein Binding, medicine.drug
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10
المؤلفون: Frank P. DiNinno, Milton L. Hammond, James M. Schaeffer, Paula M.D. Fitzgerald, Zhoupeng Zhang, Edward C. Hayes, Wanda Chan, Timothy A. Blizzard, Elizabeth T. Birzin, Nandini Sharma, Carolyn DaSilva, Ying Li, Seongkon Kim, Wei Tang, Yi Tien Yang, Jane Y. Wu, Helen Chen, Susan P. Rohrer, Jerry D. Morgan, Lee-Yuh Pai
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:107-113
مصطلحات موضوعية: Models, Molecular, Selective Estrogen Receptor Modulators, Pyrrolidines, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Alkylation, Ligands, Biochemistry, Chemical synthesis, Pyrrolidine, Oxathiins, chemistry.chemical_compound, Drug Discovery, Side chain, Molecular Biology, Alkyl, chemistry.chemical_classification, Bicyclic molecule, Ligand, Organic Chemistry, Receptors, Estrogen, chemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Linker