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المؤلفون: Percy F. Sumariwalla, Marc Feldmann, Susanna Tchilibon, Raphael Mechoulam, Ester Fride, Ruth Gallily
مصطلحات موضوعية: Central Nervous System, Lipopolysaccharides, Cyclohexanecarboxylic Acids, medicine.medical_treatment, Immunology, Anti-Inflammatory Agents, Arthritis, Mitosis, Pharmacology, Severity of Illness Index, Proinflammatory cytokine, Mice, Immune system, Rheumatology, medicine, Immunology and Allergy, HU-320, Macrophage, Animals, Cannabidiol, Humans, Pharmacology (medical), Lymphocytes, Cells, Cultured, Immunity, Cellular, Mice, Inbred BALB C, business.industry, Tumor Necrosis Factor-alpha, Macrophages, medicine.disease, Arthritis, Experimental, Mice, Inbred C57BL, Ajulemic acid, Tumor necrosis factor alpha, Cattle, Female, Joints, Cannabinoid, business, Immunosuppressive Agents, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::506531a8e4a85c177d0caf18d74dc742
https://ora.ox.ac.uk/objects/uuid:018c4232-99f6-424a-b01e-471421dab9c9 -
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المصدر: Annual reports in medicinal chemistry. 38
مصطلحات موضوعية: Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::92f0a94616fd1c1a304ff3300f8e8490
https://pubmed.ncbi.nlm.nih.gov/26640305 -
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المؤلفون: Bhalchandra V. Joshi, Heng T. Duong, Dmitry Sonin, Zhan-Guo Gao, Bruce T. Liang, Susanna Tchilibon, Kenneth A. Jacobson
المصدر: Journal of Medicinal Chemistry. 48:8103-8107
مصطلحات موضوعية: Agonist, Adenosine, Cardiotonic Agents, Adenosine A2 Receptor Agonists, Receptor, Adenosine A2A, medicine.drug_class, Stereochemistry, Myocardial Infarction, CHO Cells, Ventricular Function, Left, Article, Mice, Adenosine A3 Receptor Agonists, Cricetinae, Drug Discovery, medicine, Animals, Humans, Potency, Receptor, Cardioprotection, Receptor, Adenosine A1, Chemistry, Chinese hamster ovary cell, Receptor, Adenosine A3, Adenosine receptor, Adenosine A1 Receptor Agonists, Drug Design, Reperfusion Injury, Molecular Medicine, medicine.drug
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المؤلفون: Kenneth A. Jacobson, Qingfeng Yang, Hak Sung Kim, Harvey B. Pollard, Ofer Eidelman, Bette S. Pollard, Jian Zhang, Hung Caohuy, Susanna Tchilibon
المصدر: Biochem Pharmacol
مصطلحات موضوعية: medicine.medical_specialty, Cystic Fibrosis, Pyridinium Compounds, Respiratory Mucosa, Biology, Biochemistry, Article, Proinflammatory cytokine, Surface-Active Agents, Internal medicine, medicine, Humans, Interleukin 8, Transcription factor, Pharmacology, Dose-Response Relationship, Drug, Tumor Necrosis Factor-alpha, Kinase, Interleukin-8, NF-kappa B, IκBα, Endocrinology, Mechanism of action, Cancer research, Phosphorylation, Salts, medicine.symptom, Signal transduction, HeLa Cells, Signal Transduction
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المصدر: Biochemical Pharmacology. 68:231-237
مصطلحات موضوعية: Isatin, Agonist, P2Y receptor, medicine.drug_class, Inositol Phosphates, Allosteric regulation, Astrocytoma, Tritium, Biochemistry, Article, Receptors, G-Protein-Coupled, Receptors, Purinergic P2Y1, Adenosine Triphosphate, Allosteric Regulation, Purinergic P2 Receptor Antagonists, Tumor Cells, Cultured, Radioligand, medicine, Enzyme-linked receptor, Humans, Receptor, G protein-coupled receptor, Pharmacology, Binding Sites, Nucleotides, Chemistry, Adenosine Diphosphate, Kinetics, Competitive antagonist, Biophysics, Signal Transduction
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المؤلفون: Philippe Van Rompaey, Brian A Harris, Michihiro Ohno, Susanna Tchilibon, Ariel S. Gross, Zhan-Guo Gao, Heng T. Duong, Serge Van Calenbergh, Kenneth A. Jacobson, Soo-Kyung Kim
المصدر: Bioorganic & Medicinal Chemistry. 12:2995-3007
مصطلحات موضوعية: Models, Molecular, Agonist, Adenosine, Intrinsic activity, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Article, Structure-Activity Relationship, Drug Discovery, Purinergic P1 Receptor Agonists, medicine, Humans, Binding site, Molecular Biology, G protein-coupled receptor, Binding Sites, Deoxyadenosines, Chemistry, Organic Chemistry, Receptors, Purinergic P1, Ligand (biochemistry), Adenosine receptor, Recombinant Proteins, Docking (molecular), Molecular Medicine, medicine.drug
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المؤلفون: John B. Davis, Aniello Schiano Moriello, Ines Brandi, Vincenzo Di Marzo, Tiziana Bisogno, Susanna Tchilibon, Datta E. Ponde, Luciano De Petrocellis, Raphael Mechoulam, Lumir Hanus
المصدر: British Journal of Pharmacology. 134:845-852
مصطلحات موضوعية: Pharmacology, Cannabinoid receptor, Stereochemistry, medicine.medical_treatment, Anandamide, Endocannabinoid system, digestive system diseases, chemistry.chemical_compound, surgical procedures, operative, Mechanism of action, chemistry, Fatty acid amide hydrolase, medicine, Cannabinoid receptor type 2, lipids (amino acids, peptides, and proteins), Cannabinoid, medicine.symptom, Cannabidiol, medicine.drug
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المؤلفون: Simonetta Lanati, Susanna Tchilibon, Giovanni Fronza, Roberta Rallo, Piero Grasselli, Claudio Fuganti
المصدر: J. Chem. Soc., Perkin Trans. 1. :2927-2930
مصطلحات موضوعية: Reduction (complexity), Syn and anti addition, Hydrogen, chemistry, Stereochemistry, Absolute configuration, chemistry.chemical_element, Molecule, Hydrogen atom, Enantiomer, Yeast
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::dc08b83eb940b2ba780d05ab47f4842c
https://doi.org/10.1039/p19940002927 -
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المؤلفون: Bhalchandra V. Joshi, Heng T. Duong, Kenneth A. Jacobson, Soo-Kyung Kim, Eunjoo Roh, Stefano Costanzi, Zhan-Guo Gao, Susanna Tchilibon
المصدر: Nucleosides, nucleotidesnucleic acids. 25(12)
مصطلحات موضوعية: Models, Molecular, P2Y receptor, Intrinsic activity, Stereochemistry, Ribose, Molecular Conformation, Ligands, Biochemistry, Article, Receptors, Purinergic P2Y1, Cations, Genetics, medicine, Animals, Humans, Nucleotide, Receptor, G protein-coupled receptor, chemistry.chemical_classification, Nucleotides, Receptors, Purinergic P2, Cell Membrane, Receptor, Adenosine A3, Nucleosides, General Medicine, Genetic Therapy, Adenosine receptor, Adenosine, chemistry, Models, Chemical, Purines, Molecular Medicine, Adenosine A2B receptor, medicine.drug
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المؤلفون: Bhalchandra V. Joshi, Susanna Tchilibon, Heng T. Duong, Zhan-Guo Gao, Soo-Kyung Kim, Kenneth A. Jacobson
المصدر: Journal of medicinal chemistry. 48(6)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Stereoisomerism, CHO Cells, Chemical synthesis, Article, Nucleobase, Radioligand Assay, Structure-Activity Relationship, Cricetulus, Adenosine A3 Receptor Agonists, Cricetinae, Drug Discovery, Cyclic AMP, Structure–activity relationship, Animals, Humans, Binding site, Binding Sites, Bicyclic molecule, Chemistry, Adenine, Receptor, Adenosine A3, Nucleosides, Adenosine receptor, Rats, Molecular Medicine