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المؤلفون: Jayaprakasam Bolleddula, Xiaofei Zhou, Douglas V. Faller, Yuexian Li, Swapan Chowdhury, Dan Zhao, Hélène M. Faessel, Farhad Sedarati, Karthik Venkatakrishnan, Zsuzsanna Papai
المصدر: Investigational New Drugs. 39:488-498
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, business.industry, Urine, Carboplatin, Excretion, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Oncology, chemistry, Paclitaxel, Pharmacokinetics, Docetaxel, 030220 oncology & carcinogenesis, medicine, Pharmacology (medical), business, Feces, medicine.drug, Whole blood
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المؤلفون: Afrand Kamali, Mohammad Shadid, Michael D. Smith, Jayaprakasam Bolleddula, Abhi Shah, Swapan Chowdhury
المصدر: Drug Metabolism and Disposition. 48:1239-1245
مصطلحات موضوعية: Pharmacology, Antibody-drug conjugate, Catabolism, Chemistry, Pharmaceutical Science, 030226 pharmacology & pharmacy, Cyclase, Cathepsin B, In vitro, 03 medical and health sciences, 0302 clinical medicine, Biochemistry, Mechanism of action, In vivo, 030220 oncology & carcinogenesis, medicine, medicine.symptom, Conjugate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::73c7b913bf7e365f1149b6e3dd3ec173
https://doi.org/10.1124/dmd.120.000194 -
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المؤلفون: Suguru Kato, Swapan Chowdhury, Jayaprakasam Bolleddula, Mihaela Plesescu, Yoshinari Miyata, Abhi Shah, Xiaochun Zhu
المصدر: Drug Metabolism and Disposition. 48:934-943
مصطلحات موضوعية: Male, Metabolite, Cyproheptadine, Drug Evaluation, Preclinical, Pharmaceutical Science, Mianserin, Urine, Pharmacology, 030226 pharmacology & pharmacy, Excretion, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, In vivo, medicine, Animals, Bile, Humans, Distribution (pharmacology), Biotransformation, Transplantation Chimera, Desloratadine, Loratadine, Hepatobiliary Elimination, Liver, chemistry, 030220 oncology & carcinogenesis, Hepatocytes, Carbamates, Drug metabolism, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ced06eca08636d58fdba47f17d4f460
https://doi.org/10.1124/dmd.120.000128 -
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المؤلفون: Cindy Q. Xia, Sandeepraj Pusalkar, Yuexian Li, Karthik Venkatakrishnan, Suresh K. Balani, Lawrence Cohen, Xiaofei Zhou, Wen Chyi Shyu, Jun Johnny Yang, Swapan Chowdhury, Chuang Lu
المصدر: Drug Metabolism and Disposition. 48:217-229
مصطلحات موضوعية: Pharmacology, business.industry, CYP3A, Metabolite, Acyl glucuronidation, Aurora A kinase, Pharmaceutical Science, Urine, 030226 pharmacology & pharmacy, Excretion, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, chemistry, Pharmacokinetics, 030220 oncology & carcinogenesis, Alisertib, Medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::166eb285f2919cd372a7ec5c53356ca7
https://doi.org/10.1124/dmd.119.087338 -
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المؤلفون: P. P. Chothe, E. van de Steeg, Catherijne A. J. Knibbe, Ian P.J. Alwayn, Swapan Chowdhury, Andy Z. X. Zhu, L. J. Stevens, Joanne M. Donkers, Wouter H. J. Vaes
المصدر: Drug Metabolism and Disposition, 49(9), 780-789. AMER SOC PHARMACOLOGY EXPERIMENTAL THERAPEUTICS
مصطلحات موضوعية: Statin, medicine.drug_class, Metabolic Clearance Rate, Swine, Metabolite, Atorvastatin, Drug Evaluation, Preclinical, Pharmaceutical Science, Pharmacology, In Vitro Techniques, chemistry.chemical_compound, Medicine, Animals, Rosuvastatin, Drug Interactions, Pitavastatin, Machine perfusion, business.industry, Reproducibility of Results, Equipment Design, Hepatobiliary Elimination, Perfusion, chemistry, Liver, Inactivation, Metabolic, Hydroxymethylglutaryl-CoA Reductase Inhibitors, business, Ex vivo, medicine.drug
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79e1d07819595c8930b13ced62ae3d42
https://pubmed.ncbi.nlm.nih.gov/34330719 -
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المؤلفون: Sandeepraj Pusalkar, Xiaofei Zhou, Yuexian Li, Shawn Searle, Claudio Dansky Ullmann, Swapan Chowdhury, Karthik Venkatakrishnan
المصدر: Investigational New Drugs. 37:666-673
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, business.industry, Aurora A kinase, Urine, Excretion, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Oncology, chemistry, Pharmacokinetics, 030220 oncology & carcinogenesis, Alisertib, Medicine, Pharmacology (medical), business, Adverse effect, Drug metabolism, Feces
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المؤلفون: Xiaofei, Zhou, Farhad, Sedarati, Douglas V, Faller, Dan, Zhao, Hélène M, Faessel, Swapan, Chowdhury, Jayaprakasam, Bolleddula, Yuexian, Li, Karthik, Venkatakrishnan, Zsuzsanna, Papai
المصدر: Investigational New Drugs
مصطلحات موضوعية: Male, Dose-Response Relationship, Drug, NEDD8 Protein, pevonedistat, Cyclopentanes, Middle Aged, phase I, Pyrimidines, elimination, Area Under Curve, Neoplasms, Phase I Studies, Antineoplastic Combined Chemotherapy Protocols, Humans, Female, advanced solid tumors, Enzyme Inhibitors, Radiopharmaceuticals, pharmacokinetics, mass balance, Aged, Half-Life
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المؤلفون: Michael J. Hanley, Cindy Q. Xia, Swapan Chowdhury, Karthik Venkatakrishnan, Sandeepraj Pusalkar, Mihaela Plesescu, Xiaoquan Zhang, Neeraj Gupta, Jing-Tao Wu
المصدر: Cancer Chemotherapy and Pharmacology. 82:803-814
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Cancer Research, Metabolite, Urine, Toxicology, Tandem mass spectrometry, Ixazomib, Excretion, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Oncology, chemistry, Biotransformation, In vivo, 030220 oncology & carcinogenesis, Pharmacology (medical), Feces
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المؤلفون: Cornelis E. C. A. Hop, Swapan Chowdhury, Douglas K. Spracklin, Simone Schadt, Christoph Funk, W. Griffith Humphreys, Angus N. R. Nedderman, Fumihiko Igarashi, Josh Yuan, Chandra Prakash, Frank Runge, Holger Scheible, Mark Kagan, S. Cyrus Khojasteh, Piet Swart, R. Scott Obach, Bojan Bister, Alexander David James, Susanna Tse
المصدر: BASE-Bielefeld Academic Search Engine
مصطلحات موضوعية: 0301 basic medicine, Drug Industry, Metabolite, Pharmaceutical Science, Human metabolism, Computational biology, 030226 pharmacology & pharmacy, Food and drug administration, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Animals, Humans, Medicine, Drug Interactions, Safety testing, Pharmaceutical industry, Pharmacology, United States Food and Drug Administration, business.industry, United States, 030104 developmental biology, Pharmaceutical Preparations, chemistry, Drug development, Inactivation, Metabolic, Experimental methods, business, Drug metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::28c0739606a23742034a3be6254e08fa
https://doi.org/10.1124/dmd.117.079848 -
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المؤلفون: Karthik Venkatakrishnan, Michael J. Hanley, Sandeepraj Pusalkar, Neeraj Gupta, Steven Zhang, Mihaela Plesescu, Xiaoquan Zhang, Bingxia Wang, Dale R. Shepard, Swapan Chowdhury, Cindy Q. Xia
المصدر: Investigational New Drugs. 36:407-415
مصطلحات موضوعية: Pharmacology, Urine, 030226 pharmacology & pharmacy, Ixazomib, Excretion, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Oncology, chemistry, Pharmacokinetics, Oral administration, 030220 oncology & carcinogenesis, Pharmacology (medical), Adverse effect, Feces, ADME