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المؤلفون: Gaku Sakaguchi, Tetsuji Ito, Naoki Tsuno, Mikie Hinata, Akira Yukimasa, Yasuyoshi Iso, Satoko Funaki, Daiki Nagamatsu, Miki Tanimura, Miyuki Yamamoto, Tatsuhiko Ueno, Toshiyuki Kanemasa, Yoko Nishimura, Masahiko Soga, Natsue Yamanada, Yasuhide Morioka, Osamu Yoshida, Narumi Horita, Masayuki Imai, Takatsugu Inoue, Yusuke Ichihashi, Hiroki Yamaguchi, Hidetoshi Matsuda
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:4930-4935
مصطلحات موضوعية: 0301 basic medicine, Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Biological Availability, TRPV Cation Channels, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, ADME, Analgesics, Drug discovery, Chemistry, Organic Chemistry, Antagonist, Bioavailability, 030104 developmental biology, Competitive antagonist, Molecular Medicine, Lead compound, 030217 neurology & neurosurgery
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2
المؤلفون: Kazuto Nunomura, Bangzhong Lin, Yusuke Higuchi, Takatsugu Inoue, Toru Yoneyama, Nobuo Kato, Yoshio Honma
المصدر: Bioorganicmedicinal chemistry letters. 28(4)
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Cotylenin A, 010402 general chemistry, 01 natural sciences, Biochemistry, Protein–protein interaction, chemistry.chemical_compound, Structure-Activity Relationship, Interferon, Cell Line, Tumor, Drug Discovery, medicine, Humans, Glycosides, Molecular Biology, 14-3-3 protein, Biological evaluation, Molecular Structure, 010405 organic chemistry, Chemistry, Protein Stability, Organic Chemistry, Stereoisomerism, Semisynthesis, 0104 chemical sciences, 14-3-3 Proteins, Fusicoccin, Cancer cell, Molecular Medicine, Diterpenes, medicine.drug
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3
المؤلفون: Michael Weyand, Alfred Wittinghofer, Claudia Oecking, Takeshi Sassa, Takatsugu Inoue, Nobuo Kato, Christian Ottmann
المساهمون: Chemical Biology
المصدر: Journal of Molecular Biology, 386(4), 913-919. Academic Press Inc.
مصطلحات موضوعية: Models, Molecular, Phosphopeptides, Amino Acid Motifs, Molecular Sequence Data, Antineoplastic Agents, Plasma protein binding, Calorimetry, Biology, SDG 3 – Goede gezondheid en welzijn, Crystallography, X-Ray, Protein Structure, Secondary, Hydroxylation, Structure-Activity Relationship, chemistry.chemical_compound, Protein structure, SDG 3 - Good Health and Well-being, Structural Biology, Differentiation therapy, Tobacco, Humans, Structure–activity relationship, Amino Acid Sequence, Glycosides, Molecular Biology, Regulation of gene expression, Protein Stability, Proton-Translocating ATPases, 14-3-3 Proteins, Biochemistry, chemistry, Fusicoccin, Target protein, Diterpenes, Protein Multimerization, Protein Binding
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4
المؤلفون: Takeshi Sassa, Junko Ohkanda, Takatsugu Inoue, Manuela Molzan, Martin Schuler, Nobuo Kato, Frank Breitenbuecher, Malgorzata Skwarczynska, Stefan Kasper, Christian Ottmann, Lars Röglin
المساهمون: Chemical Biology
المصدر: ACS Chemical Biology, 8(9), 1869-1875. American Chemical Society
مصطلحات موضوعية: Models, Molecular, Somatic cell, Mutant, Medizin, Mice, SCID, Biology, SDG 3 – Goede gezondheid en welzijn, Biochemistry, Mice, SDG 3 - Good Health and Well-being, In vivo, Cell Line, Tumor, Neoplasms, medicine, Animals, Humans, Protein Interaction Maps, Gene, Biological Products, Cancer, General Medicine, medicine.disease, Molecular biology, In vitro, Proto-Oncogene Proteins c-raf, 14-3-3 Proteins, Cell culture, Cancer research, biology.protein, ras Proteins, Molecular Medicine, raf Kinases, Antibody, Diterpenes
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المؤلفون: Nobuo Kato, Koshi Kawakami, Miki Tongu, Keizo Takenaga, Yoshio Honma, Miho Akimoto, Yuriko Maruyama, Takeshi Sassa, Takaya Yamada, Takatsugu Inoue, Junji Suzumiy, Miho Hattori, Junko Ohkanda
المصدر: Anti-cancer agents in medicinal chemistry. 12(7)
مصطلحات موضوعية: Cancer Research, medicine.medical_specialty, Transplantation, Heterologous, Mice, Nude, Antineoplastic Agents, Breast Neoplasms, Mice, Cancer stem cell, Pancreatic cancer, Internal medicine, Cell Line, Tumor, medicine, Human Umbilical Vein Endothelial Cells, Cytotoxic T cell, Animals, Humans, Glycosides, Progenitor cell, Pharmacology, Ovarian Neoplasms, Mice, Inbred BALB C, biology, Tumor hypoxia, CD44, Mycotoxins, medicine.disease, Hypoxia-Inducible Factor 1, alpha Subunit, Cell Hypoxia, Pancreatic Neoplasms, Endocrinology, Cell culture, biology.protein, Cancer research, Molecular Medicine, Female, Stem cell, Diterpenes, Proto-Oncogene Proteins c-akt
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::563af2fbc51e497ce215e52e33d7ce1c
https://pubmed.ncbi.nlm.nih.gov/22263802 -
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المؤلفون: Keiji Matsumoto, Koichi Yoshioka, Toshio Tanaka, Yoshinosuke Usuki, Takatsugu Inoue, Hideo Iio
المصدر: Bioorganicmedicinal chemistry letters. 16(6)
مصطلحات موضوعية: Antifungal Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Saccharomyces cerevisiae, Gram-Positive Bacteria, Biochemistry, Chemical synthesis, Guanidines, Structure-Activity Relationship, Polyol, Drug Discovery, medicine, Structure–activity relationship, Moiety, Molecular Biology, Antibacterial agent, chemistry.chemical_classification, Chemistry, Organic Chemistry, Cell Membrane, Fungi, Antimicrobial, In vitro, Anti-Bacterial Agents, Oxidative Stress, Mechanism of action, Phosphatidylcholines, Molecular Medicine, medicine.symptom, Reactive Oxygen Species