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1
المؤلفون: Arsalan Qazi Shabbir, Brian Berman, Tanya MacNeil, Kim Mark Knudsen
المصدر: Dermatologic Surgery. 43:424-430
مصطلحات موضوعية: Adult, Average duration, medicine.medical_specialty, Ingenol Mebutate Gel, Adolescent, Keratosis, medicine.medical_treatment, Topical treatment, Dermatology, Administration, Cutaneous, Cryosurgery, Severity of Illness Index, 030207 dermatology & venereal diseases, 03 medical and health sciences, 0302 clinical medicine, Risk Factors, medicine, Humans, 030212 general & internal medicine, Scalp, business.industry, Actinic keratosis, General Medicine, medicine.disease, United States, Surgery, Keratosis, Actinic, Treatment Outcome, medicine.anatomical_structure, Multicenter study, Face, Dermatologic Agents, Diterpenes, business, Gels
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fc873523c95fc9ad508f82157242ccde
https://doi.org/10.1097/dss.0000000000000989 -
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المؤلفون: Palucki Brenda, Patrick G. Pollard, Liangqin Guo, Tung M. Fong, Matthew J. Wyvratt, Randy R. Miller, Shuwen He, Constantin Tamvakopoulos, Iyassu K. Sebhat, Qianping Peng, Ravi P. Nargund, Zhixiong Ye, Airu S. Chen, Doreen E. Cashen, David H. Weinberg, Min K. Park, Raman K. Bakshi, D. Euan MacIntyre, Howard Y. Chen, Rui Tang, Tanya MacNeil, Qingmei Hong, Alison M. Strack, Ralph A. Stearns, Jian Liu, William J. Martin
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2330-2334
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, Partial agonist, Piperazines, Rats, Sprague-Dawley, Eating, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Oral administration, In vivo, Drug Discovery, medicine, Animals, Urea, Obesity, Receptor, Molecular Biology, Organic Chemistry, Haplorhini, Rats, Disease Models, Animal, Piperazine, chemistry, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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3
المؤلفون: Yingjie Lai, Ralph A. Stearns, Qianping Peng, Ravi P. Nargund, Qingmei Hong, Jian Liu, Rui Tang, Matthew J. Wyvratt, Raman K. Bakshi, Randy R. Miller, Tianying Jian, Alison M. Strack, Tanya MacNeil, Liangqin Guo, Howard Y. Chen, James Dellureficio, Iyassu K. Sebhat, Peter H. Dobbelaar, Airu S. Chen, Constantin Tamvakopoulos, David H. Weinberg, Tung M. Fong, Christopher L. Franklin, Shuwen He, Zhixiong Ye
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4399-4405
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Pyrrolidines, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Anti-Obesity Agents, Internal medicine, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Spiro Compounds, Obesity, Molecular Biology, Mice, Knockout, Chemistry, Body Weight, Organic Chemistry, Amides, Rats, Endocrinology, Drug development, Anorectic, Receptor, Melanocortin, Type 4, Molecular Medicine
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المؤلفون: Howard Y. Chen, William J. Martin, D. Euan MacIntyre, Zhixiong Ye, Raman K. Bakshi, Alison M. Strack, Doreen E. Cashen, Jian Liu, Yingjie Lai, Tianying Jian, Constantin Tamvakopoulos, Nancy N. Tsou, Shuwen He, James Dellureficio, Tung M. Fong, Peter H. Dobbelaar, David H. Weinberg, Airu S. Chen, Qingmei Hong, Iyassu K. Sebhat, Tanya MacNeil, Christopher L. Franklin, Ravi P. Nargund, Ralph A. Stearns, Rui Tang, Richard G. Ball, Matthew J. Wyvratt, Randy R. Miller, Liangqin Guo, Qianping Peng
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2106-2110
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, Cricetulus, Dogs, Erectile Dysfunction, Cricetinae, Drug Discovery, medicine, Animals, Humans, Spiro Compounds, Receptor, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Haplorhini, Rats, Bioavailability, Indans, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding
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المؤلفون: Heather L. Sings, Mark T. Goulet, Matthew J. Wyvratt, Iyassu K. Sebhat, Liangqin Guo, Rui Tang, Ravi P. Nargund, Qianping Peng, Euan Macintyre, Feroze Ujjainwalla, Constantin Tamvakopoulos, Zhixiong Ye, Lex H.T. Van der Ploeg, David H. Weinberg, Tanya MacNeil, John Huber
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:3242-3247
مصطلحات موضوعية: Agonist, Pyrrolidines, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, Melanocortin receptor, Drug Discovery, medicine, Humans, Structure–activity relationship, Receptor, Telomerase, Molecular Biology, G protein-coupled receptor, Molecular Structure, digestive, oral, and skin physiology, Organic Chemistry, Stereoisomerism, chemistry, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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6
المؤلفون: Maria A. Bednarek, Ana Teran, Rui Tang, Tanya MacNeil, M. Angeles Cabello, Marta Maroto, Tung M. Fong
المصدر: Peptides. 28:1020-1028
مصطلحات موضوعية: Agonist, Physiology, Stereochemistry, medicine.drug_class, Peptide, CHO Cells, Biochemistry, Structure-Activity Relationship, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Cricetulus, Endocrinology, Melanocortin receptor, Cricetinae, Cyclic AMP, medicine, Animals, Humans, Amino Acid Sequence, Receptor, Pipecolic acid, chemistry.chemical_classification, Molecular Structure, Chemistry, Receptors, Melanocortin, Ligand binding assay, Receptors, Corticotropin, alpha-MSH, Melanocortin, Endogenous agonist, Protein Binding
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المؤلفون: Rui Tang, Tanya MacNeil, Ana Teran, Maria A. Bednarek, M. Angeles Cabello, Marta Maroto, Tung M. Fong
المصدر: Chemical Biology & Drug Design. 69:350-355
مصطلحات موضوعية: Agonist, medicine.drug_class, CHO Cells, Biology, Pharmacology, Biochemistry, chemistry.chemical_compound, Cricetulus, Melanocortin receptor, Cricetinae, Drug Discovery, medicine, Animals, Humans, ACTH receptor, Receptor, Receptors, Melanocortin, Organic Chemistry, Melanocortin 3 receptor, alpha-Melanocyte-stimulating hormone, Receptors, Corticotropin, chemistry, alpha-MSH, Molecular Medicine, Melanocortin, Melanocortin 1 receptor
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المؤلفون: Marta Maroto, Tung M. Fong, Maria A. Bednarek, M. Angeles Cabello, Ana Teran, Tanya MacNeil, Rui Tang
المصدر: Journal of Medicinal Chemistry. 50:2520-2526
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, CHO Cells, Binding, Competitive, Peptides, Cyclic, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Cricetulus, Melanocortin receptor, Cricetinae, Drug Discovery, Cyclic AMP, medicine, Animals, Humans, Melanocyte-Stimulating Hormones, Receptor, Melanocortins, chemistry.chemical_classification, Receptors, Melanocortin, Cyclic peptide, Melanocortin 3 receptor, alpha-Melanocyte-stimulating hormone, Receptors, Corticotropin, chemistry, Biochemistry, alpha-MSH, Molecular Medicine, Melanocortin
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المؤلفون: Christine Snedden, Mark T. Goulet, Tanya MacNeil, Matthew J. Wyvratt, David H. Weinberg, Thomas F. Walsh, Warner Daniel, Lex H.T. Van der Ploeg, Ricky D. Grisson, Rubana N. Kalyani, Rui Tang, Feroze Ujjainwalla
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:4023-4028
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Computational biology, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Inhibitory concentration 50, Structure–activity relationship, Receptor, Molecular Biology, Molecular Structure, integumentary system, Chemistry, digestive, oral, and skin physiology, Organic Chemistry, Biological activity, Melanocortin 3 receptor, Pyridazines, Drug Design, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Doreen E. Cashen, Constantin Tamvakopoulos, Qianping Peng, William J. Martin, David H. Weinberg, Charles Rosenblum, Arthur A. Patchett, Tanya MacNeil, Patrick G. Pollard, Zhixiong Ye, Raman K. Bakshi, Ralph A. Stearns, Rubana N. Kalyani, Palucki Brenda, Joseph M. Metzger, Alison M. Strack, Lex H.T. Van der Ploeg, D. Euan MacIntyre, Iyassu K. Sebhat, Aurawan Vongs, Airu S. Chen, Ravi P. Nargund, Liangqin Guo, Matthew J. Wyvratt, Randy R. Miller, Rui Tang, Howard Y. Chen, Khaled J. Barakat
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3501-3505
مصطلحات موضوعية: Male, Agonist, Quinuclidines, Time Factors, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Rodentia, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Rats, Sprague-Dawley, Eating, Structure-Activity Relationship, Piperidines, In vivo, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Aza Compounds, Bicyclic molecule, Chemistry, Penile Erection, digestive, oral, and skin physiology, Organic Chemistry, Small molecule, Rats, Microsomes, Liver, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding